ISSN (Print): 1570-1808 ISSN (Online): 1875-628X Volume 18, 12 Issues, 2021
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ISSN (Print): 1570-1808 ISSN (Online): 1875-628X
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"Letters in Drug Design & Discovery should be available in every library in the pharmaceutical industry and in universities." R. F. Borne, Associate Director Laboratory for Applied Drug Design and Synthesis, The University of Mississippi, USA
I would like to thank Bentham Science Publishers for their peerless effort to keep up scientists and students updated with the latest science and research work. Actually, Bentham assists researchers to achieve their goals to spread their reputation worldwide. I have experienced sincere, efficient and effective communication while dealing with Bentham team members. I intend to submit my work to Bentham and try to pick up journals that match my research profile. I have submitted a recent work to Medicinal Chemistry and nowadays I am drafting a manuscript targeting Current Pharmaceutical Design. Honestly, no words neither sentences would express my gratefulness and admiration. Bentham has offered my institution three months trial to access their journal lists and surf on its Board. This free access trial fulfills my literature review and broadens my horizon to absorb the recent research in pharmaceutical sciences and medicinal chemistry. Finally, I wish Bentham more success and achievement!
Has contributed: CETP Inhibitory Activity of Chlorobenzyl Benzamides: QPLD Docking, Pharmacophore Mapping and Synthesis.
Synthesis of Novel 3-(4-tert-Butylphenyl)-5-Cylopropyl-4H-1,2,4-Triazole Derivatives with Antioxidative and Antimicrobial Activities
Volume:17 Issue:8 Pp: 954-964 Nuri Yildirim* DOI: 10.2174/1570180817999200424073524
(Substituted)-benzo[b]thiophene-4-carboxamide Synthesis and Antiproliferative Activity Study
Volume:17 Issue:5 Pp: 563-573 Chandrakant Dhondiram Pawar, Dattatraya Navnath Pansare and Devanand Baburao Shinde* DOI: 10.2174/1570180815666181004114125
Lead Molecules as Novel Aromatase Inhibitors: In Silico De Novo Designing and Binding Affinity Studies
Volume:17 Issue:5 Pp: 655-665 Laxmi Banjare, Sant Kumar Verma, Akhlesh Kumar Jain and Suresh Thareja* DOI: 10.2174/1570180816666190703152659
New 2-Oxopyridine/2-Thiopyridine Derivatives Tethered to a Benzotriazole with Cytotoxicity on MCF7 Cell Lines and with Antiviral Activities
Volume:17 Issue:2 Pp: 124-137 Adel Mahmoud Attia, Ahmed Ibrahin Khodair*, Eman Abdelnasser Gendy, Mohammed Abu El-Magd and Yaseen Ali Mosa Mohamed Elshaier* DOI: 10.2174/1570180816666190220123547
Synthesis and Antimicrobial Activity of Thiohydantoins Obtained from L-Amino Acids
Volume:17 Issue:1 Pp: 94-102 Priscila Goes Camargo de Carvalho, Jhonatan Macedo Ribeiro, Renata Perugini Biasi Garbin, Gerson Nakazato, Sueli Fumie Yamada Ogatta, Ângelo de Fátima, Marcelle de Lima Ferreira Bispo and Fernando Macedo* DOI: 10.2174/1570180816666181212153011
QSAR Analysis of Selected Antimicrobial Structures Belonging to Nitro-derivatives of Heterocyclic Compounds
Volume:17 Issue:2 Pp: 214-225 Piotr Kawczak*, Leszek Bober and Tomasz Bączek DOI: 10.2174/1570180815666181004112947
Aminoalkylated Phenolic Chalcones: Investigation of Biological Effects on Acetylcholinesterase and Carbonic Anhydrase I and II as Potential Lead Enzyme Inhibitors
Volume:17 Issue:10 Pp: 1283-1292 Cem Yamali*, Halise Inci Gul*, Tahir Cakir, Yeliz Demir and Ilhami Gulcin DOI: 10.2174/1570180817999200520123510
Novel Coronavirus (COVID-19) Outbreak: Hope and Search for Effective Therapeutic Agent promotion: free to download
Volume:17 Issue:8 Pp: 940-942 Saurabh Kumar* DOI: 10.2174/1570180817999200612095513
An Environment-friendly Synthesis of Piperonal Chalcones and Their Cytotoxic and Antioxidant Evaluation
Volume:17 Issue:2 Pp: 138-144 Sanal Dev, Della Grace Thomas Parambi, Bency Baby, Githa Elizabeth Mathew, Hendawy Omnia Magdy, Monu Joy, Shine Sudev and Bijo Mathew* DOI: 10.2174/1570180815666181016155934
Synthesis of Piperidine Conjugated Dihydroquinazolin-4(1H)-ones and their Antiproliferative Activity, Molecular Docking Studies and DFT Calculations open access plus
Volume:17 Issue:1 Pp: 85-93 Kereyagalahally Honneshappa Narasimhamurthy, Chandra, Toreshettahally Ramesh Swaroop, Swamy Jagadish and Kanchugarakoppal Subbegowda Rangappa* DOI: 10.2174/1570180816666190613120349
