Search Result "InhA"


Progress on the Discovery of Inhibitors of InhA, the FAS II Enoyl-ACP Reductase TB Drug Discovery Targeted on InhA

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 6 Year: 2016 Page: 539-546
Author(s): Yi Zhang,Longxiang Xie,Jianping Xie

Synthesis of an Indoloquinoxaline Derivative as Potential Inhibitor of InhA enzyme of Mycobacterium tuberculosis

Journal: Letters in Organic Chemistry
Volume: 12 Issue: 10 Year: 2015 Page: 727-733
Author(s): Asmae Zanzoul,Aurélien Chollet,Estefania Piedra-Arroni,Jean-Luc Stigliani,Vania Bernardes-Génisson,El Mokhtar Essassi,Geneviève Pratviel

Development of Modern InhA Inhibitors to Combat Drug Resistant Strains of Mycobacterium tuberculosis

Journal: Current Topics in Medicinal Chemistry
Volume: 7 Issue: 5 Year: 2007 Page: 489-498
Author(s): Peter J. Tonge, Caroline Kisker, Richard A. Slayden

Recent Progress in the Identification and Development of InhA Direct Inhibitors of Mycobacterium tuberculosis

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 10 Issue: 3 Year: 2010 Page: 182-193
Author(s): X.Y. Lu, Q.D. You, Y.D. Chen

Review Article

Structural Basis for Inhibition of Enoyl-[Acyl Carrier Protein] Reductase (InhA) from Mycobacterium tuberculosis

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 5 Year: 2020 Page: 745-759
Author(s): Maurício Boff de Ávila,Gabriela Bitencourt-Ferreira,Walter Filgueira de Azevedo

Research Article

Identifying the Structural Features of Diphenyl Ether Analogues for InhA Inhibition: A 2D and 3D QSAR Based Study

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 1 Year: 2020 Page: 31-47
Author(s): Ashutosh Prasad Tiwari,Varadaraj Bhat Giliyar,Gurypur Gautham Shenoy,Vandana Kalwaja Eshwara

Targeting InhA, the FASII Enoyl-ACP Reductase: SAR Studies on Novel Inhibitor Scaffolds

Journal: Current Topics in Medicinal Chemistry
Volume: 12 Issue: 7 Year: 2012 Page: 672-693
Author(s): Pan Pan,Peter J. Tonge

Mini-Review Article

Enoyl-Acyl Carrier Protein Reductase (INHA): A Remarkable Target to Exterminate Tuberculosis

Journal: Anti-Infective Agents
Volume: 19 Issue: 3 Year: 2021 Page: 252-266
Author(s): Surabhi Jain,Smriti Sharma,Dhrubo Jyoti Sen,Saurabh S Pandya

Research Article

In-Silico Analysis of Imidazo[2,1-b][1,3,4]thiadiazole Analogs as Putative Mycobacterium tuberculosis Enoyl Reductase Inhibitors

Journal: Current Drug Therapy
Volume: 12 Issue: 1 Year: 2017 Page: 46-63
Author(s): Preeti Wadhwa, Sourav Bagchi, Anuj Sharma

Mini-Review Article

Recent Discoveries of Nitrogen-Containing Heterocyclic Compounds asInhA Inhibitors against Mycobacterium tuberculosis: An Overview

Journal: Infectious Disorders - Drug Targets
Volume: 22 Issue: 8 Year: 2022 Page: 19-29
Author(s): Pratibha D. Gupta,Kalpana N. Tilekar,Neha M. Upadhyay

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