Letters in Drug Design & Discovery


Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo

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Volume: 14 Issue: 9, September 2017

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Volume:14   Issue: 9
Pp: 985-985
Ilkay Erdogan Orhan
DOI: 10.2174/157018081409170810092418
Published on: 09 August, 2017

Docking-based 3D-QSAR Studies of Phosphodiesterase 9A Inhibitors

Volume:14   Issue: 9
Pp: 986-998
Changji Tan, Yinuo Wu, Yongxian Shao, Haibin Luo, Xuehua Zheng* and Laiyou Wang*
DOI: 10.2174/1570180814666170110124314
Published on: 10 January, 2017

Synthesis and Anticancer Studies of Novel N-benzyl Pyridazino ne Derivatives

Volume:14   Issue: 9
Pp: 1008-1013
Mohamed Elagawany, Mohamed A. Ibrahim, Tarek S. Ibrahim, Amany M.M. AL-Mahmoudy, Alaa Moawad, Mohammed M. Ghoneim, Mohamed M. Radwan and Siva S. Panda*
DOI: 10.2174/1570180814666170223111312
Published on: 22 February, 2017

Synthesis and Antimicrobial Activities of Hybrid Heterocyclic Molecules Based on 1-(4-Fluorophenyl)piperazine Skeleton

Volume:14   Issue: 9
Pp: 1014-1034
Serap Basoglu Ozdemir, Neslihan Demirbas*, Yıldız Uygun Cebeci, Hacer Bayrak, Arif Mermer, Sule Ceylan and Ahmet Demirbas
DOI: 10.2174/1570180814666170113145023
Published on: 13 January, 2017

Synthesis, Molecular Docking Studies and Biological Evaluation o f 3-Iminoaurones as Acetylcholinesterase and Butyrylcholinesterase Inhibitors

Volume:14   Issue: 9
Pp: 1035-1041
Ehsan Ullah Mughal*, Amina Sadiq, Bilal Ahmad Khan, Muhammad Naveed Zafar, Ishtiaq Ahmed and Muhammad Zubair
DOI: 10.2174/1570180814666170106123959
Published on: 05 January, 2017

Antimicrobial and Cytotoxicity Activities of 2-(aryl)-3-(benzo[d][1,3] dioxol-5-yl)thiazolidin-4-ones

Volume:14   Issue: 9
Pp: 1042-1047
Silvana P. Souza, Hellen G. Masteloto, Daniel S. da Silva, Juliana H. Azambuja, Elizandra Braganhol, Juliana S. Ribeiro, Rafael G. Lund and Wilson Cunico*
DOI: 10.2174/1570180814666170106143418
Published on: 06 January, 2017

Multiplication of Mycobacterium tuberculosis in Peripheral Blood of Mice and Effect of Anti-tubercular Drugs on Bacteremia

Volume:14   Issue: 9
Pp: 1048-1052
Richa Dwivedi, Shubhra Singh, Priyanka Trivedi and Vinita Chaturvedi*
DOI: 10.2174/1570180814666170223171215
Published on: 23 February, 2017

Antiproliferative Activity of Olive Oil Phenolics against Human Melan oma Cells

Volume:14   Issue: 9
Pp: 1053-1059
A. L.M. Batista de Carvalho, F. Caselli, V. Rodrigues, F. Paiva-Martins and M.P. M. Marques*
DOI: 10.2174/1570180814666170110145658
Published on: 10 January, 2017

Combination of Irbesartan with Amlodipine Enhances Nitrate/Nitrite Generation by Angiotensin II-exposed Endothelial Cells

Volume:14   Issue: 9
Pp: 1060-1064
Yuji Ishibashi, Takanori Matsui, Nobutaka Nakamura and Sho-ichi Yamagishi*
DOI: 10.2174/1570180814666170102154739
Published on: 02 January, 2017

Design, Synthesis and Evaluation of Dual-targeting Prodrug Co-modified by Organic Amine and L-ascorbic Acid for CNS Delivery

Volume:14   Issue: 9
Pp: 1065-1072
Shubing Qiu, Yi Zhao, Sha Liu, Xiaocen Li, Li Guo, Li Hai* and Yong Wu*
DOI: 10.2174/1570180814666161230161152
Published on: 30 December, 2016

Design, Synthesis, Characterization, Molecular Docking, ADME Properties and In Vivo Antipsychotic Activity of Aripiprazole Related Drugs Candidates

Volume:14   Issue: 9
Pp: 1073-1085
Selvarasu Sekar, Srinivasan Pazhamalai, Ganesan Ariharasivakumar and Mannathusamy Gopalakrishnan*
DOI: 10.2174/1570180814666161207143742
Published on: 07 December, 2016

A Brief Overview on Chemistry and Biology of Benzoxepine

Volume:14   Issue: 9
Pp: 1086-1098
Naveen Kuntala, Jhonsee R. Telu, Jaya S. Anireddy and Sarbani Pal*
DOI: 10.2174/1570180814666161227125227
Published on: 27 December, 2016

Homology Modeling in Drug Discovery-an Update on the Last Decade

Volume:14   Issue: 9
Pp: 1099-1111
Geraldene Munsamy and Mahmoud E. S. Soliman*
DOI: 10.2174/1570180814666170110122027
Published on: 10 January, 2017