Antimicrobial Activity, Antioxidant Properties and Phytochemical Screening of Aesculus hippocastanum Mother Tincture against Food-borne Bacteria
Volume:17 Issue:1 Pp: 48-56 Maria Grazia Bonomo*, Caterina Cafaro, Daniela Russo, Luana Calabrone, Luigi Milella, Carmela Saturnino, Anna Capasso and Giovanni Salzano DOI: 10.2174/1570180816666181108114115
One-pot Synthesis of Betulin Triterpenoid Quaternized Pyridine Derivatives and their Antimicrobial Activity
Volume:17 Issue:1 Pp: 79-84 Elvira Rifovna Shakurova, Darina Alexandrovna Pozdnyakova, Elena Valeryevna Tretyakova and Lyudmila Vyacheslavovna Parfenova* DOI: 10.2174/1570180816666181217123629
The 2019 Novel Coronavirus (COVID-19) Outbreak in China and World: A New Lesson for Public Health System promotion: free to download
Volume:17 Issue:4 Pp: 364-365 Kamil Kuca DOI: 10.2174/157018081704200310125801
Synthesis of Limonin Derivatives with Improved Anti-inflammatory and Analgesic Properties open access plus
Volume:17 Issue:3 Pp: 285-299 Chengshu Jia, Bin Hu, Yingying Ji, Yourui Su, Guoqing Gong, Qihua Zhu and Yungen Xu* DOI: 10.2174/1570180816666181113102359
Cephalosporin Conjugated Sulfonamides: Synthesis, Characterization and Anticancer Activities
Volume:17 Issue:3 Pp: 264-270 Rana Asif Nadeem, Muhammad Abdul Qadir, Mahmood Ahmed* and Imran Sajid DOI: 10.2174/1570180815666180820144621
Synthesis, In Silico and In Vivo Evaluation of Novel 1, 3, 4-Thiadiazole Analogues as Novel Anticancer Agents
Volume:17 Issue:4 Pp: 434-444 Swathi Krishna, Byran Gowramma*, Manal Mohammed, Rajagopal Kalirajan, Lakshman Kaviarasan and Thaggikuppe Krishnamurthy Praveen* DOI: 10.2174/1570180816666190710145939
Anti-Trypanosoma cruzi Activity and Molecular Docking Studies of 1Hpyrazolo[ 3, 4-b]pyridine Derivatives
Volume:17 Issue:2 Pp: 184-191 Camilo Henrique da Silva Lima, Júlio César de Araujo Vanelis Soares, Joana Lucius de Sousa Ribeiro, Estela Maris Freitas Muri, Sérgio de Albuquerque and Luiza Rosaria Sousa Dias* DOI: 10.2174/1570180816666190305141733
Identifying the Structural Features of Diphenyl Ether Analogues for InhA Inhibition: A 2D and 3D QSAR Based Study open access plus
Volume:17 Issue:1 Pp: 31-47 Ashutosh Prasad Tiwari, Varadaraj Bhat Giliyar*, Gurypur Gautham Shenoy and Vandana Kalwaja Eshwara DOI: 10.2174/1570180816666190611153933
Melatonin Ameliorates Radiation-induced Sciatic Nerve Injury
Volume:17 Issue:1 Pp: 21-30 Dheyauldeen Shabeeb*, Ahmed Eleojo Musa, Mansoor Keshavarz, Gholamreza Hassanzadeh, Mohammed Reza Hadian, Azin Nowrouzi, Alireza Shirazi* and Masoud Najafi DOI: 10.2174/1570180816666190617160434
Fingerprint-based 2D-QSAR Models for Predicting Bcl-2 Inhibitors Affinity
Volume:17 Issue:10 Pp: 1206-1215 Said Byadi, Hachim Mouhi Eddine, Karima Sadik, Črtomir Podlipnik and Aziz Aboulmouhajir* DOI: 10.2174/1570180817999200414155403
Design, Synthesis, In vitro and In silico Evaluation of New Hydrazonebased Antitumor Agents as Potent Akt Inhibitors
Volume:17 Issue:11 Pp: 1380-1392 Emine Merve Güngör, Mehlika Dilek Altıntop*, Belgin Sever and Gülşen Akalın Çiftçi DOI: 10.2174/1570180817999200618163507
Synthesis and Biological Evaluation of Benzodioxol Derivatives as Cyclooxygenase Inhibitors
Volume:17 Issue:9 Pp: 1117-1125 Nidal Jaradat*, Mohammed Hawash and Murad Abualhasan DOI: 10.2174/1570180817999200420114402
Natural Sesquiterpene Lactones in the Prevention and Treatment of Inflammatory Disorders and cancer: A Systematic Study of this Emerging Therapeutic Approach based on Chemical and Pharmacological Aspect
Volume:17 Issue:9 Pp: 1102-1116 Sudip Kumar Mandal, Utsab Debnath, Amresh Kumar, Sabu Thomas, Subhash Chandra Mandal, Manabendra Dutta Choudhury and Partha Palit* DOI: 10.2174/1570180817999200421144007
Molecular Docking and QSAR Studies of Coumarin Derivatives as NMT Inhibitors: Simple Structural Features as Potential Modulators of Antifungal Activity
Volume:17 Issue:10 Pp: 1293-1308 Sapna Jain Dabade, Dheeraj Mandloi* and Amritlal Bajaj DOI: 10.2174/1570180817999200617105711
Searching for Potential HDAC2 Inhibitors: Structure-activity Relationship Studies on Indole-based Hydroxamic Acids as an Anticancer Agent
Volume:17 Issue:7 Pp: 905-917 Ekta Shirbhate, Divya, Preeti Patel, Vijay K. Patel, Ravichandran Veerasamy, Prabodh C. Sharma and Harish Rajak* DOI: 10.2174/1570180817666200103125701
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