Letters in Drug Design & Discovery

Editor-in-Chief

Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo
(Italy)

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Volume: 16 Issue: 4, April 2019



Meet Our Associate Editorial Board Member free to download

Volume:16   Issue: 4
Pp: 371-371
Bruno Rizzuti
DOI: 10.2174/157018081604190220100304
Published on: 19 February, 2019



Benzothiazol Clubbed Imidazol-4-ones as Anti-fungal, Anti-tubercular and Anti-HIV-1 Agents: Their Synthesis and Molecular Docking Study

Volume:16   Issue: 4
Pp: 382-391
Navin B. Patel*, Asif R. Shaikh, Vatsal M. Patel, Edgar E. Lara-Ramirez and Gildardo Rivera
DOI: 10.2174/1570180815666180712150050
Published on: 12 July, 2018




Synthesis, Molecular Modelling and Antibacterial Activity Against Helicobacter pylori of Novel Diflunisal Derivatives as Urease Enzyme Inhibitors

Volume:16   Issue: 4
Pp: 392-400
Göknil Pelin Coşkun, Teodora Djikic, Sadık Kalaycı, Kemal Yelekçi, Fikrettin Şahin and Ş. Güniz Küçükgüzel*
DOI: 10.2174/1570180815666180627130208
Published on: 27 June, 2018




Synthesis of 3-Arylindazole-1-acetic Acids and In Vitro Study of Potential Antibacterial Effect

Volume:16   Issue: 4
Pp: 401-407
Fauzia Anjum Chattha, Samina Kousar, Mehr-un-Nisa and Munawar Ali Munawar*
DOI: 10.2174/1570180815666180702152259
Published on: 02 July, 2018




Anti-Microbial and Free Radical Scavenging Activities of Nigella Sativa Colloidal-Emulgel

Volume:16   Issue: 4
Pp: 408-416
Ahmad M. Eid*, Nidal A. Jaradat, Nagib A. Elmarzugi, Raed Alkowni, Fatima Hussen, Laila A. Ayyash, Maher Sawafta and Hadeel Danaa
DOI: 10.2174/1570180815666180620150922
Published on: 20 June, 2018




Virtual Screening, Molecular Modelling and Biochemical Studies to Exploit PF14_0660 as a Target to Identify Novel Anti-malarials

Volume:16   Issue: 4
Pp: 417-426
Vimee Raturi, Kumar Abhishek, Subhashis Jana, Subhendu Sekhar Bag and Vishal Trivedi*
DOI: 10.2174/1570180815666180727121200
Published on: 27 July, 2018




Synthesis and Anticandidal Activities of Some Aryl (5-Chloro-Benzofuran- 2-yl) Ketoximes

Volume:16   Issue: 4
Pp: 427-436
Ahmet Cagri Karaburun*
DOI: 10.2174/1570180816666181207155701
Published on: 07 December, 2018




Evaluation of the in vitro Antitumor Activity of Nanostructured Cyclotides in Polymers of Eudragit® L 100-55 and RS 30 D

Volume:16   Issue: 4
Pp: 437-445
Osmar N. Silva, Michelle F.S. Pinto, Juliane F.C. Viana, Camila G. Freitas, Isabel C.M. Fensterseifer, David J. Craik and Octavio L. Franco*
DOI: 10.2174/1570180815666180801115526
Published on: 31 July, 2018




Design and Synthesis of Novel Thiosemicarbazones as Potent Anti-breast Cancer Agents open access plus

Volume:16   Issue: 4
Pp: 446-452
Mashooq Ahmad Bhat*, M. Al-Tahhan, Mohamed A. Al-Omar, Ahmed M. Naglah and Abdullah Al-Dhfyan
DOI: 10.2174/1570180815666181008100944
Published on: 07 October, 2018




QSAR Studies on Thiazole Derivatives as HCV NS5A Inhibitors via CoMFA and CoMSIA Methods

Volume:16   Issue: 4
Pp: 453-460
Jiayu Li, Wenyue Tian, Diaohui Gao, Yuying Li, Yiqun Chang, Jun Xu, Junxia Zheng* and Pinghua Sun*
DOI: 10.2174/1570180815666180702153529
Published on: 02 July, 2018




2-Acryloyl-4,5-methylenedioxyphenol: A Small Molecule Endowed with Antidermatophytic Activity

Volume:16   Issue: 4
Pp: 461-466
Marco Zuccolo, Sabrina Dallavalle*, Raffaella Cincinelli, Luce Mattio, Stefania Mazzini, Michelandrea De Cesare and Loana Musso
DOI: 10.2174/1570180815666180803115347
Published on: 02 August, 2018




Theoretical Coupling and Stability of Boronic Acid Adducts with Catecholamines

Volume:16   Issue: 4
Pp: 467-475
Eugeniy Demianenko, Alexey Rayevsky, Marvin A. Soriano-Ursúa* and José G. Trujillo-Ferrara*
DOI: 10.2174/1570180815666180710101604
Published on: 09 July, 2018