Letters in Drug Design & Discovery

Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

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Volume:12   Issue: 7
Pp: i-v

DOI: 10.2174/157018081207150604165207
Published on: 05 June, 2015



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Volume:12   Issue: 7
Pp: 519-520
Xinyong Liu
DOI: 10.2174/157018081207150604165453
Published on: 05 June, 2015

6-Bromo-2,3-Dioxoindolin Phenylacetamide Derivatives: Synthesis, Potent CDC25B, PTP1B Inhibitors and Anticancer Activity

Volume:12   Issue: 7
Pp: 529-536
Shui-Lian Zhao, Zhou Peng, Xing-Hua Zhen, Yan Han, Hai-Ying Jiang, You-Le Qu and Li-Ping Guan
DOI: 10.2174/1570180812666141219003209
Published on: 05 June, 2015


3D-QSAR Study of Flavone Derivatives as Inhibitors of HeLa Cervix Adenocarcinoma Cell Lines

Volume:12   Issue: 7
Pp: 537-544
Yeonjoong Yong, Yearam Jung, Eunil Cho, Hyeonji Kim, Jin Sil Yoo, Dongsoo Koh, Hi Jae Cho, Somi Kim Cho and Yoongho Lim
DOI: 10.2174/1570180812666141205235800
Published on: 05 June, 2015


Proteins as Alternate Targets of Enediynes

Volume:12   Issue: 7
Pp: 545-557
Hussam M. Bdour, Snigdha Roy and Amit Basak
DOI: 10.2174/1570180812666150213224756
Published on: 05 June, 2015


Identification of Potential Mps1 Inhibitors Through Multiple Pharmacophore- based Virtual Screening and Molecular Docking

Volume:12   Issue: 7
Pp: 558-573
Xiaoli Li, Lu Zhou, Yahui Tian and Suwen Zhou
DOI: 10.2174/1570180812999150210142710
Published on: 05 June, 2015


Design, Synthesis and Biological Evaluation of Lapatinib Derivatives as HER1/HER2 Inhibitors

Volume:12   Issue: 7
Pp: 574-584
Aifeng Lyu, Lei Fang, Shaohua Gou and Xia Liu
DOI: 10.2174/1570180812999150206111626
Published on: 05 June, 2015


Synthesis and Preliminary Evaluation of Novel Bone-targeting NSAIDs Prodrugs based on Glutamic Acid Oligopeptides

Volume:12   Issue: 7
Pp: 585-590
Yi Zhao, Dongsheng He, Lifang Ma and Li Guo
DOI: 10.2174/1570180812999150217171229
Published on: 05 June, 2015


Syntheses of Ethyl Pyruvate’s Bioisosteres Inhibiting Inducible Nitric Oxide Production in Lipopolysaccharide-induced BV2 Cells

Volume:12   Issue: 7
Pp: 591-596
Ju-Young Park, Byung-Wook Kim, Soon-Jung Kwon, Dong-Kug Choi, Ja-Kyeong Lee and Sung-Hwa Yoon
DOI: 10.2174/1570180812999150225112225
Published on: 05 June, 2015


Synthesis and In vitro Evaluation of Dibenzoazepine Triazole Derivatives: A Novel Class of Antileishmanial Agents

Volume:12   Issue: 7
Pp: 597-606
Maria Aqeel Khan, Aliyan Saleem, Nida Ghouri, Abdul Hameed, M. Iqbal Choudhary and Fatima Z. Basha
DOI: 10.2174/1570180812999150225111959
Published on: 05 June, 2015


Synthesis and In Vitro Evaluation of Furan-Based Chalcone Derivatives as Antimicrobial Agents

Volume:12   Issue: 7
Pp: 607-611
Ahmet Ozdemir, Mehlika Dilek Altıntop, Zerrin Canturk and Zafer Asim Kaplancikli
DOI: 10.2174/1570180812999150202112352
Published on: 05 June, 2015