Abstract
In this work we aimed at finding a concise method for the design of the new pharmacologically active compound 6, which is a precursor to obtaining non-protein amino acid 7 considered as GABA analogue, furthermore it can be used to construct enantiopure, conformationally restricted peptides. For this purpose the Schmidt reaction was applied.
Keywords: Amino acids, schmidt reaction, natural products, terpenoids
Letters in Organic Chemistry
Title: Concise Synthesis of Non-Protein Amino Acid from Natural Product via Schmidt Reaction
Volume: 6 Issue: 3
Author(s): Kamila Gajcy, Tadeusz Librowski and Stanislaw Lochynski
Affiliation:
Keywords: Amino acids, schmidt reaction, natural products, terpenoids
Abstract: In this work we aimed at finding a concise method for the design of the new pharmacologically active compound 6, which is a precursor to obtaining non-protein amino acid 7 considered as GABA analogue, furthermore it can be used to construct enantiopure, conformationally restricted peptides. For this purpose the Schmidt reaction was applied.
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Cite this article as:
Gajcy Kamila, Librowski Tadeusz and Lochynski Stanislaw, Concise Synthesis of Non-Protein Amino Acid from Natural Product via Schmidt Reaction, Letters in Organic Chemistry 2009; 6 (3) . https://dx.doi.org/10.2174/157017809787893037
DOI https://dx.doi.org/10.2174/157017809787893037 |
Print ISSN 1570-1786 |
Publisher Name Bentham Science Publisher |
Online ISSN 1875-6255 |
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