Volume 25, Issue 6
Capivasertib: First Approved AKT inhibitor for the Treatment of Patients with Breast Cancer
Pp: 371-377
Author(s): Surya K. De*
DOI: 10.2174/0118715206360571241126080725
A Review of Anticancer Potential of Conferone, Diversin and Ferutinin; Which One is Stronger for Cancer Therapy?
Pp: 378-387
Author(s): Fariborz Keshmirshekan, Seyed-Mahdi Mohamadi-Zarch and Seyyed Majid Bagheri*
DOI: 10.2174/0118715206328175241022081832
Composition and Biological Activity of Flavonoid-containing Fractions of an Extract from Gratiola officinalis L.
Pp: 388-398
Author(s): Alexander Shirokov*, Vyacheslav Grinev, Matvey Kanevskiy, Yulia Fedonenko, Larisa Matora, Natalya Polukonova, Dmitry Mudrak, Artyom Mylnikov, Anna Polukonova, Alla Bucharskaya, Nikita Navolokin and Galina Maslyakova
DOI: 10.2174/0118715206323280241029215900
Synthesis of Chromene-linked Bis-indole Derivatives as Selective Tumor-associated Carbonic Anhydrase IX Inhibitors
Pp: 399-410
Author(s): Priti Singh*, Sridhar Goud Nerella, Baijayantimala Swain, Andrea Angeli, Samreen Kausar, Qasim Ullah, Claudiu T. Supuran* and Mohammed Arifuddin
DOI: 10.2174/0118715206341087241029064945
The Mesoionic 1,3,4-thiadiazolium Derivative, MI-D, is a Potential Drug for Treating Glioblastoma by Impairing Mitochondrial Functions Linked to Energy Provision in Glioma Cells
Pp: 411-419
Author(s): Marília Locatelli Corrêa-Ferreira, Amanda do Rocio Andrade Pires, Juan Vitor Miranda, Eduardo de Freitas Montin, Igor Resendes Barbosa, Aurea Echevarria Aznar Neves Lima, Maria Eliane Merlin Rocha, Glaucia Regina Martinez and Sílvia Maria Suter Correia Cadena*
DOI: 10.2174/0118715206329159241010052746
Amide Functionalized Novel Pyrrolo-pyrimidine Derivative as Anticancer Agents: Synthesis, Characterization and Molecular Docking Studies
Pp: 420-432
Author(s): Praveen Kumar Bandaru*, Satya Kameswara Rao Nidasanametla and Pulipaka Shyamala
DOI: 10.2174/0118715206333935241004070350
Investigation of Apoptotic and Anticancer Effects of 2-substituted Benzothiazoles in Breast Cancer Cell Lines: EGFR Modulation and Mechanistic Insights
Pp: 433-445
Author(s): Muhammed Mehdi Üremiş*, Mustafa Ceylan and Yusuf Türköz
DOI: 10.2174/0118715206335840241018053929