Letters in Drug Design & Discovery


Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo

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Volume: 12 Issue: 1, January 2014

Editorial free to download

Volume:12   Issue: 1
Pp: 1-1
DOI: 10.2174/157018081201141030111644
Published on: 30 October, 2014

Identification of Novel GSK1070916 Analogs as Potential Aurora B Inhibitors: Insights from Molecular Dynamics and MM/GBSA Based Rescoring

Volume:12   Issue: 1
Pp: 2-13
Faraz Shaikh, Soumendranath Bhakat, Abhishek Thakur, Ashish Radadiya, Mahmoud E. S. Soliman and Anamik Shah
DOI: 10.2174/1570180811666140725184953
Published on: 25 July, 2014

Design, Synthesis and Antimycobacterial Activity of Some New Azaheterocycles: Phenanthroline with p-halo-benzoyl Skeleton. Part V

Volume:12   Issue: 1
Pp: 14-19
Ramona Danac, Teofil Daniloaia, Vasilichia Antoci, Violeta Vasilache and Ionel I. Mangalagiu
DOI: 10.2174/1570180811666140819223501
Published on: 19 August, 2014

Design, Synthesis and Cytotoxic Evaluation of Novel Imatinib Amide Derivatives that Target Abl Kinase

Volume:12   Issue: 1
Pp: 20-28
Ri-Sheng Yao, Qiu-Xiang Guan, Xiao-Qin Lu and Ban-Feng Ruan
DOI: 10.2174/1570180811666140812231519
Published on: 12 August, 2014

Design, Synthesis and Antitubercular Evaluation of New 2-amino-5-(4- (benzyloxy)benzyl)thiophene-3-carboxylic Acid Derivatives. Part 3

Volume:12   Issue: 1
Pp: 29-37
Xiaoyun Lu, Jian Tang, Qidong You, Baojie Wan and Scott G. Franzblau
DOI: 10.2174/1570180811666140812231321
Published on: 12 August, 2014

Design, Synthesis and Biological Evaluation of Benzimidazole-pyridine- Piperidine Hybrids as a New Class of Potent Antimicrobial Agents

Volume:12   Issue: 1
Pp: 38-45
Kothapally. Beulah, Akula Ravi Kumara, Boddupally Peda Venkat Lingaiah, Pamulaparthy Shanthan Rao, Banda Narsaiah, Aaramadaka Sunil Kumar Reddy and Upadhyayula Surya Narayana Murty
DOI: 10.2174/1570180811666140725185713
Published on: 25 July, 2014

Structure Based Functional Annotation of Putative Conserved Proteins from Treponema pallidum: Search for a Potential Drug Target

Volume:12   Issue: 1
Pp: 46-59
Avni Sinha, Faizan Ahmad and Md. Imtaiyaz Hassan
DOI: 10.2174/1570180811666140806005822
Published on: 05 August, 2014

Theoretical Modelling of Potential Chk1 Inhibitors

Volume:12   Issue: 1
Pp: 60-65
Pedro M.M. Araujo, Luis Pinto da Silva and Joaquim C.G. Esteves da Silva
DOI: 10.2174/1570180811666140725190051
Published on: 25 July, 2014

A Screening Method for Potential Anti-pancreatic Cancer Candidate Compounds Based on Hsp90-Cdc37 Interaction Model in vitro

Volume:12   Issue: 1
Pp: 66-71
Hai Zhang, Sen Sun, Qingshan Chen, Guoqing Zhang, Zhenqing Zhang, Duxin Sun and Wenpeng Zhang
DOI: 10.2174/1570180811666140725185235
Published on: 25 July, 2014

Synthesis and Evaluation of Transdermal Permeation, Pharmacological Activity of Bornyl NSAID Esters

Volume:12   Issue: 1
Pp: 72-77
Jiufeng Lin, Kefeng Ni, Yang Zhang, Dongzhi Wei and Yuhong Ren
DOI: 10.2174/1570180811666140627004820
Published on: 26 June, 2014

Efficient Synthesis of Benzidronate Applying of Phosphorus Trichloride and Phosphorous Acid

Volume:12   Issue: 1
Pp: 78-84
Alajos Grun, Rita Kovacs, David Illes Nagy, Sandor Garadnay, Istvan Greiner and Gyorgy Keglevich
DOI: 10.2174/1570180811666141001004732
Published on: 30 September, 2014