Letters in Drug Design & Discovery

Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

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Volume:9   Issue: 9
Pp: i-iv
Bentham Science Publishers
DOI: 10.2174/157018012803307923
Published on: 27 September, 2012

In Vitro and In Vivo Investigations into the Carbene Silver Acetate Anticancer Drug Candidate SBC1

Volume:9   Issue: 9
Pp: 815-822
Iduna Fichtner, Jindrich Cinatl, Martin Michaelis, Lara C. Sanders, Ralf Hilger, Breandan N. Kennedy, Alison L. Reynolds, Frauke Hackenberg, Grainne Lally, Susan J. Quinn, Ian McRae and Matthias Tacke
DOI: 10.2174/157018012803307987
Published on: 27 September, 2012

Synthesis and Anticancer Activity of 3a,4-dihydro-3H-indeno[1, 2-c]pyrazole-2-carboxamide Analogues

Volume:9   Issue: 9
Pp: 823-827
Mohamed Jawed Ahsan
DOI: 10.2174/157018012803307996
Published on: 27 September, 2012

Antibacterial Characterization of 1-benzoyl-4-arylthiosemicarbazides and the study of their structure-activity relationship

Volume:9   Issue: 9
Pp: 828-832
Edyta Kusmierz, Agata Siwek, Urszula Kosikowska, Anna Malm and Monika Wujec
DOI: 10.2174/157018012803307914
Published on: 27 September, 2012

Synthesis and Antibacterial Activity of Novel 11-O-Phenethylcarbamoylazithromycin Derivatives with 4"-elongated Side Chains

Volume:9   Issue: 9
Pp: 833-839
Mi Yan, Jichao Cao, Xin Li, Siti Ma, Yuanze Wang, Chao Cong and Shutao Ma
DOI: 10.2174/157018012803308003
Published on: 27 September, 2012

Synthesis and Antimicrobial Evaluation of Pyrazo-thiazoles

Volume:9   Issue: 9
Pp: 840-847
Harun Patel, Vinod Ugale, Amol Ingale and Sanjay Bari
DOI: 10.2174/157018012803307950
Published on: 27 September, 2012

The Synergistic Antibacterial Effects of Water Soluble N-succinyl-chitosan with Ceftriaxone against Escherichia coli

Volume:9   Issue: 9
Pp: 848-852
Zhihui Luo, Qingsheng Wu and Meng Zhang
DOI: 10.2174/157018012803307905
Published on: 27 September, 2012

Synthesis, Antibacterial and Antifungal Activities of Novel N,N’-bipyrazole Piperazine Derivatives

Volume:9   Issue: 9
Pp: 853-857
Smaail Radi, Yahya Toubi, Abdelkader Hakkou, Faiza Souna, Imane Himri and Mohammed Bouakka
DOI: 10.2174/157018012803307941
Published on: 27 September, 2012

2D-QSAR Studies of Tacrine Analogues for Acetylcholine Esterase (AChE) Inhibition using Multiple Linear Regression Analysis

Volume:9   Issue: 9
Pp: 858-866
Prabhakar S. Achanta, Rajasekhar Reddy Alavala, Umasankar Kulandaivelu, Shireesha Boyapati and Kundan Ingale
DOI: 10.2174/157018012803307978
Published on: 27 September, 2012

Design of Peptidomimetic Based DPP-IV Inhibitors, Devoid of CYP Liabilities

Volume:9   Issue: 9
Pp: 867-873
Pradip Jadav, Rajesh Bahekar, Shailesh R. Shah, Dipam Patel, Amit Joharapurkar, Kiran Shah, Shruti Bhardwaj, Kishan Patel, Kaushil Patel, Rajendra Chopade, Mubeen Shaikh, Kalapatapu V.V.M. Sairam and Mukul Jain
DOI: 10.2174/157018012803307932
Published on: 27 September, 2012

3D-QSAR Studies on Isocoumarin-based Urokinase-type Plasminogen Activator (uPA) Inhibitors Employing Linear and Non-linear Regression Analysis Methods

Volume:9   Issue: 9
Pp: 874-880
Bhoomendra A. Bhongade, Nikhil D. Amnerkar, Sirajunisa Talath, Kishore P. Bhusari and Andanappa K. Gadad
DOI: 10.2174/157018012803308012
Published on: 27 September, 2012

Sesquiterpene Lactones with Anti-Hepatitis C Virus Activity Using Molecular Descriptors

Volume:9   Issue: 9
Pp: 881-890
Michelle Rossini, Marcus Tullius Scotti, Mauro Vicentini Correia, Harold Hilarion Fokoue, Luciana Scotti, Francisco Jaime Bezerra Mendonca Junior, Marcelo Sobral da Silva and Vicente de Paulo Emerenciano
DOI: 10.2174/157018012803307969
Published on: 27 September, 2012