Search Result "HTRF"


Research Article

Heterocyclization of Thiophenes Derived from Estrone Followed by Cytotoxic, HTRF Kinase and Pim-1 Kinase Evaluations

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2018 Page: 1711-1728
Author(s): Mahmoud A. Abdelaziz Mahmoud,Rafat Milad Mohareb,Mashari A. Al-Sharif

A High-Throughput Screening Assay for Determining Cellular Levels of Total Tau Protein

Journal: Current Alzheimer Research
Volume: 10 Issue: 7 Year: 2013 Page: 679-687
Author(s): Seameen J. Dehdashti,Wei Zheng,Joel R. Gever,Robert Wilhelm,Dac-Trung Nguyen,Gurusingham Sittampalam,John C. McKew,Christopher P. Austin,Stanley B. Prusiner

Research Article

Inhibition of EGFR Signaling by N-cyclohexyl-2-(1-(phenylsulfonyl)piperidin-4-yl) acetamide

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 11 Year: 2017 Page: 1500-1507
Author(s): Sensen Lin,Hang Li,Jun Yu,Luyong Zhang,Ming Yan,Hongyang Li,Xinxin Li,Shengtao Yuan,Li Sun

Review Article

Overview on Radiolabel-Free in vitro Assays for GPCRs

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2017 Page: 3-14
Author(s): Michela Buccioni,Claudia Santinelli,Piero Angeli,Diego Dal Ben,Catia Lambertucci,Ajiroghene Thomas,Rosaria Volpini,Gabriella Marucci

Research Article

Synthesis and Anti-Proliferative Evaluations of New Heterocyclic Derivatives Using 5,6,8,9-tetrahydropyrazolo[5,1-b]quinazolin-7(3H)-one Derivatives Derived from Cyclohexa-1,4-dione

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 21 Issue: 4 Year: 2021 Page: 408-426
Author(s): Mahmoud A.A. Mahmoud,Meshari A. Alsharif,Rafat M. Mohareb

Review Article

An Overview on Screening Methods for Lysine Specific Demethylase 1 (LSD1) Inhibitors

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 23 Year: 2017 Page: 2496-2504
Author(s): Yi-Chao Zheng,Jiao Chang,Ting Zhang,Feng-Zhi Suo,Xiao-Bing Chen,Ying Liu,Bing Zhao,Bin Yu,Hong-Min Liu

High Throughput Screening of β-Amyloid Secretion Inhibitors Using Homogenous Time-Resolved Fluorescence

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 7 Issue: 8 Year: 2004 Page: 745-756
Author(s): Hugo Albrecht, Peter Zbinden, Andrea Rizzi, Gino Villetti, Benedetta Riccardi, Paola Puccini, Silvia Catinella, Bruno P. Imbimbo

Current In Vitro Kinase Assay Technologies: The Quest for a Universal Format

Journal: Current Drug Discovery Technologies
Volume: 5 Issue: 1 Year: 2008 Page: 59-69
Author(s): Yong Jia, Christopher M. Quinn, Silvia Kwak, Robert V. Talanian

Review Article

Time-Resolved Fluorescence Resonance Energy Transfer [TR-FRET] Assays for Biochemical Processes

Journal: Current Pharmaceutical Biotechnology
Volume: 17 Issue: 1 Year: 2016 Page: 1222-1230
Author(s):

Fluorescent Agonists and Antagonists for Vasopressin/Oxytocin G Protein-Coupled Receptors: Usefulness in Ligand Screening Assays and Receptor Studies

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 996-1005
Author(s): B. Mouillac, M. Manning, T. Durroux

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