Letters in Drug Design & Discovery


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

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New Synthetic Chalcones: Cytotoxic Mannich Bases of 6-(4-Chlorocinnamoyl)-2(3H)-benzoxazolone

Volume:5   Issue: 6
Pp: 358-361
O. Petrov, Y. Ivanova, G. Momekov and V. Kalcheva
DOI: 10.2174/157018008785777342

Synthesis and Anticancer Evaluation of some Newer 2, 5-Disubstituted-1,3, 4-Oxadiazole Analogues

Volume:5   Issue: 6
Pp: 364-368
Rakesh R. Somani, Prabhakar Y. Shirodkar and Vilasrao J. Kadam
DOI: 10.2174/157018008785777360

A Preliminary Assessment of the Structure-Activity Relationship of Benzimidazole-Based Anti-Proliferative Agents

Volume:5   Issue: 6
Pp: 369-376
Leyte L. Winfield, Dayle M. Smith, Kalani Halemano and Carmine S. Leggett
DOI: 10.2174/157018008785777324

Three-Dimensional Quantitative Structure-Activity Relationships for a Large Series of Potent Antitubercular Agents

Volume:5   Issue: 6
Pp: 377-387
Carolina Horta Andrade, Livia de Barros Salum, Kerly Fernanda Mesquita Pasqualoto, Elizabeth Igne Ferreira and Adriano Defini Andricopulo
DOI: 10.2174/157018008785777289

Antimicrobial Activities of 7-Aminosterol Squalamine Analogues

Volume:5   Issue: 6
Pp: 388-393
Celine Loncle, Chanaz Salmi, Nicolas Vidal, Yves Letourneux and Jean Michel Brunel
DOI: 10.2174/157018008785777306

Octanol Water Partition Coefficient Determination for Model Steroids Using an HPLC Method

Volume:5   Issue: 6
Pp: 394-400
Sara Zargar Shoshtari, Jingyuan Wen and Raid. G. Alany
DOI: 10.2174/157018008785777333

Urease and α-Chymotrypsin Inhibitory Effects of Selected Urea Derivatives

Volume:5   Issue: 6
Pp: 401-405
Shahnaz Perveen, Khalid Mohammed Khan, Muhammad Arif Lodhi, Muhammad Iqbal Choudhary, Atta-ur-Rahman and Wolfgang Voelter
DOI: 10.2174/157018008785777315

Nimesulide Apparent Solubility Enhancement with Natural Cyclodextrins and their Polymers

Volume:5   Issue: 6
Pp: 406-415
S. Joudieh, M. Lahiani-Skiba, P. Bon, O. Ba, J. M. Le Breton and M. Skiba
DOI: 10.2174/157018008785777270

Facile Conversion of FP to TR-FRET Assays using Terbium Chelates:Nuclear Receptor Competitive Binding Assays as Examples

Volume:5   Issue: 6
Pp: 416-422
Kurt W. Vogel, Bryan D. Marks, Kevin R. Kupcho, Kevin L. Vedvik and Tina M. Hallis
DOI: 10.2174/157018008785777261

Erratum promotion: free to download

Volume:5   Issue: 6
Pp: 423-423

DOI: 10.2174/157018008785777351