Letters in Drug Design & Discovery


Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo

Personal Subscription
Become EABM
Become Reviewer
Call for Editor
Volume: 14 Issue: 11, November 2017

Meet Our Editorial Board Member free to download

Volume:14   Issue: 11
Pp: 1227-1227
Eliezer J. Barreiro
DOI: 10.2174/157018081411171003112446
Published on: 02 October, 2017

2D, 3D, G-QSAR and Docking Studies of Thiazolyl-pyrazoline Analogues as Potent (Epidermal Growth Factor Receptor-tyrosine Kinase) EGFR-TK Inhibitors

Volume:14   Issue: 11
Pp: 1228-1238
Ghodgaonkar Sunayana*, Bhandari Shashikant and Waghulde Sandeep
DOI: 10.2174/1570180814666170518171236
Published on: 18 May, 2017

Synthesis, Docking and Evaluation of Phenylacetic Acid and Trifluoro-methylphenyl Substituted Benzamide Derivatives as Potential PPARδ Agonists

Volume:14   Issue: 11
Pp: 1239-1251
Ajmer Singh Grewal, Viney Lather*, Deepti Pandita and Garima Bhayana
DOI: 10.2174/1570180814666170327164443
Published on: 27 March, 2017

Molecular Docking Studies of Novel Thiosemicarbazone-based Indoles as Potential PI3Kα Inhibitors

Volume:14   Issue: 11
Pp: 1252-1258
Dima A. Sabbah* and Kamal Sweidan
DOI: 10.2174/1570180814666170619112647
Published on: 18 June, 2017

Synthesis and Structure-activity Relationships of Chalcone Derivatives as Inhibitors of Ovarian Cancer Cell Growth

Volume:14   Issue: 11
Pp: 1259-1266
Zachary D. Tucker, Francis J. Barrios and Amanda J. Krzysiak*
DOI: 10.2174/1570180814666170505120258
Published on: 05 May, 2017

Molecular Docking and In Silico ADMET Study Reveals Flavonoids as a Potential Inhibitor of Aromatase

Volume:14   Issue: 11
Pp: 1267-1276
Umang Shah*, Samir Patel, Mehul Patel and Jagat Upadhayay
DOI: 10.2174/1570180814666170327161908
Published on: 27 March, 2017

Molecular Simulation and Activity Studies of Oxametacin as an HDAC Inhibitor

Volume:14   Issue: 11
Pp: 1277-1282
Fanbo Jing, Lei Zhang*, Yepeng Luan and Jiang Bian
DOI: 10.2174/1570180814666170505123930
Published on: 05 May, 2017

Molecular Docking Simulations as a Prominent Tool to Envisage the Preformulation Perspectives of Oral Hypoglycaemic Agents with β-cyclodextrin

Volume:14   Issue: 11
Pp: 1283-1290
Sant K. Verma and Akhlesh K. Jain*
DOI: 10.2174/1570180814666170420125907
Published on: 20 April, 2017

The Antiviral Effects of Harmine Against BoHV-1 Infection In Vitro

Volume:14   Issue: 11
Pp: 1303-1307
Xinyi Jiang, Jie Zou, Yuncheng Zhuang, Weifeng Yuan, Liqian Zhu* and Guoqiang Zhu*
DOI: 10.2174/1570180814666170425155554
Published on: 25 April, 2017

New Cyclohexylamine-dithiocarbamate Derivatives as Potential Anti-microbial Agents

Volume:14   Issue: 11
Pp: 1308-1315
Leyla Yurttas*, Betul Kaya , Meral Yilmaz Cankilic and Serkan Levent
DOI: 10.2174/1570180814666170412121402
Published on: 12 April, 2017

Synthesis and Antimicrobial Activity of Some Novel Substituted 3-(Thiophen-2-yl)pyrazole-based Heterocycles

Volume:14   Issue: 11
Pp: 1316-1323
Bakr F. Abdel-Wahab*, Abdelbasset A. Farahat, Ghada E. A. Awad and Gamal A. El-Hiti*
DOI: 10.2174/1570180814666170327162447
Published on: 27 March, 2017

Novel Thiazole Carboxylic Acid Derivatives Possessing a “Zinc Binding Feature” as Potential Human Glyoxalase-I Inhibitors

Volume:14   Issue: 11
Pp: 1324-1334
Qosay A. Al-Balasa*, Mohammad A. Hassana, Ghazi A. Al Jabala, Nizar A. Al-Shar, Ammar M. Almaaytahb and Tamam El-Elimata
DOI: 10.2174/1570180814666170306120954
Published on: 06 March, 2017

Synthesis and Antiproliferative Activity of 3-aza Steroids as 5α-reductase Inhibitors

Volume:14   Issue: 11
Pp: 1335-1346
Milanpreet Kaur, Richa Dhingra, T. R. Bhardwaj and Neelima Dhingra*
DOI: 10.2174/1570180814666170505122503
Published on: 05 May, 2017