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A Comparison of Non-Human Primate Cytochrome P450 2D Members and the Implication in Drug Discovery

Journal: Current Drug Metabolism
Volume: 17 Issue: 6 Year: 2016 Page: 520-527
Author(s): Zhi-Xu He,Xiao-Wu Chen,Yinxue Yang,Shu-Feng Zhou

Integrated Acquisition of Analytical and Biopharmaceutical Screening Data for beta-Adrenergic-Drugs Employing Diversified Macrocycle Supported Potentiometric Detection in HPLC Systems

Journal: Current Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2002 Page: 1547-1566
Author(s): Grzegorz Bazylak, Luc J. Nagels

Human Liver Enzymes Responsible for Metabolic Elimination of Tyramine, a Vasopressor Agent from Daily Food

Journal: Drug Metabolism Letters
Volume: 5 Issue: 3 Year: 2011 Page: 216-219
Author(s): Toshiro Niwa, Norie Murayama, Hiromi Umeyama, Makiko Shimizu, Hiroshi Yamazaki

Comparison of P450 Enzymes Between Cynomolgus Monkeys and Humans: P450 Identities, Protein Contents, Kinetic Parameters, and Potential for Inhibitory Profiles

Journal: Current Drug Metabolism
Volume: 14 Issue: 2 Year: 2013 Page: 239-252
Author(s): Chie Emoto,Noriaki Yoda,Yasuhiro Uno,Kazuhide Iwasaki,Ken Umehara,Eiji Kashiyama,Hiroshi Yamazaki

Pharmacophore, QSAR, and Binding Mode Studies of Substrates of Human Cytochrome P450 2D6 (CYP2D6) Using Molecular Docking and Virtual Mutations and an Application to Chinese Herbal Medicine Screening

Journal: Current Pharmaceutical Biotechnology
Volume: 13 Issue: 9 Year: 2012 Page: 1640-1704
Author(s): Sui-Lin Mo,Wei-Feng Liu,Chun-Guang Li,Zhi-Wei Zhou,Hai-Bin Luo,Helen Chew,Jun Liang,Shu-Feng Zhou

Research Article

Assessment of Inhibition of Bovine Hepatic Cytochrome P450 by 43 Commercial Bovine Medicines Using a Combination of In Vitro Assays and Pharmacokinetic Data from the Literature

Journal: Drug Metabolism Letters
Volume: 13 Issue: 2 Year: 2019 Page: 123-131
Author(s): Steven X. Hu,Chase A. Mazur,Kenneth L. Feenstra

Comparison of Cytochrome P450 2D6 and Variants in Terms of Drug Oxidation Rates and Substrate Inhibition

Journal: Current Drug Metabolism
Volume: 12 Issue: 5 Year: 2011 Page: 412-435
Author(s): Toshiro Niwa, Norie Murayama, Hiroshi Yamazaki

Review Article

Benzofuran: A Key Heterocycle - Ring Closure And Beyond

Journal: Mini-Reviews in Organic Chemistry
Volume: 17 Issue: 3 Year: 2020 Page: 224-276
Author(s): Andiappan Lavanya,Kilambi Narasimhan,Vediappen Padmini

Research Article

Inhibition of Cytochrome P450 Enzyme and Drug-Drug Interaction Potential of AcidReducing Agents Used in Management of CDK Inhibitors for Breast Cancer Chemotherapy

Journal: Current Drug Metabolism
Volume: 23 Issue: 2 Year: 2022 Page: 137-149
Author(s): Prajakta Harish Patil,Puralae Channabasavaiah Jagadish,Gurupur Gautham Shenoy

Impact of Impurities on IC50 Values of P450 Inhibitors

Journal: Drug Metabolism Letters
Volume: 5 Issue: 3 Year: 2011 Page: 156-162
Author(s): Zeqi Huang

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