Search Result "agonism"


A Pharmacological Primer of Biased Agonism

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 11 Issue: 2 Year: 2011 Page: 92-98
Author(s): Bradley T. Andresen

Review Article

Aripiprazole, A Drug that Displays Partial Agonism and Functional Selectivity

Journal: Current Neuropharmacology
Volume: 15 Issue: 8 Year: 2017 Page: 1192-1207
Author(s): Erin W Tuplin,Matthew R Holahan

Intrinsic Activity at Adenosine A1 Receptors: Partial and Inverse Agonism

Journal: Current Pharmaceutical Design
Volume: 8 Issue: 2 Year: 2002 Page: 2333-2344
Author(s): Rianne A.F. de Ligt, Ad P. Ijzerman

Antipsychotic Medication: The Potential Role of 5-HT1A Receptor Agonism

Journal: Current Pharmaceutical Design
Volume: 16 Issue: 5 Year: 2010 Page: 516-521
Author(s): Andrew C. McCreary, Caitlin A. Jones

TRPV1 Activation is Not An All-Or-None Event: TRPV1 Partial Agonism/Antagonism and Its Regulatory Modulation

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 1 Year: 2011 Page: 2151-2158
Author(s): Peter M. Blumberg, Larry V. Pearce, Jeewoo Lee

Review Article

Biased Agonism as an Emerging Strategy in the Search for Better Opioid Analgesics

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 9 Year: 2020 Page: 1562-1575
Author(s): Justyna Piekielna-Ciesielska,Karol Wtorek,Anna Janecka

Biased Agonism at the Parathyroid Hormone Receptor: A Demonstration of Functional Selectivity in Bone Metabolism

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 9 Year: 2012 Page: 856-865
Author(s): B. N. Bohinc,D. Gesty-Palmer

Atypical antipsychotics and inverse agonism at 5-HT2 receptors

Journal: Current Pharmaceutical Design
Volume: 21 Issue: 26 Year: 2015 Page: 3732-3738
Author(s): Laura C. Sullivan,William P Clarke,Kelly A. Berg

Binding Modes and Pharmacophoric Features of Muscarinic Antagonism and β2 Agonism (MABA) Conjugates

Journal: Current Topics in Medicinal Chemistry
Volume: 13 Issue: 1 Year: 2013 Page: 1650-1655
Author(s): Srinivas Bandaru, M. Hema Prasad, A. Jyothy, Anuraj Nayarisseri, Mukesh Yadav

Novel Insights into Biased Agonism at G Protein-Coupled Receptors and their Potential for Drug Design

Journal: Current Pharmaceutical Design
Volume: 19 Issue: 2 Year: 2013 Page: 5156-5166
Author(s): Maria Marti-Solano, Ramon Guixa-Gonzalez, Ferran Sanz, Manuel Pastor, Jana Selent

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