Anti-Cancer Agents in Medicinal Chemistry

(Formerly Current Medicinal Chemistry - Anti-Cancer Agents)

Editor-in-Chief

Simone Carradori
Department of Pharmacy
“G. d’Annunzio” University of Chieti-Pescara
Chieti
(Italy)

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Volume: 17 Issue: 1, January 2016



Meet Our Editorial Board Member free to download

Volume:17   Issue: 1
Pp: 1-1
Luigi Quintieri
DOI: 10.2174/187152061701161207125431
Published on: 07 December, 2016

Overview

Volume:17   Issue: 1
Pp: 2-2
Michelle Prudhomme
DOI: 10.2174/187152061701161207125921
Published on: 07 December, 2016

PREFACE

Volume:17   Issue: 1
Pp: 3-3
Michelle Prudhomme
DOI: 10.2174/187152061701161207130106
Published on: 07 December, 2016



Thiol-Activated Anticancer Agents: The State of the Art

Volume:17   Issue: 1
Pp: 4-20
Daniele Dalzoppo, Veronica Di Paolo, Laura Calderan, Gianfranco Pasut, Antonio Rosato, Anna Maria Caccuri and Luigi Quintieri
DOI: 10.2174/1871520616666160817110310
Published on: 17 August, 2016




Anticancer Drug Combinations, How Far We can Go Through?

Volume:17   Issue: 1
Pp: 21-28
Da-Yong Lu, En-Hong Chen, Hong-Ying Wu, Ting-Ren Lu, Bin Xu and Jian Ding
DOI: 10.2174/1871520616666160404112028
Published on: 04 April, 2016




Ruthenium(II) Complexes as Potential Apoptosis Inducers in Chemotherapy

Volume:17   Issue: 1
Pp: 29-39
Kangdi Zheng, Qiong Wu, Chengxi Wang, Weijun Tan and Wenjie Mei
DOI: 10.2174/1871520616666160622085441
Published on: 21 June, 2016




Killing Glioma ‘Stem-like’ Cells via Drug-Induced Relocation of Endosomal Urokinase Proteins

Volume:17   Issue: 1
Pp: 40-47
Fredric A. Gorin, Nagarekha Pasupuleti, Dinesh Mahajan and Sundeep Dugar
DOI: 10.2174/1871520616666160628122901
Published on: 28 June, 2016




Rapamycin-loaded Immunoliposomes Functionalized with Trastuzumab: A Strategy to Enhance Cytotoxicity to HER2-positive Breast Cancer Cells

Volume:17   Issue: 1
Pp: 48-56
Josimar O. Eloy, Raquel Petrilli, Robert W. Brueggemeier, Juliana Maldonado Marchetti and Robert J. Lee
DOI: 10.2174/1871520616666160526103432
Published on: 25 May, 2016




Novel 2-Thienyl- and 2-Benzothienyl-Substituted 6-(2-Imidazolinyl)Benzothiazoles: Synthesis; in vitro Evaluation of Antitumor Effects and Assessment of Mitochondrial Toxicity

Volume:17   Issue: 1
Pp: 57-66
Livio Racané, Mirela Sedić, Nataša Ilić, Maja Aleksić, Sandra Kraljević Pavelić and Grace Karminski-Zamola
DOI: 10.2174/1871520615666160504094753
Published on: 03 May, 2016




Design, Synthesis and Evaluation of 5-pyridin-4-yl-2-thioxo-[1,3,4]oxadiazol-3-yl Derivatives as Anti-angiogenic Agents Targeting VEGFR-2

Volume:17   Issue: 1
Pp: 67-74
Umesh Bhanushali, Samidha Kalekar-Joshi, Renuka Kulkarni-Munshi, Swapna Yellanki, Raghavender Medishetty, Pushkar Kulkarni and Ramaa Subramanian Chelakara
DOI: 10.2174/1871520615666160504094222
Published on: 03 May, 2016




