Letters in Drug Design & Discovery

Editor-in-Chief

Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo
(Italy)

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Volume: 11 Issue: 1, January 2013

GRAPHICAL ABSTRACTS

Volume:11   Issue: 1
Pp: i-vii

DOI: 10.2174/157018081101131127104022
Published on: 26 November, 2013

Editorial

Volume:11   Issue: 1
Pp: 1-1
Atta- ur- Rahman
DOI: 10.2174/157018081101131127104153
Published on: 26 November, 2013

Synthesis of resveratrol acrylamides derivatives and biological evaluation of their anti-proliferative effect on cancer cell lines

Volume:11   Issue: 1
Pp: 2-9
Ban-Feng Ruan, Si-Qi Wang, Xiao-Lin Ge and Ri-Sheng Yao
DOI: 10.2174/15701808113109990057
Published on: 05 August, 2013

Anticancer Studies of Leucovorin against Methotrexate Induced Genotoxicity in Swiss Albino Mice

Volume:11   Issue: 1
Pp: 10-14
Chandra Sekhar Singh Bhaludra, Adharvana Chari Murugulla, Chakrapani Pullagummi, Ajay kumar Polkampally and Roja Rani Anupalli
DOI: 10.2174/15701808113109990052
Published on: 01 August, 2013

In Silico, Spectroscopic, and Biological Insights on Annelated Pyrrolo[3,2- e]Pyrimidines with Antiproliferative Activity

Volume:11   Issue: 1
Pp: 15-26
Antonino Lauria, Alessio Terenzi, Carla Gentile, Annamaria Martorana, Giuseppe Gennaro, Giampaolo Barone and Anna Maria Almerico
DOI: 10.2174/15701808113109990058
Published on: 05 August, 2013

Dimer and Tetramer of Gallic Acid: Facile Synthesis, Antioxidant and Antiproliferative Activities

Volume:11   Issue: 1
Pp: 27-32
Junzhu Pan, Dongqin Yin, Lifang Ma, Yi Zhao, Jing Zhao and Li Guo
DOI: 10.2174/15701808113109990032
Published on: 26 June, 2013

Improvement of Virtual Screening Predictions using Computational Intelligence Methods

Volume:11   Issue: 1
Pp: 33-39
Gaspar Cano, José García-Rodríguez and Horacio Pérez-Sánchez
DOI: 10.2174/15701808113109990054
Published on: 01 August, 2013

Virtual Screening and Molecular Descriptor Analysis on Dietary Phytochemicals Against Heat Shock Protein 90 Enzyme

Volume:11   Issue: 1
Pp: 40-49
Salam Pradeep Singh and Bolin Kumar Konwar
DOI: 10.2174/15701808113109990044
Published on: 16 July, 2013

The Docking Based 3D-QSAR Studies on Isoindolinone Derived Inhibitors of p53-MDM2 Binding

Volume:11   Issue: 1
Pp: 50-58
Huazhou Ying, Chunlei Wu and Chunqi Hu
DOI: 10.2174/15701808113109990053
Published on: 01 August, 2013

A QSAR Study of the Acrylpimaric Acid Derivatives as the Inhibitors of NCI-H460

Volume:11   Issue: 1
Pp: 59-66
Jian Li, Guomin Xiao, Shibin Shang and Xiaoping Rao
DOI: 10.2174/15701808113109990062
Published on: 19 August, 2013

Antifungal Activity of a Library of Cyclitols and Related Compounds

Volume:11   Issue: 1
Pp: 67-75
Ana Bellomo, Ana Bertucci, Victoria de la Sovera, Gonzalo Carrau, Marcela Raimondi, Susana Zacchino, Helio A. Stefani and David Gonzalez
DOI: 10.2174/15701808113109990036
Published on: 08 July, 2013

Synthesis and Antimicrobial Activity of New Pyrimidine-Hydrazones

Volume:11   Issue: 1
Pp: 76-81
Zafer Asım Kaplancıklı, Leyla Yurttas, Gülhan Turan-Zitouni, Ahmet Özdemir, Gamze Göger, Fatih Demirci and Usama Abu Mohsen
DOI: 10.2174/15701808113109990037
Published on: 08 July, 2013

Design, Green Synthesis, and Anti-Inflammatory Activity of Schiff Base of 1,3,4-oxadiazole Analogues

Volume:11   Issue: 1
Pp: 82-89
Biswa Mohan Sahoo, Subas Chandra Dinda, BVV Ravi Kumar, Jnyanaranjan Panda and Pathik S Brahmkshatriya
DOI: 10.2174/15701808113109990041
Published on: 09 July, 2013

Biological Evaluation of Imidazobenzoxazines, Imidazobenzoxazin-5-ones and Imidazobenzoxazin-5-thiones as Sodium Channel Blockers

Volume:11   Issue: 1
Pp: 90-97
Mirko Rivara, Valentina Zuliani and Manoj K. Patel
DOI: 10.2174/15701808113109990050
Published on: 01 August, 2013

Synthesis and Bio-Evaluation of Novel Salicylic Acid-Oriented Thiourea Derivatives with Potential Applications in Agriculture

Volume:11   Issue: 1
Pp: 98-103
Shaowei Li, Huangyong Li, Xiufang Cao and Changshui Chen
DOI: 10.2174/15701808113109990045
Published on: 23 July, 2013

Synthesis and Characterization of Furo[3,2-h]Quinoliniums as Potent Non- Detergent Spermicides

Volume:11   Issue: 1
Pp: 104-113
Maitreyee Banerjee, Shrabanti Kumar, Rupankar Paira, Soma Ghosh, Sanmoy Karmakar and Nirup B Mondal
DOI: 10.2174/15701808113109990046
Published on: 23 July, 2013

O-Arylation of Iodophenols with 2-Fluorobenzaldehyde Under Microwave Conditions

Volume:11   Issue: 1
Pp: 114-120
Erika Bálint, Mónika Kállai, Orsolya Kovács, Hedvig Bölcskei and György Keglevich
DOI: 10.2174/15701808113106660096
Published on: 29 October, 2013