Letters in Drug Design & Discovery


Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo

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Volume: 8 Issue: 3, March

Graphical Abstracts

Volume:8   Issue: 3
Pp: i-iv

DOI: 10.2174/157018011794578268
Published on: 01 March, 2012

Alteration of Warfarins Pharmacologic Properties in Clathrates with Glycyrrhizic Acid and Arabinogalactan

Volume:8   Issue: 3
Pp: 201-204
Tatjana G. Tolstikov, Mikhail V. Khvostov, Galina I. Lifshits, Alexander V. Dushkin and Elezaveta S. Meteleva
DOI: 10.2174/157018011794578222
Published on: 01 March, 2012

Novel Aglycones of Steroidal Glycoalkaloids as Potent Tyrosine Kinase Inhibitors: Role in VEGF and EGF Receptors Targeted Angiogenesis

Volume:8   Issue: 3
Pp: 205-215
Salman Akhtar, Othman A. Al-Sagair and Jamal M. Arif
DOI: 10.2174/157018011794578187
Published on: 01 March, 2012

Molecular Insight into the Inhibitory Mechanism of Galangin Towards Human Cytochrome P450 1A2. A Modeling Study

Volume:8   Issue: 3
Pp: 216-222
Yunyun Chen, Guo-Wen Chen and Hai-Bin Luo
DOI: 10.2174/157018011794578150
Published on: 01 March, 2012

Prediction of Specificity and Cross-Reactivity of Kinase Inhibitors

Volume:8   Issue: 3
Pp: 223-228
Nitish Kumar Mishra and Gajendra P.S. Raghava
DOI: 10.2174/157018011794578204
Published on: 01 March, 2012

3D-QSAR and Docking Studies on Pyrrolopyrimidine Derivatives as LIM-Kinase 2 Inhibitors

Volume:8   Issue: 3
Pp: 229-240
Jun-Rong Sun, Ping Lan, Ping-Hua Sun and Wei-Min Chen
DOI: 10.2174/157018011794578178
Published on: 01 March, 2012

Synthesis and Biological Evaluation of a Range of Thiosemicarbazone - Based Compounds as Potential Inhibitors of Estrone Sulfatase (ES)

Volume:8   Issue: 3
Pp: 241-245
Amit Kumar, Sukriti Singh, Hadi Bordbar, Timothy Cartledge and Sabbir Ahmed
DOI: 10.2174/157018011794578231
Published on: 01 March, 2012

Targeting Catechol-O-Methyl Transferase (COMT) Inhibitors for Schizophrenia:An Approach to Target Validation and Rational Drug Design

Volume:8   Issue: 3
Pp: 246-252
Deepak Purushotham, Chaiti Ganguly and Chiranjib Chakraborty
DOI: 10.2174/157018011794578277
Published on: 01 March, 2012

In Silico Studies of (2E,5E)-2,5-bis(3-methoxy-4-hydroxy-benzylidene) Cyclopentanone on Proteins AChE and BChE Involved in Alzheimers disease and Ameliorative Effects on Paraquat Induced Oxidative Stress Markers in Drosophila melanogaster

Volume:8   Issue: 3
Pp: 260-267
Balladka Kunhanna Sarojini, Chenna Govindaraju Darshan Raj, Modalkoppalu Kyathegowda Ramakrishna, Saraf R Ramesh, Basavapattana Rudresh Bharath and Hanumanthappa Manjunatha
DOI: 10.2174/157018011794578213
Published on: 01 March, 2012

Microwave-Assisted Synthesis and Evaluation of Substituted Aryl Propyl Acridone-4-Carboxamides as Potential Chemosensitizing Agents for Cancer

Volume:8   Issue: 3
Pp: 268-275
Vinaykumar S. Velingkar and Vikrant D. Dandekar
DOI: 10.2174/157018011794578169
Published on: 01 March, 2012

Synthesis, Characterization of Some New Five Membered Heterocycles Based on Imidazole Moiety and their Applications on Therapeutics

Volume:8   Issue: 3
Pp: 276-283
V. S.V. Satyanarayana, A. Sivakumar and Asit Ranjan Ghosh
DOI: 10.2174/157018011794578196
Published on: 01 March, 2012

Gallic Acid-Phospholipid Complex: Drug Incorporation and Physicochemical Characterization

Volume:8   Issue: 3
Pp: 284-291
Devendra Singh, Mohan Singh Maniyari Rawat, Ajay Semalty and Mona Semalty
DOI: 10.2174/157018011794578240
Published on: 01 March, 2012

Retraction Notice: Solubilization and Amorphization of Non Steroidal Anti-Inflammatory Drug with Low Molecular Weight Chitosan for a New Guar-Based Colon Delivery Formulation free to download

Volume:8   Issue: 3
Pp: 292-301
Kadria A. Elkhodairy, Nahla S. Barakat and Fars K. Alanazi
DOI: 10.2174/157018011794578141
Published on: 01 March, 2012