Letters in Drug Design & Discovery

Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

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Preface free to download

Volume:18   Issue: 1
Pp: 1-1
Kamil Kuca
DOI: 10.2174/157018081801201217095239
Published on: 26 February, 2021



Meet Our Editorial Board Member free to download

Volume:18   Issue: 1
Pp: 2-2
Mehlika Dilek Altintop
DOI: 10.2174/157018081801201217094130
Published on: 26 February, 2021



Synthesis of New Bis-pyrazolines Endowed with Potent Antifungal Activity against Candida albicans and Aspergillus niger

Volume:18   Issue: 1
Pp: 3-15
Belgin Sever, Mehlika Dilek Altintop* and Ahmet Özdemir
DOI: 10.2174/1570180817999201008155247
Published on: 26 February, 2021




Molecular Docking Analysis of Flavonoid Compounds with Matrix Metalloproteinase- 8 for the Identification of Potential Effective Inhibitors

Volume:18   Issue: 1
Pp: 16-45
Amir Taherkhani, Athena Orangi, Shirin Moradkhani and Zahra Khamverdi*
DOI: 10.2174/1570180817999200831094703
Published on: 26 February, 2021




Design, Synthesis and Biological Evaluation of 3-(2-(benzo[d]thiazol-2- ylthio)acetamido)benzoic Acid Derivatives as Inhibitors of Protein Tyrosine Phosphatase 1B

Volume:18   Issue: 1
Pp: 46-56
Monika Rakse*, Chandrabose Karthikeyan, Narayana Subbiah Hari Narayana Moorthy and Ram Kishore Agrawal
DOI: 10.2174/1570180817999200819122350
Published on: 26 February, 2021




Unveiling the Anti-tubercular Properties of Biscoumarins, through Biological Evaluation and Docking Studies

Volume:18   Issue: 1
Pp: 57-66
Poornima Acharya, M.M.V. Ramana*, Manish Upadhyay and Ganesh Pavale
DOI: 10.2174/1570180817999200724173656
Published on: 26 February, 2021




Preliminary Identification of Hamamelitannin and Rosmarinic Acid as COVID-19 Inhibitors Based on Molecular Docking

Volume:18   Issue: 1
Pp: 67-75
Kaushik Sarkar and Rajesh Kumar Das*
DOI: 10.2174/1570180817999200802032126
Published on: 26 February, 2021




Triazolylthioacetamides Confer Inhibitory Efficacy against Metallo-β- Lactamase IMP-1

Volume:18   Issue: 1
Pp: 76-84
Yue-Juan Zhang, Le Zhai, Yi Wan and Ke-Wu Yang*
DOI: 10.2174/1570180817999200831094019
Published on: 26 February, 2021




Synthesis of PF-543 Derivatives Using Simple Synthetic Methods and Their Biological Effect Analysis for the Development of Anticolorectal Cancer Agents

Volume:18   Issue: 1
Pp: 85-92
Jitendra Shrestha, Joo-Youn Lee, Eun-Young Park* and Dong Jae Baek*
DOI: 10.2174/1570180817999200908093524
Published on: 26 February, 2021




In Silico Based Structural and Fingerprint Analysis of Structurally Diverse AT1 inhibitors

Volume:18   Issue: 1
Pp: 93-103
Narayana Subbiah Hari Narayana Moorthy*
DOI: 10.2174/1570180817999200818155601
Published on: 26 February, 2021




A Novel Combinational Nanodrug Delivery System Induces Synergistic Inhibition of Lung Adenocarcinoma Cells In vitro

Volume:18   Issue: 1
Pp: 104-110
Mingliang Fan and Jiping Li*
DOI: 10.2174/1570180817999200719152426
Published on: 26 February, 2021