Drug Metabolism Letters

Editor-in-Chief

Zhiyang Zhao
Alliance Pharma
Malvern, PA
(USA)

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Volume:10   Issue: 3
Pp: 151-151
M. Kajbaf
DOI: 10.2174/187231281003160929160728



New Screening Criteria Setting on Evaluation of Cytochrome P450 Induction Using HepaRG Cells with Multiplex Branched DNA Technologies in Early Drug Discovery promotion: free to download

Volume:10   Issue: 3
Pp: 152-160
Akira Ogasawara, Nao Torimoto, Naoki Tsuda, Fumika Aohara, Rikiya Ohashi, Yasuhiro Yamada and Hideki Taniguchi
DOI: 10.2174/1872312810666160822110011




Intracellular Retention of Three Quinuclidine Derivatives in Caco-2 Permeation Experiments: Mechanisms and Impact on Estimating Permeability and Active Efflux Ratio promotion: free to download

Volume:10   Issue: 3
Pp: 161-171
Hong Jin, Sudarshan Kapadnis, Ting Chen, Dooyoung Lee, Andrew McRiner, Andrew Cook, Duane A. Burnett, Gerhard Koenig and Cuyue Tang
DOI: 10.2174/1872312810666160725123322




Application of a “Fit for Purpose” PBPK Model to Investigate the CYP3A4 Induction Potential of Enzalutamide promotion: free to download

Volume:10   Issue: 3
Pp: 172-179
Rangaraj Narayanan, Matthew Hoffmann, Gondi Kumar and Sekhar Surapaneni
DOI: 10.2174/1872312810666160729124745




An Investigation of Sodium Fusidate and Recombinant Cytochrome P450 Enzymes Inhibition In-Vitro promotion: free to download

Volume:10   Issue: 3
Pp: 180-186
John Mishriky, Jacqueline Balassone, Zenah Bashour, Simranjit Kaur, Vini Raman, Robel Getachew, Narin Osman, Daniel Guidone, Vincent Chan and Peter J. Little
DOI: 10.2174/1872312810666160607015045




Inhibition of Procarcinogen Activating Enzyme CYP1A2 Activity and Free Radical Formation by Caffeic Acid and its Amide Analogues promotion: free to download

Volume:10   Issue: 3
Pp: 187-194
Paitoon Narongchai, Kanokporn Niwatananun, Siripun Narongchai, Winthana Kusirisin and Churdsak Jaikang
DOI: 10.2174/1872312810666160608123113




The Uremic Toxin Indoxyl-3-Sulfate Induces CYP1A2 In Primary Human Hepatocytes promotion: free to download

Volume:10   Issue: 3
Pp: 195-199
Hong Liu, Rangaraj Narayanan, Matthew Hoffmann and Sekhar Surapaneni
DOI: 10.2174/1872312810666160719143703




Identification and Characterization of the Human Cytosolic Sulfotransferases Mediating the Sulfation of Clioquinol and Iodoquinol promotion: free to download

Volume:10   Issue: 3
Pp: 200-205
Akihiro Yamamoto, Maame Debrah-Pinamang, Nicholas J. DiModica, Katsuhisa Kurogi, Ali A. Naqvi, Ying Hui, Yoichi Sakakibara, Masahito Suiko and Ming-Cheh Liu
DOI: 10.2174/1872312810666160719142850




UHPLC Quantitation Method for New Thiazolidinedione LPSF/GQ-02 and In Vitro/In Vivo Kinetic Studies promotion: free to download

Volume:10   Issue: 3
Pp: 206-212
Carla Monalizi Vieira, Michel Leandro de Campos, Elias Carvalho Padilha, Marina Pitta, Ivan da Rocha Pitta, Maria do Carmo Alves de Lima and Rosângela Gonçalves Peccinini
DOI: 10.2174/1872312810666160725124554




CYP2B6 and OPRM1 Receptor Polymorphisms at Methadone Clinics And Novel OPRM1 Haplotypes: A Cross-Sectional Study promotion: free to download

Volume:10   Issue: 3
Pp: 213-218
Ahmad Abdulrahman AlMeman, Rusli Ismail and Markus Perola
DOI: 10.2174/1872312810666160810104040




Effect of Cardiovascular Injury on Catabolism of Adenosine and Adenosine 5-‘Triphosphate in Systemic Blood in a Freely Moving Rat Model In Vivo promotion: free to download

Volume:10   Issue: 3
Pp: 219-226
Pollen K. Yeung, Shyam S. Kolathuru and Remigius U. Agu
DOI: 10.2174/1872312810666160607013859