Combinatorial Chemistry & High Throughput Screening

Accelerated Technologies for Biotechnology, Bioassays, Medicinal Chemistry and Natural Products Research


Gerald H. Lushington
LiS Consulting, Lawrence

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3D QSAR and Docking Study of Gliptin Derivatives as DPP-IV Inhibitors

Volume:16   Issue: 4
Pp: 249-273
Ritesh Agrawal, Pratima Jain, Subodh Narayan Dikshit and Radhe Shyam Bahare
DOI: 10.2174/1386207311316040001
Published on: 24 February, 2013

Probing a Chemical Space for Fragmental Topology-Activity Landscapes (FRAGTAL): Application for Diketo Acid and Catechol HIV Integrase Inhibitor Offspring Fragments

Volume:16   Issue: 4
Pp: 274-287
Andrzej Bak, Tomasz Magdziarz, Agata Kurczyk, Katarzyna Serafin and Jaroslaw Polanski
DOI: 10.2174/1386207311316040002
Published on: 24 February, 2013

The Effect of Leverage and/or Influential on Structure-Activity Relationships

Volume:16   Issue: 4
Pp: 288-297
Sorana D. Bolboaca and Lorentz Jantschi
DOI: 10.2174/1386207311316040003
Published on: 24 February, 2013

Imidazoline-1 Receptor Ligands as Apoptotic Agents: Pharmacophore Modeling and Virtual Docking Study

Volume:16   Issue: 4
Pp: 298-319
Katarina Nikolic, Nevena Veljkovic, Branislava Gemovic, Tatjana Srdic-Rajic and Danica Agbaba
DOI: 10.2174/1386207311316040004
Published on: 24 February, 2013

Ligand-Peroxidase Conjugates for Quantification of Receptor-Mediated Transport into Cells

Volume:16   Issue: 4
Pp: 320-323
Jie Chen and Amandio Vieira
DOI: 10.2174/1386207311316040005
Published on: 24 February, 2013

Rapid Characterization of a Novel Taspine Derivative-HMQ1611 Binding to EGFR by a Cell Membrane Chromatography Method

Volume:16   Issue: 4
Pp: 324-329
Hui Du, Nan Lv, Sicen Wang and Langchong He
DOI: 10.2174/1386207311316040006
Published on: 24 February, 2013