Current Organic Synthesis

One-Pot Green Synthesis of Acridine Alkaloid Derivatives and Screening of in vitro Anti-cancer Activity Against Cdc25b and SHP1

Volume: 18   Issue: 4
Pp: 399-405
Hao Li, Buer Song, Mamtimin Mahmut* and Mukhtar Imerhasan*
DOI: 10.2174/1570179417666201228165500

Catalyst-free Synthesis of Aminomethylphenol Derivatives in Cyclopentyl Methyl Ether via Petasis Borono-Mannich Reaction

Volume: 18   Issue: 3
Pp: 294-300
Jia-Qi Di, Hao-Jie Wang, Zhen-Shui Cui, Jin-Yong Hu* and Zhan-Hui Zhang*
DOI: 10.2174/1570179417666201216161143

Applications of the Dess-Martin Oxidation in Total Synthesis of Natural Products

Volume: 18   Issue: 2
Pp: 125-196
Majid M. Heravi*, Tayebe Momeni, Vahideh Zadsirjan* and Leila Mohammadi
DOI: 10.2174/1570179417666200917102634

An Overview of Recent Development in Visible Light-mediated Organic Synthesis over Heterogeneous Photo-nanocatalysts

Volume: 18   Issue: 1
Pp: 23-36
Yasser Mahmoud A. Mohamed*, Yasser A. Attia, Hossam A. El Nazer and Eirik Johansson Solum
DOI: 10.2174/1570179417666201005145103

Direct Gas-Phase Oxidation of Propylene to Acetone in the Presence of H₂ and O₂ over Au/TS-1 Catalyst promotion: free to download

Volume: 17   Issue: 8
Pp: 685-690
Jinsong Fu, Xiaoming Zhang*, Wuyang Liang, Qian Lei, Bing Sun, Wujun He and Guowei Deng*
DOI: 10.2174/1570179417666200615154837

Short Protecting Group-free Syntheses of CDE Synthon of Racemic Camptothecin

Volume: 17   Issue: 7
Pp: 588-591
Pingxuan Shao, Wei Lu and Lei Wang*
DOI: 10.2174/1570179417666200611125740

Green Solvent: Green Shadow on Chemical Synthesis

Volume: 17   Issue: 6
Pp: 426-439
Tejaswini Sahoo, Jagannath Panda, Jnanaranjan Sahu, Dayananda Sarangi, Sunil K. Sahoo, Braja. B. Nanda and Rojalin Sahu*
DOI: 10.2174/1570179417666200506102535

Eco-friendly and Enantiospecific Biginelli Synthesis Using (+)-Myrtenal as the Substrate – An Impeccable and Unequivocal Analysis of the Product

Volume: 17   Issue: 5
Pp: 389-395
Luiza Albino Dias Benincá, Carolina Bastos Pereira Ligiéro, Jonas da Silva Santos, Joel Jones Junior* and Flavia Martins da Silva
DOI: 10.2174/1570179417666200506103137

Electrophilic Aromatic Synthesis of Radioiodinated Aripiprazole: Experimental and DFT Investigations

Volume: 17   Issue: 4
Pp: 295-303
Moustapha E. Moustapha, Mohammed H. Geesi, Zeinab R. Farag and El Hassane Anouar*
DOI: 10.2174/1570179417666200409145824

A New Synthesis of Poly Heterocyclic Compounds Containing [1,2,4]triazolo and [1,2,3,4]tetrazolo Moieties and their DFT Study as Expected Anti-cancer Reagents

Volume: 17   Issue: 3
Pp: 211-223
El-sayed M. Abdelrehim * and Doaa S. El-Sayed
DOI: 10.2174/1570179417666200226092516

Synthesis, Docking Study, Cytotoxicity, Antioxidant, and Anti-microbial Activities of Novel 2,4-Disubstituted Thiazoles Based on Phenothiazine

Volume: 17   Issue: 2
Pp: 151-159
Tran Nguyen Minh An*, Pham Thai Phuong, Nguyen Minh Quang, Nguyen Van Son, Nguyen Van Cuong, Le Van Tan, Mai Dinh Tri, Mahboob Alam and Pham Van Tat
DOI: 10.2174/1570179417666191220100614

Revision of the Regioselectivity of the Beirut Reaction of Monosubstituted Benzofuroxans with Benzoylacetonitrile. 6-Substituted quinoxaline-2-carbonitrile 1,4- dioxides: Structural Characterization and Estimation of Anticancer Activity and Hypoxia Selectivity

Volume: 17   Issue: 1
Pp: 29-39
Galina I. Buravchenko, Alexander M. Scherbakov, Alexander А. Korlukov, Pavel V. Dorovatovskii and Andrey E. Shchekotikhin*
DOI: 10.2174/1570179416666191210100754

Unexpected Reactions of Terminal Alkynes in Targeted “Click Chemistry’’ Coppercatalyzed Azide-alkyne Cycloadditions

Volume: 16   Issue: 8
Pp: 1143-1148
Tammar H. Ali*, Thorsten Heidelberg*, Rusnah S.D. Hussen and Hairul A. Tajuddin
DOI: 10.2174/1570179416666191105152714

Polymer-Bound Triphenylphosphine and 4,4′-Dinitroazobenzene as a Coupling Reagents for Chromatography-Free Esterification Reaction

Volume: 16   Issue: 7
Pp: 1024-1031
Diparjun Das, Kalyani Rajkumari and Lalthazuala Rokhum*
DOI: 10.2174/1570179416666190919152424

Novel Heterocyclic Hybrids Based on 2-Pyrazoline: Synthesis and Assessment of Anti-Inflammatory and Analgesic Activities

Volume: 16   Issue: 6
Pp: 921-930
Ahmed A.O. Abeed, Gehad A.A. Jaleel and Mohamed S.K. Youssef*
DOI: 10.2174/1570179416666190703115133

Preparation of Carbon-14 Labeled 2-(2-mercaptoacetamido)-3-phenylpropanoic Acid as Metallo-beta-lactamases Inhibitor (MBLI), for Coadministration with Beta-lactam Antibiotics

Volume: 16   Issue: 5
Pp: 765-771
Ali Maleki*, Reza Taheri-Ledari, Reza Eivazzadeh-Keihan, Miguel de la Guardia and Ahad Mokhtarzadeh*
DOI: 10.2174/1570179416666190423114704

The History of the Glycosidase Inhibiting Hyacinthacine C-type Alkaloids: From Discovery to Synthesis. open access plus

Volume: 16   Issue: 4
Pp: 498-522
Anthony W. Carroll* and Stephen G. Pyne*
DOI: 10.2174/1570179416666190126100312

How to Start a Total Synthesis from the Wieland-Miescher Ketone?

Volume: 16   Issue: 3
Pp: 328-341
Zai-Qun Liu *
DOI: 10.2174/1570179416666190328233710

Alkynes as Privileged Synthons in Selected Organic Name Reactions

Volume: 16   Issue: 2
Pp: 205-243
Majid M. Heravi*, Mahzad Dehghani, Vahideh Zadsirjan* and Manijheh Ghanbarian
DOI: 10.2174/1570179416666190126100744

Highly Selective Gold-Catalyzed Cycloisomerization of Furanolabdanoid Dialkynes with Alkynyl Substituents in the Furan Ring

Volume: 15   Issue: 8
Pp: 1147-1153
Yurii V. Kharitonov , Makhmut M. Shakirov and Elvira E. Shults*
DOI: 10.2174/1570179415666180918160421