Letters in Drug Design & Discovery

Editor-in-Chief

Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo
(Italy)

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Volume: 8 Issue: 5, June

Graphical Abstracts

Volume:8   Issue: 5
Pp: i-iv

DOI: 10.2174/157018011795514177
Published on: 01 March, 2012

Novel RGD Peptidomimetics Embedding 1,2,3-Triazole as Central Scaffold; Synthesis and αvβ3 Integrin Affinity

Volume:8   Issue: 5
Pp: 401-405
Ming Hong Ni, Emiliano Esposito, Massimo Castorina and Alma Dal Pozzo
DOI: 10.2174/157018011795514258
Published on: 01 March, 2012

Synthesis and Biological Evaluation of Spiro-δ-lactones as Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 2 (17β-HSD2) open access plus

Volume:8   Issue: 5
Pp: 406-421
Kuiying Xu, Marie Wetzel, Rolf W. Hartmann and Sandrine Marchais-Oberwinkler
DOI: 10.2174/157018011795514230
Published on: 01 March, 2012

Quantitative Structure Activity Relationship Studies on a Novel Indolediones as Long Chain Fatty Acid Elongase 6 (ELOVL6) Inhibitors

Volume:8   Issue: 5
Pp: 422-429
Junxia Zheng, Zhiwei Wu, Mibei Dai, Zhihui Xu, Xiaomei Li, Shanshan Zhu, Chuyun Lin, Peijian Hu, Luo Zhang, Huarong Huang, Suqing Zhao, Kun Zhang and Pinghua Sun
DOI: 10.2174/157018011795514168
Published on: 01 March, 2012

CoMFA and CoMSIA Analyses of Highly Selective Pipecolic Acid Based TNF-α Converting Enzyme (TACE) Inhibitors Using Docked Conformations for Molecular Alignment

Volume:8   Issue: 5
Pp: 430-439
Malkeet Singh Bahia, Sukhvir Chand, Shravan Kumar Gunda, Shwetha Reddy Gade, Saikh Mahmood and Om Silakari
DOI: 10.2174/157018011795514195
Published on: 01 March, 2012

Homology Modeling of α-Glucosidase and its Interactions with Andrograpolide Derivatives

Volume:8   Issue: 5
Pp: 440-451
Jun Xu, Yijing Lu, Weizai Shen, Haibin Luo, Sichao Huang, Jiaolin Bao, Shaohui Cai and Yuqiang Wang
DOI: 10.2174/157018011795514203
Published on: 01 March, 2012

Synthesis, Cytotoxic and Phytotoxic Effects of Some New N4-Aryl Substituted Isatin-3-thiosemicarbazones

Volume:8   Issue: 5
Pp: 452-458
Humayun Pervez, Muhammad Ramzan, Muhammad Yaqub and Khalid Mohammed Khan
DOI: 10.2174/157018011795514159
Published on: 01 March, 2012

Synthesis and Antimicrobial Activity of 8-Alkylpalmatine Derivatives

Volume:8   Issue: 5
Pp: 464-468
Teng-Wen Ma, Xiao-Li Ye, Xue-Gang Li, Bao-Shun Zhang, Xiao-Fei Jiang and Zu Chen
DOI: 10.2174/157018011795514186
Published on: 01 March, 2012

Modern Methods & Web Resources in Drug Design & Discovery

Volume:8   Issue: 5
Pp: 469-490
Feroz Khan, Dharmendra Kumar Yadav, Anupam Maurya and Santosh Kumar Srivastava
DOI: 10.2174/157018011795514249
Published on: 01 March, 2012

Evaluation of N-(2-Thienylidene)amines, N-(2-Hydroxybenzylidene)amines and 3-Iminoindolin-2-ones as Antileishmanial Agents

Volume:8   Issue: 5
Pp: 491-495
Yasser M.S.A. Al-Kahraman, Girija S. Singh and Masoom Yasinzai
DOI: 10.2174/157018011795514221
Published on: 01 March, 2012