ISSN (Print): 1570-1808
ISSN (Online): 1875-628X

Volume 17, 12 Issues, 2020

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Letters in Drug Design & Discovery

ISSN (Print): 1570-1808
ISSN (Online): 1875-628X

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55^th of 59 in Chemistry, Medicinal

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Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

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R. F. Borne, Associate Director
Laboratory for Applied Drug Design and Synthesis, The University of Mississippi, USA

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Dima Sabbah
(Department of Pharmacy, Faculty of Pharmacy, Al-Zaytoonah University of Jordan, Amman, Jordan.)

Has contributed: CETP Inhibitory Activity of Chlorobenzyl Benzamides: QPLD Docking, Pharmacophore Mapping and Synthesis.

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Meet Our Editorial Board Member free to download

Volume:17 Issue: 4
Pp: 363-363
Janina Baranowska-Kortylewicz
DOI: 10.2174/157018081704200228122644

Editorial

The 2019 Novel Coronavirus (COVID-19) Outbreak in China and World: A New Lesson for Public Health System free to download

Volume:17 Issue: 4
Pp: 364-365
Kamil Kuca
DOI: 10.2174/157018081704200310125801

Review Article

Carbon Nanotubes Enhance the Chemotherapy Sensitivity of Tumors with Multidrug Resistance

Volume:17 Issue: 4
Pp: 366-378
Zhijie Wang, Jinhua Tao, Jianan Chen and Qian Liu*
DOI: 10.2174/1570180816666190405110858

Review Article

Phage Display as A Bio-Technique for Cancer Immunotherapy

Volume:17 Issue: 4
Pp: 379-387
Shirin Mahmoodi, Navid Nezafat* and Younes Ghasemi*
DOI: 10.2174/1570180816666190611160443

Research Article

3D-QSAR Studies on 4,5-Dihydro-1H-pyrazolo [4,3-h] Quinazolines as Plk-1, CDK2/A and Aur-A Serine/Threonine Kinase Inhibitors

Volume:17 Issue: 4
Pp: 388-395
Bhoomendra A. Bhongade*, Nikhil D. Amnerkar* and Andanappa K. Gadad
DOI: 10.2174/1570180816666190611161332

Research Article

Synthesis of New 4-Chloro-6-Methylpyrimidin-2-yl-Aminophosphonates as Potential DU145 and A549 Cancer Cell Inhibitors

Volume:17 Issue: 4
Pp: 396-410
Gajjala Raghavendra Reddy, Chinta Raveendra Reddy, Gopireddy Venkata Subba Reddy, Pasupuleti Visweswara Rao, Meenakshisundaram Swaminathan, Balam Satheeh Krishna and Cirandur Suresh Reddy*
DOI: 10.2174/1570180816666190329223207

Research Article

Antiglycation Activity of N, N-Diethylthiobarbiturates Derivatives

Volume:17 Issue: 4
Pp: 411-417
Momin Khan*, Ghulam Ahad, Ajmal Khan, Sana Shah, Kanwal, Uzma Salar, Syed Muhammad Salman and Khalid Mohammed Khan*
DOI: 10.2174/1570180816666190516111516

Research Article

Design, Synthesis and In Vitro Evaluation of 2-Oxo-N-substituted Phenyl- 2H-chromene-3-carboxamide Derivatives as HIV Integrase Strand Transfer Inhibitors

Volume:17 Issue: 4
Pp: 418-427
Pankaj Wadhwa*, Priti Jain and Hemant R. Jadhav
DOI: 10.2174/1570180816666190617150803

Research Article

In vitro and In Vivo Evaluation of Quinoxaline 1,4-di-N-oxide Against Giardia lamblia

Volume:17 Issue: 4
Pp: 428-433
Elizabeth Barbosa-Cabrera, Rosa Moo-Puc, Antonio Monge, Alma Delia Paz-González, Virgilio Bocanegra-García and Gildardo Rivera*
DOI: 10.2174/1570180816666190618115854

Research Article

Synthesis, In Silico and In Vivo Evaluation of Novel 1, 3, 4-Thiadiazole Analogues as Novel Anticancer Agents

Volume:17 Issue: 4
Pp: 434-444
Swathi Krishna, Byran Gowramma*, Manal Mohammed, Rajagopal Kalirajan, Lakshman Kaviarasan and Thaggikuppe Krishnamurthy Praveen*
DOI: 10.2174/1570180816666190710145939

Research Article

In Silico Elucidation of the Molecular Recognition of Phenol Derivative Compounds and Hippuryl-histidyl-leucine as an Artificial Substrate with the Experimental Target: Angiotensin-converting Enzyme

Volume:17 Issue: 4
Pp: 445-466
Víctor Hugo Vázquez-Valaldez*, Manuel Alejandro Hernández S, Ivonne Carrillo Cedillo, Ana María Velázquez Sanchez, Mildred Sauce Guevara, Rafael López Castañares and Enrique Ángeles
DOI: 10.2174/1570180816666190906155034

Research Article

Studies on the pIC50 of 4,5-Diarylisoxazole as HSP90 Inhibitors

Volume:17 Issue: 4
Pp: 467-478
Jing Ouyang, Xiaoqian Liu, Yutao Zhao, Ying Liu, Hongzong Si* and Honglin Zhai
DOI: 10.2174/1570180816666190329221959

Research Article

Evaluating Radioprotection of Rat’s Jejunum by a Combination of Melatonin and Metformin

Volume:17 Issue: 4
Pp: 479-484
Nasim Ahmadi Azar, Abdolreza Javadi, Masoud Najafi*, Alireza Shirazi*, Elham Tajabadi, Dheyauldeen Shabeeb and Ahmed Eleojo Musa
DOI: 10.2174/1570180816666190617153004

Research Article

Synthesis of Thiazole, Thiophene, Pyran and Pyridine Derivatives Derived from 3-phenyl-1H-pyrazol-5(4H)-one with Anti-proliferative, Tyrosine Kinase and PIM-1 Kinase Inhibitions

Volume:17 Issue: 4
Pp: 485-501
Rafat Milad Mohareb* and Ibram Refat Mikhail
DOI: 10.2174/1570180816666190618105907

Research Article

New Hydrazone Derivatives of Pyrazole-4-carboxaldehydes Exhibited Anti-inflammatory Properties

Volume:17 Issue: 4
Pp: 502-511
Mingxia Song, Bing Liu, Shengwang Yu, Shihui He, Yuqiu Liang, Sifan Li, Qiuyan Chen and Xianqing Deng*
DOI: 10.2174/1570180816666190731113441

Research Article

Synthesis and Cytotoxicity of New Mannich Bases of 6-[3-(3,4,5-Trimetoxyphenyl)-2- propenoyl]-2(3H)-Benzoxazolone

Volume:17 Issue: 4
Pp: 512-517
Ognyan Ivanov Petrov, Yordanka Borisova Ivanova*, Mariana Stefanova Gerova and Georgi Tsvetanov Momekov
DOI: 10.2174/1570180816666190730164952