Letters in Drug Design & Discovery

Editor-in-Chief

Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo
(Italy)

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Volume: 14 Issue: 12, December 2017



Meet Our Editorial Board Member free to download

Volume:14   Issue: 12
Pp: 1347-1347
Enrico Garattini
DOI: 10.2174/157018081412171031113907
Published on: 31 October, 2017



QSAR Modeling of Aminopeptidase N/CD13 (APN) Inhibitory Activity of some Leucine Ureido Derivatives by GA-MLR and SW-MLR Methods

Volume:14   Issue: 12
Pp: 1348-1357
Naser Faraji, Tannaz Zebardast, Afshin Zarghi* and Zahra Hajimahdi*
DOI: 10.2174/1570180814666170529084557
Published on: 28 May, 2017




A Study on Identification of Nutraceutical Value of New Imidazolone Schiff Base Analogues

Volume:14   Issue: 12
Pp: 1358-1370
Subbulakshmi N. Karanth, Badiadka Narayana*, Balladka K. Sarojini, Saleemulla Khan and Shashidhara S. Kenkere
DOI: 10.2174/1570180814666170412120555
Published on: 12 April, 2017




An Improved Preparation of (R)-3-Aminobutanol, a Key Intermediate for the Synthesis of Dolutegravir Sodium

Volume:14   Issue: 12
Pp: 1371-1375
Y. Srinivasa Rao, B. Hari Babu*, I. Aminual, D. Nageshwar and P.V.V. Satyanarayana
DOI: 10.2174/1570180814666170602083756
Published on: 01 June, 2017




Design and Synthesis of Amino Acid Tethered Thiazolones to Screen for Hepatitis C NS5B Polymerase Inhibitors

Volume:14   Issue: 12
Pp: 1376-1381
Yili Ding*, Kenneth L. Smith and Chamakura V.N.S. Varaprasad
DOI: 10.2174/1570180814666170505121156
Published on: 05 May, 2017




Design, Synthesis and Antiproliferative Activities Evaluation of Thiazolopyrimidines Derivatives through Biginelli Reaction

Volume:14   Issue: 12
Pp: 1382-1390
Pengju Zhu, Huansheng Fu and Hao Fang*
DOI: 10.2174/1570180814666170512123132
Published on: 12 May, 2017




CETP Inhibitory Activity of Chlorobenzyl Benzamides: QPLD Docking, Pharmacophore Mapping and Synthesis

Volume:14   Issue: 12
Pp: 1391-1400
Reema Abu Khalaf*, Hamada Abd El-Aziz, Dima Sabbah, Ghadeer Albadawi and Ghassan Abu Sheikha
DOI: 10.2174/1570180814666170412122304
Published on: 12 April, 2017




Preparation and Characterization of Mixed Polymeric Micelles as a Versatile Strategy for Meloxicam Oral Administration

Volume:14   Issue: 12
Pp: 1401-1408
Claudia Amaral, Mariana Magalhaes, Celia Cabral, Francisco Veiga and Ana Figueiras*
DOI: 10.2174/1570180814666170505120728
Published on: 05 May, 2017




The Impact of 5-Substituted Uracil Derivatives on Immortalized Embryo Lung Cells

Volume:14   Issue: 12
Pp: 1409-1414

DOI: 10.2174/1570180814666170502171640
Published on: 02 May, 2017




A SAR Study: Evaluation of Bromo Derivatives of 8-Substituted Quinolines as Novel Anticancer Agents

Volume:14   Issue: 12
Pp: 1415-1424
Salih Okten*, Osman Cakmak, Saban Tekin and Tugba Kul Koprulu
DOI: 10.2174/1570180814666170504150050
Published on: 04 May, 2017




Synthesis and Anti-Oxidant Evaluation of Some Novel Sulfa Drugs

Volume:14   Issue: 12
Pp: 1425-1432
Moustafa A. Gouda* and Belal H.M. Hussein
DOI: 10.2174/1570180814666170607144811
Published on: 07 June, 2017




Spices Chemoconstituents as Persuasive Inhibitor of S. typhimurium Virulent Protein L-asparaginase

Volume:14   Issue: 12
Pp: 1433-1454
Archana Vimal and Awanish Kumar*
DOI: 10.2174/1570180814666170602080822
Published on: 01 June, 2017




In Silico Prioritization, Synthesis and In Vitro Evaluation of Tembamide Analogs for Anti-HIV Activity

Volume:14   Issue: 12
Pp: 1455-1464
Shiv Gupta, Sanjay Kumar, Nisha Jariwala, Deepali Bhadane, Kamlesh Kumar Bhutani, Smita Kulkarni* and Inder Pal Singh*
DOI: 10.2174/1570180814666170419115526
Published on: 19 April, 2017




Neurokinin-1 Receptor Antagonists in Lung Cancer Therapy

Volume:14   Issue: 12
Pp: 1465-1476
Miguel Munoz*, Marisa Rosso and Rafael Covenas
DOI: 10.2174/1570180814666170327163854
Published on: 27 March, 2017




Acknowledgements to Reviewers free to download

Volume:14   Issue: 12
Pp: 1477-1477

DOI: 10.2174/157018081412171031150240
Published on: 31 October, 2017