Current Organic Synthesis

A New Synthesis of Poly Heterocyclic Compounds Containing [1,2,4]triazolo and [1,2,3,4]tetrazolo Moieties and their DFT Study as Expected Anti-cancer Reagents

Volume: 17   Issue: 3
Pp: 211-223
El-sayed M. Abdelrehim * and Doaa S. El-Sayed
DOI: 10.2174/1570179417666200226092516

Synthesis, Docking Study, Cytotoxicity, Antioxidant, and Anti-microbial Activities of Novel 2,4-Disubstituted Thiazoles Based on Phenothiazine

Volume: 17   Issue: 2
Pp: 151-159
Tran Nguyen Minh An*, Pham Thai Phuong, Nguyen Minh Quang, Nguyen Van Son, Nguyen Van Cuong, Le Van Tan, Mai Dinh Tri, Mahboob Alam and Pham Van Tat
DOI: 10.2174/1570179417666191220100614

Revision of the Regioselectivity of the Beirut Reaction of Monosubstituted Benzofuroxans with Benzoylacetonitrile. 6-Substituted quinoxaline-2-carbonitrile 1,4- dioxides: Structural Characterization and Estimation of Anticancer Activity and Hypoxia Selectivity

Volume: 17   Issue: 1
Pp: 29-39
Galina I. Buravchenko, Alexander M. Scherbakov, Alexander А. Korlukov, Pavel V. Dorovatovskii and Andrey E. Shchekotikhin*
DOI: 10.2174/1570179416666191210100754

Unexpected Reactions of Terminal Alkynes in Targeted “Click Chemistry’’ Coppercatalyzed Azide-alkyne Cycloadditions

Volume: 16   Issue: 8
Pp: 1143-1148
Tammar H. Ali*, Thorsten Heidelberg*, Rusnah S.D. Hussen and Hairul A. Tajuddin
DOI: 10.2174/1570179416666191105152714

Polymer-Bound Triphenylphosphine and 4,4′-Dinitroazobenzene as a Coupling Reagents for Chromatography-Free Esterification Reaction

Volume: 16   Issue: 7
Pp: 1024-1031
Diparjun Das, Kalyani Rajkumari and Lalthazuala Rokhum*
DOI: 10.2174/1570179416666190919152424

Novel Heterocyclic Hybrids Based on 2-Pyrazoline: Synthesis and Assessment of Anti-Inflammatory and Analgesic Activities

Volume: 16   Issue: 6
Pp: 921-930
Ahmed A.O. Abeed, Gehad A.A. Jaleel and Mohamed S.K. Youssef*
DOI: 10.2174/1570179416666190703115133

Preparation of Carbon-14 Labeled 2-(2-mercaptoacetamido)-3-phenylpropanoic Acid as Metallo-beta-lactamases Inhibitor (MBLI), for Coadministration with Beta-lactam Antibiotics

Volume: 16   Issue: 5
Pp: 765-771
Ali Maleki*, Reza Taheri-Ledari, Reza Eivazzadeh-Keihan, Miguel de la Guardia and Ahad Mokhtarzadeh*
DOI: 10.2174/1570179416666190423114704

The History of the Glycosidase Inhibiting Hyacinthacine C-type Alkaloids: From Discovery to Synthesis. open access plus

Volume: 16   Issue: 4
Pp: 498-522
Anthony W. Carroll* and Stephen G. Pyne*
DOI: 10.2174/1570179416666190126100312

How to Start a Total Synthesis from the Wieland-Miescher Ketone?

Volume: 16   Issue: 3
Pp: 328-341
Zai-Qun Liu *
DOI: 10.2174/1570179416666190328233710

Alkynes as Privileged Synthons in Selected Organic Name Reactions

Volume: 16   Issue: 2
Pp: 205-243
Majid M. Heravi*, Mahzad Dehghani, Vahideh Zadsirjan* and Manijheh Ghanbarian
DOI: 10.2174/1570179416666190126100744

Highly Selective Gold-Catalyzed Cycloisomerization of Furanolabdanoid Dialkynes with Alkynyl Substituents in the Furan Ring

Volume: 15   Issue: 8
Pp: 1147-1153
Yurii V. Kharitonov , Makhmut M. Shakirov and Elvira E. Shults*
DOI: 10.2174/1570179415666180918160421

