Abstract
A simple and practical method to prepare ‘libraries’ of substituted 1-phenylpiperazine building blocks in parallel format has been developed.
Keywords: Bis-alkylation, N-arylpiperazines, nitrogen mustard, parallel synthesis, solvent-free synthesis, SAR-informative, 1-phenylpiperazines, morpholine, iminodiethanol, ethanamine
Letters in Organic Chemistry
Title: Practical Method for Parallel Synthesis of Diversely Substituted 1- henylpiperazines
Volume: 8 Issue: 9
Author(s): Igor Konstantinov, Konstantin Bukhryakov, Yuri Gezentsvey and Mikhail Krasavin
Affiliation:
Keywords: Bis-alkylation, N-arylpiperazines, nitrogen mustard, parallel synthesis, solvent-free synthesis, SAR-informative, 1-phenylpiperazines, morpholine, iminodiethanol, ethanamine
Abstract: A simple and practical method to prepare ‘libraries’ of substituted 1-phenylpiperazine building blocks in parallel format has been developed.
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Konstantinov Igor, Bukhryakov Konstantin, Gezentsvey Yuri and Krasavin Mikhail, Practical Method for Parallel Synthesis of Diversely Substituted 1- henylpiperazines, Letters in Organic Chemistry 2011; 8 (9) . https://dx.doi.org/10.2174/157017811799304386
DOI https://dx.doi.org/10.2174/157017811799304386 |
Print ISSN 1570-1786 |
Publisher Name Bentham Science Publisher |
Online ISSN 1875-6255 |
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