Letters in Drug Design & Discovery

Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

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Volume:17   Issue: 2
Pp: 103-103
Miguel Munoz
DOI: 10.2174/157018081702191227121937



Progress in Synthesis and Bioactivity Evaluation of Pyrazoloquinazolines

Volume:17   Issue: 2
Pp: 104-113
Hui Zhao, Xiaoxia Hu, Yue Zhang, Chunlei Tang* and Bainian Feng*
DOI: 10.2174/1570180815666181017120100




Desirability Based Optimization of New Mesalazine Modified Release Formulations: Compression Coated Tablets and Mini Tablets in Capsules

Volume:17   Issue: 2
Pp: 114-123
Marilena Vlachou*, Angeliki Siamidi and Yannis Dotsikas
DOI: 10.2174/1570180816666190110125812




New 2-Oxopyridine/2-Thiopyridine Derivatives Tethered to a Benzotriazole with Cytotoxicity on MCF7 Cell Lines and with Antiviral Activities

Volume:17   Issue: 2
Pp: 124-137
Adel Mahmoud Attia, Ahmed Ibrahin Khodair*, Eman Abdelnasser Gendy, Mohammed Abu El-Magd and Yaseen Ali Mosa Mohamed Elshaier*
DOI: 10.2174/1570180816666190220123547




An Environment-friendly Synthesis of Piperonal Chalcones and Their Cytotoxic and Antioxidant Evaluation

Volume:17   Issue: 2
Pp: 138-144
Sanal Dev, Della Grace Thomas Parambi, Bency Baby, Githa Elizabeth Mathew, Hendawy Omnia Magdy, Monu Joy, Shine Sudev and Bijo Mathew*
DOI: 10.2174/1570180815666181016155934




Synthesis, Antiproliferative, and Antioxidant Activities of Substituted N-[(1,3,4-Oxadiazol-2-yl) Methyl] Benzamines

Volume:17   Issue: 2
Pp: 145-154
Mohamed Jawed Ahsan*, Lakshya Bhandari, Shally Makkar, Rajan Singh, Mohd. Zaheen Hassan, Mohammed H. Geesi, Mohamed Afroz Bakht, Surender Singh Jadav, Tuniki Balaraju, Yassine Riadi , Sandhya Rani, Habibullah Khalilullah, Vasubabu Gorantla and Afzal Hussain
DOI: 10.2174/1570180816666181113110033




3D-QSAR Assisted Design of Novel 7-Deazapurine Derivatives as TNNI3K Kinase Inhibitors Using Molecular Docking and Molecular Dynamics Simulation

Volume:17   Issue: 2
Pp: 155-168
Pavithra K. Balasubramanian, Anand Balupuri, Swapnil P. Bhujbal and Seung Joo Cho*
DOI: 10.2174/1570180816666190110121300




p-Trifluoroacetophenone Oxime Ester Derivatives: Synthesis, Antimicrobial and Cytotoxic Evaluation and Molecular Modeling Studies

Volume:17   Issue: 2
Pp: 169-183
İrem Bozbey, Suat Sari, Emine Şalva, Didem Kart and Arzu Karakurt*
DOI: 10.2174/1570180816666181128112249




Anti-Trypanosoma cruzi Activity and Molecular Docking Studies of 1Hpyrazolo[ 3, 4-b]pyridine Derivatives

Volume:17   Issue: 2
Pp: 184-191
Camilo Henrique da Silva Lima, Júlio César de Araujo Vanelis Soares, Joana Lucius de Sousa Ribeiro, Estela Maris Freitas Muri, Sérgio de Albuquerque and Luiza Rosaria Sousa Dias*
DOI: 10.2174/1570180816666190305141733




Synthesis and Herbicidal Activities of Novel Thiazole PPO Inhibitors

Volume:17   Issue: 2
Pp: 192-198
Shu Chen, Guihua Ren, Dan Pei, Fan Zhang, Jie Liu, Donglin Zhang, Ren Yang, Jianjun Shi, Tianming Xu and Chengxia Tan*
DOI: 10.2174/1570180816666190329221521




QSAR Analysis of Selected Antimicrobial Structures Belonging to Nitro-derivatives of Heterocyclic Compounds

Volume:17   Issue: 2
Pp: 214-225
Piotr Kawczak*, Leszek Bober and Tomasz Bączek
DOI: 10.2174/1570180815666181004112947




Correction to: Computational Identification of Inhibitors Against DPP-IV for Checking Type-2 Diabetes promotion: free to download

Volume:17   Issue: 2
Pp: 226-226
Sarvesh Kumar Gupta, Kamal Kumar Chaudhary, Utkarsh Raj and Nidhi Mishra*
DOI: 10.2174/157018081702191227145451