Double C–H Activation for the C–C bond Formation Reactions

Volume: 15   Issue: 7
Pp: 882-903
Jialin Liu, Xiaoyu Xiong, Jie Chen, Yuntao Wang, Ranran Zhu* and Jianhui Huang*
DOI: 10.2174/1570179415666180720111422

Reductive Amination/Alkylation Reactions: The Recent Developments, Progresses, and Applications in Protein Chemical Biology Studies

Volume: 15   Issue: 6
Pp: 755-761
Zhipeng A. Wang*, Yan-Yu Liang and Ji-Shen Zheng*
DOI: 10.2174/1570179415666180522093905

Pericyclic Reactions in the Syntheses of Densely Functionalized Heterocylces

Volume: 15   Issue: 4
Pp: 438-486
Rabia Qamar and Aamer Saeed*
DOI: 10.2174/1570179414666171025144740

A Straightforward Synthesis of 4,7-Disubstituted 1,4-Oxazepanes via a Bronsted Acid-Catalyzed Intramolecular Etherification Reaction

Volume: 15   Issue: 3
Pp: 370-379
Juan-Carlos Castillo, Jaime Portilla, Braulio Insuasty, Jairo Quiroga and Rodrigo Abonia*
DOI: 10.2174/1570179414666171011160917

Synthesis and Antitumor Evaluation of Novel N-substituted Norcantharidin Imidazolium Derivatives

Volume: 15   Issue: 2
Pp: 237-245
Rong-Rong Sun, Jia-Hui Guo, Cui Yang, Li-Juan Yang* and Chao Huang*
DOI: 10.2174/1570179414666170824160901

First Total Synthesis of Pamamycin-621D

Volume: 15   Issue: 1
Pp: 105-109
Hassan Norouzi-Arasi, Xavier J. Salom-Roig, Steve Lanners* and Gilles Hanquet*
DOI: 10.2174/1570179414666170525103947

Oxazolidine- and Oxazoline-2-thiones: An Update

Volume: 14   Issue: 8
Pp: 1109-1131
Estibaliz Sansinenea*, Aurelio Ortiz, Patrick Rollin and Sandrina Silva*
DOI: 10.2174/1570179414666170503165413

Photochemical Reactions: Synthesis of Six-membered N-heterocycles

Volume: 14   Issue: 7
Pp: 972-998
Navjeet Kaur*
DOI: 10.2174/1570179414666170201150701

Diversifying Polyhydroxyalkanoates – End-Group and Side-Chain Functionality

Volume: 14   Issue: 6
Pp: 757-767
Michal Michalak*, Iwona Kwiecien, Michal Kwiecien, Grazyna Adamus, Karin Odelius, Minna Hakkarainen and Piotr Kurcok*
DOI: 10.2174/1570179414666161115150146

A Review on Advances in Organoborane-Chemistry: Versatile Tool in Asymmetric Synthesis

Volume: 14   Issue: 5
Pp: 665-682
Paranjeet Kaur, Gopal L. Khatik* and Surendra Kumar Nayak
DOI: 10.2174/1570179414666161104162038

Diversity and Chemoselectivity in the Acid-Catalyzed Rearrangements of N,N’- Diarylhydrazines

Volume: 14   Issue: 4
Pp: 511-530
Jiaxi Xu*
DOI: 10.2174/1570179413666161021103952

Constructing Heterocycles by Visible Light Photocatalysis

Volume: 14   Issue: 3
Pp: 398-429
Maria E. Buden, Javier I. Bardagi and Roberto A. Rossi
DOI: 10.2174/1570179413666160624100439

An Overview on Polylactic Acid, its Cellulosic Composites and Applications

Volume: 14   Issue: 2
Pp: 156-170
Naheed Saba*, Mohammad Jawaid* and Othman Al-Othman
DOI: 10.2174/1570179413666160921115245

Synthesis, Stereochemical Studies and Antimycobacterial Activity of New Acetyl- Hydrazine Pyridazinones

Volume: 14   Issue: 1
Pp: 112-119
Dorina Mantu, Vasilichia Antoci, Alina Nicolescu, Calin Deleanu, Violeta Vasilache and Ionel I. Mangalagiu*
DOI: 10.2174/1570179413999160219164248

Propylene Carbonate in Organic Synthesis: Exploring its Potential as a Green Solvent open access plus

Volume: 13   Issue: 6
Pp: 834-846
Josué S. Bello Forero, July A. Hernández Muñoz, Joel Jones Junior and Flavia M. da Silva
DOI: 10.2174/1570179413999160211094705

