Search Result "k-Ras"


Review Article

Recent Advances in Developing K-Ras Plasma Membrane Localization Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 2 Year: 2019 Page: 2114-2127
Author(s): Na Ye,Qingfeng Xu,Wanwan Li,Pingyuan Wang,Jia Zhou

K-Ras, Intestinal Homeostasis and Colon Cancer

Journal: Current Clinical Pharmacology
Volume: 10 Issue: 1 Year: 2015 Page: 73-81
Author(s): Sanjay Goel,Jie Huang,Lidija Klampfer

Across the Universe of K-Ras Mutations in Non-Small-Cell-Lung Cancer

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 24 Year: 2014 Page: 3933-3943
Author(s): Sheila Piva,Monica Ganzinelli,Marina Chiara Garassino,Elisa Caiola,Gabriella Farina,Massimo Broggini,Mirko Marabese

Modulation of k-Ras Signaling by Natural Products

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 14 Year: 2012 Page: 2273-2291
Author(s): S.B. Bharate, B. Singh, R.A. Vishwakarma

Mini-Review Article

Targeting K-Ras Mutations Show Promise Towards Ending Ras’s“Undruggable” Era

Journal: Protein & Peptide Letters
Volume: 29 Issue: 12 Year: 2022 Page: 1007-1015
Author(s): Paul D. Adams

Research Article

Polyisoprenylated Cysteinyl Amide Inhibitors Deplete K-Ras and Induce Caspase-dependent Apoptosis in Lung Cancer Cells

Journal: Current Cancer Drug Targets
Volume: 19 Issue: 1 Year: 2019 Page: 838-851
Author(s): Augustine T. Nkembo,Felix Amissah,Elizabeth Ntantie,Rosemary A. Poku,Olufisayo O. Salako,Offiong Francis Ikpatt,Nazarius S. Lamango

Research Article

Exploring the Lapse in Druggability: Sequence Analysis, Structural Dynamics and Binding Site Characterization of K-RasG12C Variant, a Feasible Oncotherapeutics Target

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2018 Page: 1540-1550
Author(s): Emmanuel A. Adeniji,Fisayo A. Olotu,Mahmoud E.S. Soliman

p53 Activation by Blocking Snail : A Novel Pharmacological Strategy for Cancer

Journal: Current Pharmaceutical Design
Volume: 17 Issue: 6 Year: 2011 Page: 610-617
Author(s): Sun-Hye Lee, Bum-Joon Park

Strategies for Overcoming Inherent and Acquired Resistance to EGFR Inhibitors by Targeting Downstream Effectors in the RAS/PI3K Pathway

Journal: Current Cancer Drug Targets
Volume: 10 Issue: 8 Year: 2010 Page: 824-833
Author(s): A. J. Weickhardt, N. C. Tebbutt, J. M. Mariadason

How to Target Activated Ras Proteins: Direct Inhibition vs. Induced Mislocalization

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 5 Year: 2016 Page: 358-369
Author(s): Ethan J. Brock,Kyungmin Ji,John J. Reiners,Raymond R. Mattingly

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