Letters in Drug Design & Discovery

Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

Personal Subscription
Become EABM
Become Reviewer
Call for Editor

Molecular Docking and 3D-QSAR Studies on Quinolone-based HDAC Inhibitors

Volume:13   Issue: 7
Pp: 577-586
Yi Bi, Zeyun Liu, Xianxuan Liu, Xiaochen Zhang and Jing Lu
DOI: 10.2174/1570180812666150924000500
Published on: 29 June, 2016


Biological Evaluation of Small Molecule Inhibitors of Mtb-ASADH Enzyme

Volume:13   Issue: 7
Pp: 587-590
Rajender Kumar, Ratnika Sethi, Purvi Shah, Ipsita Roy, Inder Pal Singh, P. V. Bharatam, Rupinder Tewari and Prabha Garg
DOI: 10.2174/1570180813666160617102813
Published on: 29 June, 2016


Arginine-rich Cyclic Peptides Enhance Cellular Delivery of Anticancer Agents: Molecular Insights

Volume:13   Issue: 7
Pp: 591-604
Antara Banerjee, Naser Sayeh, Amir Nasrolahi Shirazi, Rakesh Tiwari, Keykavous Parang and Arpita Yadav
DOI: 10.2174/1570180813999160429113034
Published on: 29 June, 2016


Natural Alpha-Glucosidase Inhibitors: Therapeutic Implication and Structure- Activity Relation Ship

Volume:13   Issue: 7
Pp: 605-637
Sanae Abid, Ali Berraaouan and Mohamed Bnouham
DOI: 10.2174/1570180812666150918193508
Published on: 29 June, 2016


Modeling Ensembles of Loop Conformations by Iterative Stochastic Elimination

Volume:13   Issue: 7
Pp: 646-651
Amit Michaeli and Anwar Rayan
DOI: 10.2174/1570180813666160617103437
Published on: 29 June, 2016


Synthesis of Chalcone Derivatives and Their Effects on Proliferation and Tubulin Dynamics Instability of HT-29 Cells

Volume:13   Issue: 7
Pp: 662-667
Yasmin Tajuddin, Zaliha Harun, Ahmad Rohi Ghazali, Juriyati Jalil and Malina Jasamai
DOI: 10.2174/157018081307160630182605
Published on: 29 June, 2016


Reversal of Multi-Drug Resistance in Staphylococcus aureus by Natural Product-Way Forward

Volume:13   Issue: 7
Pp: 668-675
Saba Farooq, Atia-tul-Wahab, Ali Azarpira, Atta-ur-Rahman and M. Iqbal Choudhary
DOI: 10.2174/1570180813666151117212606
Published on: 29 June, 2016


Synthesis of Some Novel 2-Azetidinones/4-Thiazolidinones Bearing 1, 3, 4- Thiadiazole Nucleus and Screening for its Anti-Imflammatory Activity

Volume:13   Issue: 7
Pp: 676-683
B. Gowramma, T. K. Praveen, R. Kalirajan and B. Babu
DOI: 10.2174/1570180813666151123235546
Published on: 29 June, 2016


Synthesis and Anticancer Activity of 2-Aryl-6-diethylaminoquinazolinone Derivatives

Volume:13   Issue: 7
Pp: 684-690
Thanh Nguyen Le, Daulat Bikram Khadka, Giap Huu Tran, Dung Anh Nguyen, Yifeng Jin, Hue Thi My Van, Van Hung Nguyen and Won-Jea Cho
DOI: 10.2174/1570180813666160125222936
Published on: 29 June, 2016


Synthesis and Evaluation of Compounds Containing 4-arylpiperazinyl Moieties Linked to a 2-(pyridin-3-yl)-1H-benzimidazole as p38 MAP Kinase Inhibitors

Volume:13   Issue: 7
Pp: 691-696
Mohamed Ashraf Ali, Hasnah Osman, Raju Suresh Kumar, Abdulrahman I. Almansour, Natarajan Arumugam, Vijay H. Masand and Theivendren Panneerselvam
DOI: 10.2174/1570180812666151022221401
Published on: 29 June, 2016


Preparation of Chlorotoxin-conjugated Superparamagnetic Nanoparticle and its Magnetic Resonance Imaging In Vitro

Volume:13   Issue: 7
Pp: 697-705
Chen Zhu, Xiao Enhua, Shang Quanliang, Kang Zhen, Tan Huilong, Pengfei Xu and Zeng Wenbin
DOI: 10.2174/1570180813666160130003723
Published on: 29 June, 2016


Novel Biphenyl Derivatives with α-Aminophosphonate Moiety: Design, Synthesis and Antivirus Activity

Volume:13   Issue: 7
Pp: 706-714
Guo-Ping Zhang and Min Liu
DOI: 10.2174/1570180813666160125222813
Published on: 29 June, 2016


Synthesis and Antimicrobial Evaluation of Amphipathic Peptide Models

Volume:13   Issue: 7
Pp: 715-724
Marianna Sakka, Alexandra Balliou, Asimina Marianou, Dimitris Krikorian, Margarita Tsirogianni, Artemis Tsiligianni, Katerina Vartzeli, Anna-Irini Koukkou, Maria Sakarellos-Daitsiotis and Eugenia Panou- Pomonis
DOI: 10.2174/1570180813666160616122410
Published on: 29 June, 2016