Synthesis, in vitro Antiproliferative and Antiinflammatory Activities, and Kinase Inhibitory effects of New 1,3,4-triarylpyrazole Derivatives

Volume:17   Issue: 1
Pp: 75-84
Mohammed I. El-Gamal, Mohammed S. Abdel-Maksoud, Mahmoud M. Gamal El-Din, Ji-Sun Shin, Kyung-Tae Lee, Kyung Ho Yoo and Chang-Hyun Oh
DOI: 10.2174/1871520616666160620074534
Published on: 19 June, 2016




New 2-Imino-2H-Chromene-3(N-aryl)carboxamides as Potential Cytotoxic Agents

Volume:17   Issue: 1
Pp: 85-92
Rupinder Kaur Gill, Jyoti Kumari and Jitender Bariwal
DOI: 10.2174/1871520616666160310142949
Published on: 10 March, 2016




Effect of PUFAs Oral Administration on the Amount of Apoptotic Caspases Enzymes in Gastric Cancer Patients Undergoing Chemotherapy

Volume:17   Issue: 1
Pp: 93-101
Homayun Dolatkhah, Ahmad Movahedian, Mohammad-Hossein Somi, Mahmud Aghaei, Naser Samadi, Ahmad Mirza-Aghazade and Ali Esfahani
DOI: 10.2174/1871520616666160520113503
Published on: 20 May, 2016




Glycodendrimer PPI as a Potential Drug in Chronic Lymphocytic Leukaemia. The Influence of Glycodendrimer on Apoptosis in In Vitro B-CLL Cells Defined by Microarrays

Volume:17   Issue: 1
Pp: 102-114
Ida Franiak-Pietryga, Ewelina Ziółkowska, Barbara Ziemba, Dietmar Appelhans, Henryk Maciejewski, Brigitte Voit, Aleksandra Kaczmarek, Tadeusz Robak, Barbara Klajnert-Maculewicz, Barbara Cebula-Obrzut, Piotr Smolewski, Maciej Borowiec and Maria Bryszewska
DOI: 10.2174/1871520616666160622092947
Published on: 21 June, 2016




Induction of Autophagic Cell Death in Apoptosis-resistant Pancreatic Cancer Cells using Benzo[α]phenoxazines Derivatives, 10-methyl-benzo[α]phenoxazine-5-one and benzo[α]phenoxazine-5-one

Volume:17   Issue: 1
Pp: 115-125
Sanjima Pal, Sunita Salunke-Gawalib and V. Badireenath Konkimallaa
DOI: 10.2174/1871520616666160624091519
Published on: 23 June, 2016




In Vivo Performance of a Ruthenium-cyclopentadienyl Compound in an Orthotopic Triple Negative Breast Cancer Model

Volume:17   Issue: 1
Pp: 126-136
Nuno Mendes, Francisco Tortosa, Andreia Valente, Fernanda Marques, António Matos, Tânia S. Morais, Ana Isabel Tomaz, Fátima Gärtner and M. Helena Garcia
DOI: 10.2174/1871520616666160922165133
Published on: 22 September, 2016




Synthesis of Icaritin and β-anhydroicaritin Mannich Base Derivatives and Their Cytotoxic Activities on Three Human Cancer Cell Lines

Volume:17   Issue: 1
Pp: 137-142
Van-Son Nguyen, Ling Shi, Sheng-Chun Wang and Qiu-An Wang
DOI: 10.2174/1871520616666160404111210
Published on: 04 April, 2016




Cordycepin Affects Multiple Apoptotic Pathways to Mediate Hepatocellular Carcinoma Cell Death

Volume:17   Issue: 1
Pp: 143-149
Yulin Zhou, Zhihua Guo, Qingfan Meng, Jiahui Lu, Ning Wang, Hui Liu, Qiming Liang, Yutong Quan, Di Wang and Jing Xie
DOI: 10.2174/1871520616666160526114555
Published on: 26 May, 2016