Letters in Drug Design & Discovery


Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo

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Volume: 9 Issue: 2, February

Graphical Abstracts

Volume:9   Issue: 2
Pp: i-iv

DOI: 10.2174/157018081120902000i
Published on: 01 March, 2012

In Vitro Antimycobacterial Activity of New 7-Chloroquinoline Derivatives

Volume:9   Issue: 2
Pp: 126-134
Juan Bueno, Fernando A. Rojas Ruiz, Santiago Villabona Estupinan and Vladimir V. Kouznetsov
DOI: 10.2174/157018012799079761
Published on: 01 March, 2012

Acyl Hydrazides: Potent Antioxidants

Volume:9   Issue: 2
Pp: 135-139
Khalid Mohammed Khan, Mubeen Rani, Nida Ambreen, Asma Ejaz, Shahnaz Perveen, Syed Moazzam Haider, Mohammad Iqbal Choudhary and Wolfgang Voelter
DOI: 10.2174/157018012799079798
Published on: 01 March, 2012

Design, Synthesis and Biological Evaluation of Hybrid Molecules Containing Conjugated Styryl Ketone and α-Bromoacryloyl Moieties

Volume:9   Issue: 2
Pp: 140-152
Romeo Romagnoli, Pier Giovanni Baraldi, Olga Cruz-Lopez, Maria Kimatrai Salvador, Delia Preti, Mojgan Aghazadeh Tabrizi, Jan Balzarini, Alessandro Canella, Enrica Fabbri and Roberto Gambari
DOI: 10.2174/157018012799079842
Published on: 01 March, 2012

QSAR Studies of Some Substituted 1,3-Diaryl Propenone Derivatives as Plasmodium falciparum Growth Inhibitors

Volume:9   Issue: 2
Pp: 153-162
Nitendra K. Sahu, Sanjaykumar B. Bari and D. V. Kohli
DOI: 10.2174/157018012799079644
Published on: 01 March, 2012

Design, Synthesis and In Vitro Antimalarial Evaluation of New Quinolinylhydrazone Derivatives

Volume:9   Issue: 2
Pp: 163-168
Le Thi Thuy, Hoang Xuan Tien, Vu Dinh Hoang and Tran Khac Vu
DOI: 10.2174/157018012799079815
Published on: 01 March, 2012

Docking Prediction for Luteolin Inhibiting TNF-α and NF-κB Pathway

Volume:9   Issue: 2
Pp: 169-176
Jui-Chiang Sun, S. T. Wua, Kuei-Jen Lee and Yu-Ming Sun
DOI: 10.2174/157018012799079707
Published on: 01 March, 2012

QSAR Study of SMMC7721 Inhibitors from Diterpenoids with a Dehydroabietyl Skeleton

Volume:9   Issue: 2
Pp: 177-184
Xiaoping Rao, Zhanqian Song, Zongde Wang, Yong Wu, Shibin Shang, Ling He and Qin Huang
DOI: 10.2174/157018012799079680
Published on: 01 March, 2012

Elaboration of New Anti-Inflammatory Agents Using Pharmacophore Based 3D QSAR of 4, 5-Diaryl Imidazoline as P2X7 Receptor Antagonists

Volume:9   Issue: 2
Pp: 185-198
Nisha Mehta, Sukhvir Chand, Malkeet Singh Bahia and Om Silakari
DOI: 10.2174/157018012799079860
Published on: 01 March, 2012

Novel 3-(1-(2-(2,7a-dihydrobenzo[d]thiazol-2-ylthio)acetyl)-5-substitutedphenyl-4,5-dihydro-1H-pyrazol-3-yl)-Coumarins: Synthesis and Anticancer Activity

Volume:9   Issue: 2
Pp: 199-203
Xian-Hai Lv, Xiu-Li Zhang, Xin-Hua Liu and Lei Shi
DOI: 10.2174/157018012799079743
Published on: 01 March, 2012

Novel 1,2,4-Triazolo[3,4-b]-1,3,4-thiadiazole Derivatives as Dual Analgesic/Anti-inflammatory and Antimicrobial Agents

Volume:9   Issue: 2
Pp: 204-212
Birsen Tozkoparan, Sevim Peri Aytac, Sule Gursoy, Selami Gunal and Goknur Aktay
DOI: 10.2174/157018012799079626
Published on: 01 March, 2012

Fat-Soluble Vitamins Release Based on Clinoptilolite Zeolite as an Oral Drug Delivery System

Volume:9   Issue: 2
Pp: 213-217
Mehdi Rahimi, Hamid Mobedi, Aliasghar Behnamghader, Alireza Nateghi Baygi, Houri Mivehchi and Esmaeil Biazar
DOI: 10.2174/157018012799079833
Published on: 01 March, 2012

Synthesis and Computational Studies on Aryloxypropyl Piperazine Derivatives as Potential Atypical Antipsychotic Agents

Volume:9   Issue: 2
Pp: 218-224
Alka Bali, Abhishek Bhalla, Suman Bala and Rajesh Kumar
DOI: 10.2174/157018012799079725
Published on: 01 March, 2012