Letters in Drug Design & Discovery


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

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Volume:17   Issue: 3
Pp: 227-227
Dimitra Hadjipavlou-Litina
DOI: 10.2174/157018081703200203143859

Nitric Oxide Synthases and Their Inhibitors: A Review

Volume:17   Issue: 3
Pp: 228-252
Anshika Mittal and Rita Kakkar*
DOI: 10.2174/1570180816666190222154457

Application of Topological Descriptors in QSAR Modeling: Substituted Hydrazones Used As a Model System

Volume:17   Issue: 3
Pp: 253-263
Vesna Dimova* and Mirjana Stojan Jankulovska
DOI: 10.2174/1570180816666181226145411

Cephalosporin Conjugated Sulfonamides: Synthesis, Characterization and Anticancer Activities

Volume:17   Issue: 3
Pp: 264-270
Rana Asif Nadeem, Muhammad Abdul Qadir, Mahmood Ahmed* and Imran Sajid
DOI: 10.2174/1570180815666180820144621

New Hybrids Derived from the Natural Compound (-)-β-Pinene and Amides or Acylthioureas as Antitumor Agents open access plus

Volume:17   Issue: 3
Pp: 271-284
Shengliang Liao, Xiaoping Rao, Minggui Shen, Hongyan Si, Jie Song, Shibin Shang* and Zhanqian Song*
DOI: 10.2174/1570180816666181107094427

Synthesis of Limonin Derivatives with Improved Anti-inflammatory and Analgesic Properties open access plus

Volume:17   Issue: 3
Pp: 285-299
Chengshu Jia, Bin Hu, Yingying Ji, Yourui Su, Guoqing Gong, Qihua Zhu and Yungen Xu*
DOI: 10.2174/1570180816666181113102359

Novel Strobilurin Derivatives Containing Carboxylate Unit as Potential Antifungal Agents open access plus

Volume:17   Issue: 3
Pp: 300-311
Longzhu Bao, Shuangshuang Wang, Di Song, Jingjing Wang, Xiali Yue and Xiufang Cao*
DOI: 10.2174/1570180816666190325164452

A Series of Furan-based Hydrazones: Design, Synthesis, and Evaluation of Antimicrobial Activity, Cytotoxicity and Genotoxicity open access plus

Volume:17   Issue: 3
Pp: 312-322
Mehlika Dilek Altintop*, Belgin Sever, Özlem Atli Eklioğlu, Merve Baysal, Rasime Demirel and Ahmet Özdemir
DOI: 10.2174/1570180816666190325163948

Drug Discovery of Acetophenone Derivatives as BRD4 Inhibitors open access plus

Volume:17   Issue: 3
Pp: 323-329
Zhimin Zhang, Wenhai Huang, Xiaoliang Zheng, Chuansheng Li and Zhengrong Shen*
DOI: 10.2174/1570180816666190329223559

An Efficient Protocol for the Synthesis, Biological Screening and Molecular Docking Studies of 3,4-Dihydropyrimidine-2-one/thione Derivatives

Volume:17   Issue: 3
Pp: 330-340
Ehsan Ullah Mughal*, Hafiz Umar Farooq, Amina Sadiq, Hummera Rafique, Sajjad Hussain Sumrra, Muhammad Naveed Zafar, Nighat Fatima, Syed Aun Muhammad, Abdul Manan, Chaudhary Omer Javed and Muhammad Tayyab
DOI: 10.2174/1570180816666190329224458

3D-QSAR and Docking Studies on Pyrimidine Derivatives as CSF-1R Inhibitors

Volume:17   Issue: 3
Pp: 341-355
Ya-ting Deng, Jun-wei Wang, Han Chu, Juan Wang, Yong Hu, Yong lin, Mao Shu and Zhi-hua Lin*
DOI: 10.2174/1570180816666190329224946

5-Nitrofuran-2-yl Thiohydrazones as Double Antibacterial Agents Synthesis and In Vitro Evaluation

Volume:17   Issue: 3
Pp: 356-361
Alexey Yurjevich Lukin, Tatiana Sergeevna Vedekhina and Mikhail Vassiljevich Chudinov*
DOI: 10.2174/1570180816666190221162055