Medicinal Chemistry

Editor-in-Chief

Dimitra Hadjipavlou-Litina
Aristotle University of Thessaloniki
Thessaloniki
(Greece)

Nobel Laureate on Editorial Board

Prof. Ferid Murad
(USA)

Personal Subscription
Become EABM
Become Reviewer



Meet Our Editorial Board Member free to download

Volume:14   Issue: 7
Pp: 651-651
Roberta Ettari
DOI: 10.2174/157340641407180815113743



Design, Synthesis and Biological Evaluation of New 1,3-diphenyl-3- (phenylamino)propan-1-ones as Selective Cyclooxygenase (COX-2) Inhibitors

Volume:14   Issue: 7
Pp: 652-659
Shabnam Farzaneh, Soraya Shahhosseini, Hadi Arefi, Bahram Daraei, Marjan Esfahanizadeh and Afshin Zarghi*
DOI: 10.2174/1573406414666180525133221




Synthesis, Cyclooxygenase-2 Inhibition, Anti-inflammatory Evaluation and Docking Study of Substituted-N-(3,4,5-trimethoxyphenyl)-benzo[d]oxazole Derivatives

Volume:14   Issue: 7
Pp: 660-673
Avneet Kaur, Sharad Wakode*, Dharam P. Pathak, Vidushi Sharma and Ashok K. Shakya
DOI: 10.2174/1573406414666180322091832




Diclofenac 1,3,4-Oxadiazole Derivatives; Biology-Oriented Drug Synthesis (BIODS) in Search of Better Non-Steroidal, Non-Acid Antiinflammatory Agents

Volume:14   Issue: 7
Pp: 674-687
Shazia Shah, Arshia, Nida Siraj Kazmi, Almas Jabeen, Aisha Faheem, Nida Dastagir, Tariq Ahmed, Khalid Mohammed Khan*, Shakil Ahmed, Abeer Raza and Shahnaz Perveen
DOI: 10.2174/1573406414666180321141555




An Expedient Synthesis of CMF-019: (S)-5-Methyl-3-{1-(pentan-3-yl)-2- (thiophen-2-ylmethyl)-1H-benzo[d]imidazole-5-carboxamido}hexanoic Acid, a Potent Apelin Receptor (APJ) Agonist

Volume:14   Issue: 7
Pp: 688-694
Lena Trifonov, Michal Afri, Krzysztof Palczewski, Edward E. Korshin* and Arie Gruzman*
DOI: 10.2174/1573406414666180412154952




Benzoin Schiff Bases: Design, Synthesis, and Biological Evaluation as Potential Antitumor Agents

Volume:14   Issue: 7
Pp: 695-708
Dima A. Sabbah*, Fatima Al-Tarawneh, Wamidh H. Talib, Kamal Sweidan, Sanaa K. Bardaweel, Eveen Al-Shalabi, Haizhen A. Zhong, Ghassan Abu Sheikha, Reema Abu Khalaf and Mohammad S. Mubarak
DOI: 10.2174/1573406414666180412160142




Synthesis of a Tyr-Tyr Dipeptide Library and Evaluation Against Tumor Cells

Volume:14   Issue: 7
Pp: 709-714
Stanley N.S. Vasconcelos, Juliana M. Sciani, Nicole M. Lisboa and Helio A. Stefani*
DOI: 10.2174/1573406414666180309153142




Inhibition of Mutated Isocitrate Dehydrogenase 1 in Cancer

Volume:14   Issue: 7
Pp: 715-724
Fangrui Wu, Gang Cheng, Yuan Yao, Mari Kogiso, Hong Jiang, Xiao-Nan Li and Yongcheng Song*
DOI: 10.2174/1573406414666180524093659




Synthesis of Thiocarbohydrazones and Evaluation of their in vitro Antileishmanial Activity

Volume:14   Issue: 7
Pp: 725-732
Munira T. Muhammad, Nida Ghouri, Khalid M. Khan*, Arshia, Muhammad I. Choudhary* and Shahnaz Perveen
DOI: 10.2174/1573406414666180115094630




QSAR and Pharmacophore Mapping Studies on Benzothiazinimines to Relate their Structural Features with anti-HIV Activity

Volume:14   Issue: 7
Pp: 733-740
Gopiraja Geethaavacini, Go Poh Poh, Lim Yi Yan, Rajindran Deepashini , Sivadasan Shalini, Rajak Harish, Krishnan Sureshkumar and Veerasamy Ravichandran*
DOI: 10.2174/1573406414666180529091618




Design of Bactericidal Peptides Against Escherichia coli O157:H7, Pseudomonas aeruginosa and methicillin-resistant Staphylococcus aureus

Volume:14   Issue: 7
Pp: 741-752
Jenniffer Cruz, Paola Rondon-Villarreal, Rodrigo G. Torres, Mauricio Urquiza, Fanny Guzman, Claudio Alvarez, Maria A. Abengozar, Daniel A. Sierra, Luis Rivas, Roberto Fernandez-Lafuente and Claudia C. Ortiz*
DOI: 10.2174/1573406414666180508120024