Letters in Drug Design & Discovery

Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

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Volume:12   Issue: 3
Pp: 165-165
James David Adams
DOI: 10.2174/157018081203141202095204
Published on: 02 December, 2014

Quantitative Structure – Activity Relationship Study on Saponins as Cytotoxicity Enhancers

Volume:12   Issue: 3
Pp: 166-171
Reneta Gevrenova, Alexander Weng, Laurence Voutguenne-Nazabadioko, Mayank Thakur and Irini Doytchinova
DOI: 10.2174/1570180811666140915221432
Published on: 02 December, 2014


The Disulfide Analogues of Isophosphoramide Mustard for Anticancer Therapy

Volume:12   Issue: 3
Pp: 172-179
Joanna Cytarska, Krzysztof Skowerski, Szymon Jaworski, Konrad Misiura, Beata Filip-Psurska and Joanna Wietrzyk
DOI: 10.2174/1570180811666141010001007
Published on: 02 December, 2014


Acyl Thiourea Derivatives Containing Pyrazole Ring Selective Targeting of Human Aurora Kinases in Breast and Bone Cancer

Volume:12   Issue: 3
Pp: 180-189
Aykut Ozgur, Eren Yenidunya, Irfan Koca and Yusuf Tutar
DOI: 10.2174/1570180811666141001005129
Published on: 02 December, 2014


6,7-Dimethoxyquinazolines as Potential Cytotoxic Agents: Synthesis and in vitro Activity

Volume:12   Issue: 3
Pp: 190-205
Mange Ram Yadav, Bishram Singh Chauhan, Prashant Naik, Hardik Gandhi and Rajani Giridhar
DOI: 10.2174/1570180811666141010000716
Published on: 02 December, 2014


Synthesis and Biological Evaluations of Novel Nitric Oxide-donating Derivatives of [1,2,4]triazol-5(4H)-one with N-phenylpyrrolyl-2-tetrazole Moiety as Anti-hypertension Candidates

Volume:12   Issue: 3
Pp: 206-210
Yanchun Zhanga, Jichao Chen, Jinyi Xub*, Jinpei Zhou and Xiaoming Wu*
DOI: 10.2174/1570180811666141009235816
Published on: 02 December, 2014


Biological Effect of Glycosyl-Oxadiazolinethione and Glycosyl-sulfanyloxadiazole Derivatives through their in vitro Inhibition of Glycosidases from Bacteria and Normal or Diabetic Rats

Volume:12   Issue: 3
Pp: 211-218
Mahmoud Balbaa, Aseel Shibli, Riham Hosna, Hoda Yusef, Ahmed T. A. Boraei and El Sayed H. El Ashry
DOI: 10.2174/1570180811666141010001221
Published on: 02 December, 2014


3D-QSAR and Docking Studies on 2-acyliminobenzimidazoles Derivatives as Potent ALK Inhibitors

Volume:12   Issue: 3
Pp: 219-233
Qianqian Lva, Zhi Wang, Zhonghua Wanga*, Fanhong Wu* and Liping Cheng
DOI: 10.2174/1570180811666141010001624
Published on: 02 December, 2014


Phenylacrylamides as Novel FtsZ-targeted Potential Antimicrobials

Volume:12   Issue: 3
Pp: 234-240
Xin Li, Juzheng Sheng, Di Song, Liwei Guo and Shutao Ma
DOI: 10.2174/1570180811666141009235409
Published on: 02 December, 2014


Synthesis and Insecticidal Activity of Acylthiourea Derivatives from β-pinene

Volume:12   Issue: 3
Pp: 241-249
Yanqing Gao*, Jian Li*, Shibin Shang and Dan Wang
DOI: 10.2174/1570180811666141009234615
Published on: 02 December, 2014