Search Result "3-d]pyrimidin-4(3H)-ones"


Research Article

Directed Search of Anti-inflammatory Agents among (3HQuinazoline- 4-ylidene)hydrazides of N-protected Amino acids and their Heterocyclization Products

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 19 Issue: 1 Year: 2020 Page: 60-71
Author(s): Yulya Martynenko,Oleksii Antypenko,Inna Nosulenko,Galina Berest,Sergii Kovalenko

Research Article

In Silico Bioactivity Prediction of Methoxime-3,4-dephostatin Derivatives on Human PTP1B: Search for Novel Antidiabetic Leads

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 5 Year: 2018 Page: 500-507
Author(s): Sabina B. Choudhury,Anupam D. Talukdar,Manabendra D. Choudhury,Monjur A. Laskar,Abhishek Chowdhury

Research Article

Synthesis and Herbicidal Evaluation of Aryloxyphenoxypropionate Derivatives Containing Purine Moiety

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 1 Year: 2018 Page: 15-20
Author(s): Jianjun Shi,Guihua Ren,Zhimeng Dai,Ningjie Wu,Jianquan Weng,Tianming Xu,Xinghai Liu,Chengxia Tan

Synthesis of 4-amino-5-cyano-2, 6-Disubstituted Pyrimidines as a Potential Antifilarial DNA Topoisomerase II Inhibitors

Journal: Medicinal Chemistry
Volume: 4 Issue: 6 Year: 2008 Page: 577-585
Author(s): Ashok Kumar, J. K. Saxena, Prem M.S. Chauhan

Research Article

Microwave-assisted Synthesis and Antifungal Activity of Novel 1,2,4- Triazole Thioether Derivatives Containing Pyrimidine Moiety

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 4 Year: 2018 Page: 347-352
Author(s): Meng Xu,Ya-Bo Zhu,Mei Wang,Ikhlas A. Khan,Xing-Hai Liu,Jian-Quan Weng

Research Article

Synthesis, Characterization and Antibacterial Activity of Some New 1,2,4- Triazole Schiff bases and 1,2,4-triazolo[3,4-b][1,3,4]thiadiazines

Journal: Letters in Organic Chemistry
Volume: 15 Issue: 7 Year: 2018 Page: 575-582
Author(s): Kooi-Mow Sim,Pei-Qie Chan,Xin-Lik Boo,Ker-Sin Heng,Kah-Whei Lye,Kah-Cheng Teo

Design, Synthesis and Bioactivities of Phenylamino-Pyrimidine Derivatives as Novel Protein Tyrosine Kinase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 7 Year: 2011 Page: 596-601
Author(s): Xinfu Hong, Xianzhao Kuang, Guohua Ding, Yilin Liu, Jinlin Liu, Yanjin Zhao, Shuxin Li

Research Article

Synthesis and Urease Inhibitory Activity of Some 5-Aminomethylene Barbituric/Thiobarbituric Acid Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 4 Year: 2018 Page: 428-436
Author(s): Mehdi Asadi,Mohammad Mahdavi,Shabnam Mahernia,Zahra Rezaei,Maliheh Safavi,Mina Saeedi,Massoud Amanlou

Synthesis of a Novel Heterocyclic System - Pyrimido[5,4:5,6]thiopyrano [2,3-b]indole

Journal: Letters in Organic Chemistry
Volume: 6 Issue: 7 Year: 2009 Page: 526-528
Author(s): Jurgis Sudzius, Sigitas Tumkevicius

Research Article

1, 2, 4-triazoles Clubbed Pyrimidine Compounds with Synthesis, Antimicrobial, Antituberculosis, Antimalarial, and Anti-protozoal Studies

Journal: Letters in Organic Chemistry
Volume: 18 Issue: 8 Year: 2021 Page: 617-624
Author(s): Navin B. Patel,Hetal I. Soni,Rahul B. Parmar,Manuel J. Chan-Bacab,Gildardo Rivera

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