Letters in Drug Design & Discovery

Editor-in-Chief

Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo
(Italy)

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Volume: 5 Issue: 3, April

Microwaves-Assisted Syntheses of Imidazolylbenzamides and their Antioxidant Activities

Volume:5   Issue: 3
Pp: 152-157
Khalid Mohammed Khan, Uzma Rasool Mughal, Iman Omar and M. Iqbal Choudhary
DOI: 10.2174/157018008784083974
Published on: 01 March, 2012

Natural Products Biological Screening and Ligand-Based Virtual Screening for the Discovery of New Antileishmanial Agents

Volume:5   Issue: 3
Pp: 158-161
Fernanda C. Costa, Ricardo P. Nicoluci, Marcio Silva, Waldireny C. Rocha, Paulo C. Vieira, Glaucius Oliva, Otavio H. Thiemann and Adriano D. Andricopulo
DOI: 10.2174/157018008784083956
Published on: 01 March, 2012

Determination of Molecular Properties Effectuating the Growth Inhibition of Mycobacterium Tuberculosis by Various Small Molecule Hydrazides

Volume:5   Issue: 3
Pp: 162-168
Ronald Bartzatt, Suat L.G. Cirillo and Jeffrey D. Cirillo
DOI: 10.2174/157018008784083929
Published on: 01 March, 2012

New 3-Aminosteroid Derivatives as a New Family of Topical Antibacterial Agents Active against Methicillin-Resistant Staphylococcus aureus (MRSA)

Volume:5   Issue: 3
Pp: 169-172
Chanaz Salmi, Celine Loncle, Nicolas Vidal, Michele Laget, Yves Letourneux and Jean Michel Brunel
DOI: 10.2174/157018008784084018
Published on: 01 March, 2012

A QSAR Study on some Series of ATP-Sensitive Potassium Channel Openers

Volume:5   Issue: 3
Pp: 173-177
V. S.A. Kumar Satuluri and S. P. Gupta
DOI: 10.2174/157018008784084027
Published on: 01 March, 2012

Synthesis and Antimalarial Activity of Novel Hydroxyethylamines,Potential Aspartyl Protease Inhibitors

Volume:5   Issue: 3
Pp: 178-181
Wilson Cunico, Maria de Lourdes G. Ferreira, Thais G. Ferreira, Carmen Penido, Maria G.M.O. Henriques, Luisa G. Krettli, Fernando P. Varotti and Antoniana U. Krettli
DOI: 10.2174/157018008784083938
Published on: 01 March, 2012

Estrogen Receptor: Structural Differences and Potential Implications on Selectivity Examined by the GRID/CPCA Approach

Volume:5   Issue: 3
Pp: 182-192
I. R.A. de Menezes, A. Leitao and C. A. Montanari
DOI: 10.2174/157018008784083947
Published on: 01 March, 2012

Inherent Gene Expression Variabilities and the Need for Personalized Drug Dosage

Volume:5   Issue: 3
Pp: 193-208
Hamid Bolouri
DOI: 10.2174/157018008784084036
Published on: 01 March, 2012

Intravenous Thrombolysis with rt-PA in Acute Stroke Patients Aged ≥80 Years

Volume:5   Issue: 3
Pp: 209-213
S. Lorenzano, F. Orzi, E. Puca and D. Toni
DOI: 10.2174/157018008784084009
Published on: 01 March, 2012

Synthesis and Biological Evaluation of a Series of 2-(3,4,5-Trimethoxybenzoyl)-Indol-3-yl Acetic Acid Derivatives as Potential Agents against Human Leukemia K562 Cells

Volume:5   Issue: 3
Pp: 214-220
Romeo Romagnoli, Pier Giovanni Baraldi, Olga Cruz-Lopez, Maria Dora Carrion, Carlota Lopez Cara, Jan Balzarini, Enrica Fabbri and Robero Gambari
DOI: 10.2174/157018008784083983
Published on: 01 March, 2012

Synthesis and Biological Evaluation of N-(Alkyl)-2-Thiophen-2-Ylacetamides Series As A New Class of Antitubercular Agents

Volume:5   Issue: 3
Pp: 221-224
Marcus Vinicius Nora de Souza, Marcelle de Lima Ferreira, Thais Cristina Mendonca Nogueira, Raoni Schroeder Borges Goncalves, Monica Amado Peralta, Maria Cristina Silva Lourenco and Felipe Rodrigues Vicente
DOI: 10.2174/157018008784083965
Published on: 01 March, 2012

Novel 1, 2, 3-Triazole-Linked Norcantharidin Analogues: Synthesis and Evaluation of Growth Inhibition in a Panel of Selected Tumor-Cell Lines

Volume:5   Issue: 3
Pp: 225-231
Liping Deng, Bo yang, Qiaojun He and Yongzhou Hu
DOI: 10.2174/157018008784083992
Published on: 01 March, 2012