Letters in Drug Design & Discovery


Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo

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Volume: 15 Issue: 9, September 2018

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Volume:15   Issue: 9
Pp: 913-913
Janina Baranowska-Kortylewicz
DOI: 10.2174/157018081509180716155406
Published on: 16 July, 2018

Synthesis, Biological Evaluation and Computational Study of New Quinoline Hybrids as Antitubercular Agent

Volume:15   Issue: 9
Pp: 914-922
Zahid Zaheer*, Sameer I. Shaikh, Santosh N. Mokale and Deepak K. Lokwani
DOI: 10.2174/1570180814666171026155930
Published on: 26 October, 2017

Synthesis and Biological Evaluation of N-(5-(2,5-dimethyl-phenoxy)-2,2-dimethylpentyl)-benzamide Derivatives as Novel Farnesoid X Receptor (FXR) Antagonist

Volume:15   Issue: 9
Pp: 923-936
Siyun Nian, Zhenpeng Yu, Xiangduan Tan, Xia Gan, Mohan Huang, Yihuan Zhou and Guoping Wang*
DOI: 10.2174/1570180815666171226150403
Published on: 26 December, 2017

Design, Synthesis and anti-HIV-1 Activity of Modified Styrylquinolines

Volume:15   Issue: 9
Pp: 937-944
Shivani Mahajan, Shiv Gupta, Nisha Jariwala, Deepali Bhadane, Late K.K. Bhutani, Smita Kulkarni* and Inder Pal Singh*
DOI: 10.2174/1570180815666171212143339
Published on: 12 December, 2017

Synthesis and Bioevaluation of Shikonin Derivatives

Volume:15   Issue: 9
Pp: 945-950
Sufen Cao, Jiangang Zhang and Wenhu Duan*
DOI: 10.2174/1570180815666171229152139
Published on: 29 December, 2017

Synthesis and Mosquiticidal Activity of Novel Hydrazone Containing Pyrimidine Derivatives against Aedes aegypti

Volume:15   Issue: 9
Pp: 951-956
Zhong-Hua Shen, Zhao-Hui Sun, James J. Becnel, Alden Estep, David E. Wedge*, Cheng-Xia Tan, Jian-Quan Weng, Liang Han and Xing-Hai Liu*
DOI: 10.2174/1570180815666180102141640
Published on: 02 January, 2018

4-Acetamidobenzaldehyde Derivatives as Biological Active Candidates; Synthesis, Anti-oxidant, Anti-Alzheimer and DNA Binding Studies

Volume:15   Issue: 9
Pp: 957-968
Shahzad Murtaza* and Adina Tatheer
DOI: 10.2174/1570180814666171026161646
Published on: 26 October, 2017

The Possible Potency of Ocimum basilicum New Constituent on Glucosestimulated Insulin Secretion In Vitro and β-cell Function In Vivo

Volume:15   Issue: 9
Pp: 969-978
Huma Aslam Bhatti*, Kiran Maryam, Rizwana S. Waraich, Abdul Hameed and Rahman M. Hafizur
DOI: 10.2174/1570180814666171113155732
Published on: 13 November, 2017

3D-QSAR Modeling of Some S-trityl-L-Cysteine Analogues as Inhibitors of Mitotic Kinesin Eg5 by CoMFA, CoMSIA and H-QSAR Methodologies

Volume:15   Issue: 9
Pp: 979-987
Fatemeh Mousavi and Mohammad Hossein Fatemi*
DOI: 10.2174/1570180814666171026162737
Published on: 26 October, 2017

Theoretical Modeling and Systemic Analysis of Various Active Dipeptides and Analogues with 3D-QSAR Methods

Volume:15   Issue: 9
Pp: 988-1001
Guanghui Tang, Cheng Chen, Yuping Zhang, Ya Zhang, Yuanqiang Wang* and Zhihua Lin*
DOI: 10.2174/1570180814666171027162400
Published on: 27 October, 2017

Charting the Bromodomain BRD4: Towards the Identification of Novel Inhibitors with Molecular Similarity and Receptor Mapping

Volume:15   Issue: 9
Pp: 1002-1011
Fernando D. Prieto-Martinez and Jose L. Medina-Franco*
DOI: 10.2174/1570180814666171121145731
Published on: 21 November, 2017

Molecular and Cellular Mechanism of Cutaneous Injuries Due to Exposure to Sulfur Mustard

Volume:15   Issue: 9
Pp: 1012-1018
Yunes Panahi, Seyyed Mahdi Rajaee and Amirhossein Sahebkar*
DOI: 10.2174/1570180814666171026160410
Published on: 26 October, 2017