Medicinal Chemistry

Editor-in-Chief

Dimitra Hadjipavlou-Litina
Aristotle University of Thessaloniki
Thessaloniki
(Greece)

Nobel Laureate on Editorial Board

Prof. Ferid Murad
(USA)

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Application of Bioinformatics in Search for Cleavable Peptides of SARSCoV Mpro and Chemical Modification of Octapeptides

Volume:1   Issue: 3
Pp: 209-213
Qishi Du, Shuqing Wang, Zhiqin Jiang, Weina Gao, Yun Li, Dongqing Wei and Kuo-Chen Chou
DOI: 10.2174/1573406053765468

Variously Substituted (Phosphonoacetamido)Oxy Analogues of Geranylgeranyl Diphosphate (GGdP) as GGdP-transferase (GGTase) Inhibitors and Antiproliferative Agents

Volume:1   Issue: 3
Pp: 239-244
Filippo Minutolo, Valentina Asso, Simone Bertini, Laura Betti, Massimiliano Ciriaco, Romano Danesi, Gianbattista Gervasi, Elisa Ghilardi, Elisa Giovanetti and Gino Giannaccini
DOI: 10.2174/1573406053765512

Synthesis and Biological Evaluation of 2-, 3-, and 4-Acylaminocinnamyl-Nhydroxyamides as Novel Synthetic HDAC Inhibitors

Volume:1   Issue: 3
Pp: 245-254
A. Mai, S. Massa, R. Pezzi, S. Valente, P. Loidl and G. Brosch
DOI: 10.2174/1573406053765431

Synthesis and Evaluation of a Novel Gene Reporter Molecule: Detection of b-galactosidase Activity Using 19F NMR of a Fluorinated Vitamin B6 Conjugate+

Volume:1   Issue: 3
Pp: 255-262
Jianxin Yu, Zhenyi Ma, Yingming Li, Kenneth S. Koeneman, Li Liu and Ralph P. Mason
DOI: 10.2174/1573406053765495

Discovery of HIV-1 Integrase Inhibitors through a Novel Combination of Ligand and Structure-based Drug Design

Volume:1   Issue: 3
Pp: 263-275
A. Brigo, G. Iurcu Mustata, J. M. Briggs and S. Moro
DOI: 10.2174/1573406053765440

Evaluation of Hyperforin Analogues for Inhibition of 5-lipoxygenase

Volume:1   Issue: 3
Pp: 287-291
Christian Feißt, Dana Albert, Luisella Verotta and Oliver Werz
DOI: 10.2174/1573406053765503

Protein Phosphorylation and Signal Transduction Modulation: Chemistry Perspectives for Small-Molecule Drug Discovery

Volume:1   Issue: 3
Pp: 293-319
T. K. Sawyer, W. C. Shakespeare, Y. Wang, R. Sundaramoorthi, W. S. Huang, C. A. Metcalf III, M. Thomas, B. M. Lawrence, L. Rozamus and J. Noehre
DOI: 10.2174/1573406053765486