Letters in Drug Design & Discovery


Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo

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Volume: 8 Issue: 9, November

Graphical Abstracts

Volume:8   Issue: 9
Pp: i-v

DOI: 10.2174/157018011797200885
Published on: 01 March, 2012

Rapid and Facile Synthesis of N-Benzenesulfonyl Derivatives of Heterocycles and their Antimicrobial Properties

Volume:8   Issue: 9
Pp: 778-791
Romina J. Pagliero, Reesa Mercado, Vance McCracken, Maria R. Mazzieri and Marcelo J. Nieto
DOI: 10.2174/157018011797200803
Published on: 01 March, 2012

Isonicotinic Acid Hydrazide Derivatives: Synthesis, Antimycobacterial, Antiviral, Antimicrobial Activity and QSAR Studies

Volume:8   Issue: 9
Pp: 792-810
Vikramjeet Judge, Balasubramanian Narasimhan, Munish Ahuja, Dharmarajan Sriram and Perumal Yogeeswar
DOI: 10.2174/157018011797200795
Published on: 01 March, 2012

Synthesis, Antibacterial and Antifungal Activities of Some Carbazole Dithiocarbamate Derivatives

Volume:8   Issue: 9
Pp: 811-815
Ahmet Cagri Karaburun, Zafer Asim Kaplancikli, Nalan Gundogdu-Karaburun and Fatih Demirci
DOI: 10.2174/157018011797200858
Published on: 01 March, 2012

Synthesis and Biological Evaluation of Andrographolide Derivatives as Potent Antibacterial Agents

Volume:8   Issue: 9
Pp: 816-821
Chunlei Tang, Wenjie Zhang, Xinyang Wang, Bin Wang, Xiaoyun Zhu, Dandan Huang, Xiaoyong Du, Hai Qian, Wenlong Huang and Jing Li
DOI: 10.2174/157018011797200740
Published on: 01 March, 2012

Synthesis and In Vitro Antiviral Evaluation of Novel 1-Arylpyrazoles and Their N- and S-Glycosides

Volume:8   Issue: 9
Pp: 822-829
Emad M. El-Telbani, Sara M. Ghanem, Farrag A. El-Essawy and Aly F. El-Sayed
DOI: 10.2174/1570180811108090822
Published on: 01 March, 2012

Synthesis of Some Benzothiazole Based Piperazine-Dithiocarbamate Derivatives and Evaluation of Their Anticancer Activities

Volume:8   Issue: 9
Pp: 830-837
Gulhan Turan-Zitouni, Yusuf Ozkay, Ahmet Ozdemir, Zafer Asim Kaplancikli and Mehlika Dilek Altintop
DOI: 10.2174/157018011797200786
Published on: 01 March, 2012

Thiazole Containing Nitrogen Mustards: Synthesis, Structural Evaluation, Cytotoxicity and DNA Binding Studies

Volume:8   Issue: 9
Pp: 838-842
Nulgulmnalli Manjunathiah Raghavendra, Surampudi Renuka, Sayan Dutta Gupta and Pingili Divya
DOI: 10.2174/157018011797200830
Published on: 01 March, 2012

Synthesis and In Vitro Antitumor Activity of Novel Fluorine Containing Pyrazoles and Pyrazolines

Volume:8   Issue: 9
Pp: 843-849
Ashish Sharma, Tabreskhan Pathan, Rhea Mohan and C. S. Ramaa
DOI: 10.2174/157018011797200812
Published on: 01 March, 2012

Use of Physicochemical and Topological Parameters in Estimating Anti-Cancer Activity of Benzothiazole Derivatives

Volume:8   Issue: 9
Pp: 850-856
Deepali Gupta, Basheerulla Shaik, Jyoti Singh, Neelu Singh and Vijay K. Agrawal
DOI: 10.2174/157018011797200759
Published on: 01 March, 2012

Cytotoxicity Study on Some Synthetic Aromatic Esters of 4-Demethyl-4-deoxypodophyllotoxin

Volume:8   Issue: 9
Pp: 857-860
Juan-Juan Wang, Hong-Jin Han, Guang-Zhi Zeng, Hui Xu and Ning-Hua Tan
DOI: 10.2174/157018011797200849
Published on: 01 March, 2012

Doxorubicin Sensitizes the Non-Small Cell Lung Cancer Cells to Tumor Necrosis Factor-Related Apoptosis-Inducing Ligand-Mediated (TRAIL) Apoptosis In Vitro but not In Vivo

Volume:8   Issue: 9
Pp: 861-867
Li Fan, Liangran Guo, Jinfeng Ren, Yulong Ren, Zhiqing Pang and Xinguo Jiang
DOI: 10.2174/157018011797200867
Published on: 01 March, 2012

A QSAR Analysis of Coumarin Derivatives as TNF-α Inhibitor - A Rational Approach to Anticancer Drug Design

Volume:8   Issue: 9
Pp: 868-876
Malleshappa N. Noolvi, Harun M. Patel and Tarandeep Kaur
DOI: 10.2174/157018011797200768
Published on: 01 March, 2012

Synthesis, Crystal Structure and Biological Evaluation of 4, 5, 6, 7-tetrahydropravastatin as HMG-CoA Reductase Inhibitor

Volume:8   Issue: 9
Pp: 884-888
Jing Li, Huan Li and Lei Zhang
DOI: 10.2174/157018011797200876
Published on: 01 March, 2012