Suzuki-Miyaura Cross-Coupling Reaction in the Functionalization of the C Ring of Morphinans

Author(s): Attila Sipos, Sandor Berenyi

Journal Name: Letters in Organic Chemistry

Volume 4 , Issue 2 , 2007

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Abstract:

New methods have been developed for the functionalization of the non-aromatic C ring of morphinans with Suzuki-Miyaura cross-coupling of sulfonates and bromides.

Keywords: Suzuki-Miyaura cross-coupling of tosylates and mesylates, spatially hindered position, 14-arylmorphinan, opioid receptor binding affinity, microwave activation

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Article Details

VOLUME: 4
ISSUE: 2
Year: 2007
Page: [146 - 150]
Pages: 5
DOI: 10.2174/157017807780414145
Price: $65

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