Microwave-Assisted Biginelli Reaction: An Old Reaction, a New Perspective open access plus

Volume: 13   Issue: 4
Pp: 569-600
Majid M. Heravi, Mahdieh Ghavidel and Bahareh Heidari
DOI: 10.2174/1570179413666151218202307

The Povarov Reaction as a Versatile Strategy for the Preparation of 1, 2, 3, 4-Tetrahydroquinoline Derivatives: An Overview

Volume: 13   Issue: 2
Pp: 157-175
Josue S. Bello Forero, Joel Jones Junior and Flavia M. da Silva
DOI: 10.2174/1570179412666150706183906

Indoloquinolines: Possible Biogenesis from Common Indole Precursors and their Synthesis using Domino Strategies promotion: free to download

Volume: 13   Issue: 1
Pp: 58-72
Prakash T. Parvatkar and Perunninakulath S. Parameswaran
DOI: 10.2174/1570179412666150511224648

Application of Bio-Based Solvents in Catalysis

Volume: 12   Issue: 6
Pp: 675-695
Arlene G. Corrêa, Márcio W. Paixão and Ricardo S. Schwab
DOI: 10.2174/157017941206150828102108

Recent Advances in Using Niobium Compounds as Catalysts in Organic Chemistry

Volume: 12   Issue: 5
Pp: 570-583
Bruno Henrique Arpini, Aloísio de Andrade Bartolomeu, Carlos Kleber Z. Andrade, Luiz Carlos da Silva-Filho and Valdemar Lacerda
DOI: 10.2174/157017941205150821125817

Superparamagnetic Nanoparticle-Supported Imidazole as an Efficient and Magnetically Recyclable Organocatalyst for Konevenagel Condensation

Volume: 12   Issue: 4
Pp: 466-474
Zhifeng Li, Huanan Hu, Yanxian Jin, Rongrong Li, Anguo Ying and Songlin Xu
DOI: 10.2174/1570179412999150513140221

Preparation of Saccharide Microarrays

Volume: 12   Issue: 2
Pp: 136-139
Gangliang Huang, Qilin Tang, Ping Li, Min Li, Xueqin Zhang, Zhangmei Liu, Deqi Luo and Xinya Mei
DOI: 10.2174/1570179412666141208225037

Two Neglected Multicomponent Reactions: Asinger and Groebke Reaction for Constructing Thiazolines and Imidazolines promotion: free to download

Volume: 12   Issue: 1
Pp: 20-60
Zai-Qun Liu
DOI: 10.2174/1570179411999141112144441

Biomimetic Synthesis of Benzimidazoles, Benzoxazoles, and Benzothiadazole via the Group Transfer of Tetrahydrofolate Models

Volume: 11   Issue: 6
Pp: 911-915
Xueshan Wen, Jianxin Chen, Yanqin Zhao, Xingmao Chang, Jiachun Ma and Wenjun Zheng
DOI: 10.2174/1570179411666140708173654

Synthesis of Glycosylated Natural Products

Volume: 11   Issue: 6
Pp: 874-878
Gangliang Huang, Xueqin Zhang, Min Li, Ping Li, Deqi Luo and Zhangmei Liu
DOI: 10.2174/1570179411666140812233904

Synthesis of Triazole-linked LNA-based Non-ionic Nucleoside Dimers Using Cu(I)- Catalyzed 'Click' Reaction

Volume: 11   Issue: 5
Pp: 757-766
Sunil K. Singh, Vivek K. Sharma, Kapil Bohra, Carl E. Olsen and Ashok K. Prasad
DOI: 10.2174/1570179411666140204155505

Safer, Greener, and More Facile Alternatives for Synthesis with Organic Azides

Volume: 11   Issue: 5
Pp: 732-750
Meaghan M. Sebeika and Graham B. Jones
DOI: 10.2174/1570179411666140328221938

Synthesis of Oxazolo-, Thiazolo-, Pyrazolo-, and Imidazo-Fused Heterocycles by Multi-Component Reactions (Part 2)

Volume: 11   Issue: 4
Pp: 471-525
Mohamed R. Shaaban and Ahmed H.M. Elwahy
DOI: 10.2174/15701794113106660076

Green Chlorination of Organic Compounds Using Trichloroisocyanuric Acid (TCCA)

Volume: 10   Issue: 6
Pp: 820-836
Gabriela F. Mendonca and Marcio C.S. de Mattos
DOI: 10.2174/157017941006140206102255