Letters in Drug Design & Discovery


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

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Synthesis, DNA-Binding Ability and Biological Activity of C8 Linked G1 Dendrimer-Pyrrolobenzodiazepine Conjugates as Anticancer Agents

Volume:5   Issue: 7
Pp: 424-432
Ahmed Kamal, G. Balakishan, Rajender, K. Sreekanth, D. Rajasekhar Reddy, M. Kashi Reddy, Subrata Sen, Nisha Kurian, Aarti S. Juvekar and Surekha M. Zingde
DOI: 10.2174/157018008785909859

Sesquiterpene Lactones and their Anti-Tumor Activity from the Flowers of Inula Britannica

Volume:5   Issue: 7
Pp: 433-436
Jin-Long Qi, Yan Fu, Xiao-Wei Shi, Yi-Bing Wu, Yun-Zhi Wang, Di-Qun Zhang and Qing-Wen Shi
DOI: 10.2174/157018008785909813

3D-QSAR Analysis on N-Phenylacetanoyl-L-Homoserine Lactones as Inhibitors of Bacterial Quorum Sensing via CoMFA Approach

Volume:5   Issue: 7
Pp: 449-453
Ping-Hua Sun, Zhao-Qi Yang, Wei-Min Chen, Qian Liu and Xin-Sheng Yao
DOI: 10.2174/157018008785909831

Synthesis and In Vitro Antiproliferative Activity of Diphenyl(piperidin-4- yl)thioamide Methanol Derivatives

Volume:5   Issue: 7
Pp: 454-461
Salekoppal Boregowda Benaka Prasad, Mallappanahally Kambappa Vinaya, Channapille Koppal Siddegowda Ananda Kumar, Sanjay Swarup and Kanchugarakoppal Subbegowda Rangappa
DOI: 10.2174/157018008785909804

Release of a Poorly Soluble Drug from Cross-Linked β-Cyclodextrin-Based Polymer Pellets Prepared via Extrusion/Spheronisation

Volume:5   Issue: 7
Pp: 462-470
Pierre Bon, Samer Joudieh, Malika Lahiani-Skiba, Frederic Bounoure, Pierre Dechelotte and Mohamed Skiba
DOI: 10.2174/157018008785909822

96-Well Plate Surface Tension Measurements for Fast Determination of Drug Solubility

Volume:5   Issue: 7
Pp: 471-476
Tiina Heikkila, Leena Peltonen, Saila Taskinen, Timo Laaksonen and Jouni Hirvonen
DOI: 10.2174/157018008785909840