Letters in Drug Design & Discovery

Editor-in-Chief

Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo
(Italy)

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Volume: 6 Issue: 1, January

Synthesis of 4-substituted-3-hydroxy-5-oxo-10-oxa-4-azatricyclo[5.2.1]dec- 3-yl Acetic Acid Ethyl Esters as Norcantharidin Analogues

Volume:6   Issue: 1
Pp: 1-7
Benjamin Sauer, Jayne Gilbert, Jennette A. Sakoff and Adam McCluskey
DOI: 10.2174/157018009787158535
Published on: 01 March, 2012

Involvement of Serotonin in the Acute Dependence Produced by μ, and K Opioid Agonists

Volume:6   Issue: 1
Pp: 8-12
Anna Capasso
DOI: 10.2174/157018009787158562
Published on: 01 March, 2012

Buprenorphine and Methadone Maintenance Treatment - Sexual Behaviour and Dysfunction Prevalence

Volume:6   Issue: 1
Pp: 13-13
S. M. Giacomuzzi, A. Khreis, Y. Riemer, K. Garber and M. Ertl
DOI: 10.2174/157018009787158580
Published on: 01 March, 2012

Computer-Aided Drug Design for Cancer-Causing H-Ras p21 Mutant Protein

Volume:6   Issue: 1
Pp: 14-20
Mannu Jayakanthan, Gulshan Wadhwa, Thangavel Madhan Mohan, Loganathan Arul, Ponnusamy Balasubramanian and Durai Sundar
DOI: 10.2174/157018009787158526
Published on: 01 March, 2012

Synthesis, Antibacterial Activity of 2,4-Disubstituted Oxazoles and Thiazoles as Bioisosteres

Volume:6   Issue: 1
Pp: 21-28
Mohamed Kaspady, Venugopala Katharigatta Narayanaswamy, Mohana Raju and Gopal Krishna Rao
DOI: 10.2174/157018009787158481
Published on: 01 March, 2012

Identification of GCP II Inhibitors Based on 4-Arylmethyl-3-(4- carboxyphenyl)-5-hydroxyisoxazole Scaffold

Volume:6   Issue: 1
Pp: 29-32
M. Teus, A. Jirgensons, M. Dambrova, R. Mezhapuke, C. G. Parsons and W. Danysz
DOI: 10.2174/157018009787158544
Published on: 01 March, 2012

Structural and Morphological Studies of Cationic Liposomes-DNA Complexes

Volume:6   Issue: 1
Pp: 33-37
Yan Sun, Itziar Migueliz, Gemma Navarro and Conchita Tros de Ilarduya
DOI: 10.2174/157018009787158571
Published on: 01 March, 2012

Pharmacophore Searching of Benzofuran Derivatives for Selective CYP19 Aromatase Inhibition

Volume:6   Issue: 1
Pp: 38-45
Shuchi Nagar, Md Ataul Islam, Suvadra Das, Arup Mukherjee and Achintya Saha
DOI: 10.2174/157018009787158607
Published on: 01 March, 2012

Evaluation of In-Vivo Anti-Implantation and In-Vitro Anti-Proliferative Activities of Substituted 3-phenyl-4-phenylvinyl Benzopyranone Derivatives

Volume:6   Issue: 1
Pp: 46-50
Atul Gupta, Ramesh Sharma, Anil Kumar Balapure, Govind Keshri, M. M. Singh and Suprabhat Ray
DOI: 10.2174/157018009787158508
Published on: 01 March, 2012

Synthesis and Antitumor Activity of Novel 4-Chloro-3-Arylmaleimide Derivatives

Volume:6   Issue: 1
Pp: 51-55
Guiqing Xu, Qiaojun He, Bo Yang and Yongzhou Hu
DOI: 10.2174/157018009787158490
Published on: 01 March, 2012

DNA Binders: 1. Evaluation of DNA-Interactive Ability, Design, and Synthesis of Novel Intercalating Agents

Volume:6   Issue: 1
Pp: 56-62
Mario Sechi, Marco Derudas, Roberto Dallocchio, Alessandro Dessì, Alessia Cosseddu and Giuseppe Paglietti
DOI: 10.2174/157018009787158472
Published on: 01 March, 2012

Susceptibility of Staphylococcus spp. Isolated from Milk of Goats with Mastitis to Antibiotics and Green Propolis Extracts

Volume:6   Issue: 1
Pp: 63-68
T. M. Santos Neto, R. A. Mota, L. B.G. Silva, D. A. Viana, J. L. Lima-Filho, L. A. Sarubbo, A. Converti and A. L.F. Porto
DOI: 10.2174/157018009787158599
Published on: 01 March, 2012

Synthesis and Antibacterial and Antifungal Activity of 5-Substituted Imidazolones

Volume:6   Issue: 1
Pp: 69-77
Khalid Mohammed Khan, Uzma Rasool Mughal, Sadia Khan, Saira Khan, Shahnaz Perveen and M. Iqbal Choudhary
DOI: 10.2174/157018009787158553
Published on: 01 March, 2012

Solution-Phase Parallel Synthesis of N-Arylisoquinuclidines

Volume:6   Issue: 1
Pp: 78-81
Ronald F. Borne, Mark S. Levi, M. O. Faruk Khan and Norman H. Wilson
DOI: 10.2174/157018009787158517
Published on: 01 March, 2012

Development of an Economical, Single Step Synthesis of FAZA, a Clinical Hypoxia Marker, and Potential Synthons to Prepare its Positional Analogs

Volume:6   Issue: 1
Pp: 82-85
P. Kumar, S. Emami, A. J.B. McEwan and L. I. Wiebe
DOI: 10.2174/157018009787158616
Published on: 01 March, 2012