Search Result "FXR"


Natural Products as Farnesoid X Receptor (FXR) Agonists: Their Interactions with FXR Ligand Binding Region

Journal: Mini-Reviews in Organic Chemistry
Volume: 13 Issue: 2 Year: 2016 Page: 97-108
Author(s): Hsiang-Ru Lin

Regulation of Apo E Expression by the Nuclear Receptors- LXRs and FXR

Journal: Current Medicinal Chemistry - Immunology, Endocrine & Metabolic Agents
Volume: 3 Issue: 3 Year: 2003 Page: 245-249
Author(s): Anne Perez, Eric J. Niesor

FXR, A Therapeutic Target for Bile Acid and Lipid Disorders

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 5 Issue: 8 Year: 2005 Page: 719-727
Author(s): Stefan Westin, Richard A. Heyman, Richard Martin

Research Article

Medicinal Chemistry and Pharmacological Effects of Farnesoid X Receptor (FXR) Antagonists

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 19 Year: 2014 Page: 2188-2205
Author(s): Christina Lamers,Manfred Schubert-Zsilavecz,Daniel Merk

Review Article

Farnesoid-X Receptor (FXR) as a Promising Pharmaceutical Target in Atherosclerosis

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 1 Year: 2017 Page: 1147-1157
Author(s): Demetrios Moris,Constantinos Giaginis,Gerasimos Tsourouflis,Stamatios Theocharis

Knocking on FXR's Door:The Hammerhead-Structure Series of FXRs Agonists - Amphiphilic Isoxazoles with Potent In Vitro and In Vivo Activities

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 19 Year: 2014 Page: 2143-2158
Author(s): Christian Gege,Olaf Kinzel,Christoph Steeneck,Andreas Schulz,Claus Kremoser

Development of FXR, PXR and CAR Agonists and Antagonists for Treatment of Liver Disorders

Journal: Current Topics in Medicinal Chemistry
Volume: 12 Issue: 6 Year: 2012 Page: 605-624
Author(s): Stefano Fiorucci, Angela Zampella, Eleonora Distrutti

Role of FXR in Regulating Bile Acid Homeostasis and Relevance for Human Diseases

Journal: Current Drug Targets - Immune, Endocrine & Metabolic Disorders
Volume: 5 Issue: 3 Year: 2005 Page: 289-303
Author(s): G. Rizzo, B. Renga, A. Mencarelli, R. Pellicciari, S. Fiorucci

Recent Advances in Non-Steroidal FXR Antagonists Development for Therapeutic Applications

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 19 Year: 2014 Page: 2175-2187
Author(s): Huang Huang,Yong Xu,Jin Zhu,Jian Li

Beyond Bile Acids: Targeting Farnesoid X Receptor (FXR) with Natural and Synthetic Ligands

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 19 Year: 2014 Page: 2129-2142
Author(s): Andrea Carotti,Maura Marinozzi,Chiara Custodi,Bruno Cerra,Roberto Pellicciari,Antimo Gioiello,Antonio Macchiarulo

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