Letters in Drug Design & Discovery


Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo

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Volume: 11 Issue: 9, November 2014

Modeling the Active Conformation of Human µ Opioid Receptor

Volume:11   Issue: 9
Pp: 1053-1061
Agnieszka A. Kaczor, Damian Bartuzi and Dariusz Matosiuk
DOI: 10.2174/1570180811666140322001506
Published on: 28 May, 2014

Synthesis and In vitro Evaluation of Thiadiazole Derivatives as AChE, Bu- ChE and LOX Inhibitors

Volume:11   Issue: 9
Pp: 1062-1069
Mehlika Dilek Altintop, Ahmet Ozdemir, Usama Abu Mohsen, Halide Edip Temel, Gulsen Akal n Ciftci and Zafer Asim Kaplancikli
DOI: 10.2174/1570180811666140529004517
Published on: 28 May, 2014

Synthesis and Studies on Anticonvulsant and Antibacterial Activities of 1- Alkyl-4-(4H-1,2,4-triazol-4-yl)piperidine Derivatives

Volume:11   Issue: 9
Pp: 1070-1078
Yan-Ping Yuan, Shi-Ben Wang, Guo-Hua Gong and Zhe-Shan Quan
DOI: 10.2174/1570180811666140623204022
Published on: 23 June, 2014

Design, Synthesis and Antitumor Activities of Bis-arylureas and Bis-arylamides Based on1H-benzo[d]imidazole Moiety as Novel BRafV600E/VEGFR2 Dual inhibitors

Volume:11   Issue: 9
Pp: 1079-1089
Weimin Yang, Yadong Chen, Yanmin Zhang, Sanzhi Tang, Hongli Chen, Weifang Tang and Tao Lu
DOI: 10.2174/1570180811666140724184806
Published on: 24 July, 2014

To Preliminarily Evaluate The Anticancer Activiy of 1,2-di(quinazolin-4- yl)diselane Against MDA-MB-435 Cells in vitro

Volume:11   Issue: 9
Pp: 1090-1095
Yinjiu Huang, Hong Xie, Gang Liu, Xiaomei Hu, Lin Su, Jianguo Hu, Qiyi Wang and Yibo Ding
DOI: 10.2174/1570180811666140617212723
Published on: 17 June, 2014

Evaluation of Alkylating and Intercalating Properties of Mannich Bases for Cytotoxic Activity

Volume:11   Issue: 9
Pp: 1096-1106
Huseyin Istanbullu, Yalcin Erzurumlu, Petek Ballar Kirmizibayrak and Ercin Erciyas
DOI: 10.2174/1570180811666140529005029
Published on: 28 May, 2014

Synthesis and Antifungal Activity of 1,3,4-Thiadiazole Derivatives Containing Pyridine Group

Volume:11   Issue: 9
Pp: 1107-1111
Lin-Jiong Zhang, Ming-Yan Yang, Zhao-Hui Sun, Cheng-Xia Tan, Jian-Quan Weng, Hong-Ke Wu and Xing-Hai Liu
DOI: 10.2174/1570180811666140610212731
Published on: 10 June, 2014

Pharmacokinetic Modeling of Caco-2 Cell Permeability Using Genetic Programming (GP) Method

Volume:11   Issue: 9
Pp: 1112-1118
Renu Vyas, Purva Goel, M. Karthikeyan, S.S. Tambe and B.D. Kulkarni
DOI: 10.2174/1570180811666140610213438
Published on: 10 June, 2014

Synthesis and Bioactivities of Novel 1,3,4-oxadiazole Derivatives Containing Pyridine Moiety

Volume:11   Issue: 9
Pp: 1119-1123
Guo-Xiang Sun, Yan-Xia Shi, Zhao-Hui Sun, Ming-Yan Yang, Hong-Ke Wu, Jian-Quan Weng, Cheng-Xia Tan, Xing-Hai Liu, Bao-Ju Li and Yong-Gang Zhang
DOI: 10.2174/1570180811666140522002929
Published on: 21 May, 2014

Solvent-Free Synthesis and Insecticidal Activities of C6-Esterified Coumarins

Volume:11   Issue: 9
Pp: 1124-1132
Ying Xie, Zheng-Lin Lei and Yan-Ping Luo
DOI: 10.2174/1570180811666140603003043
Published on: 02 June, 2014