Abstract
Boron-based mixed anhydrides are rapidly reactive, easy to prepare, cheap, efficient, and general acylating reagents capable of selectivity when chelation is possible. High yields of various esters, amides and thioesters are quickly obtainable and the products are easy to isolate in high purity. The method is readily used under multiple parallel synthesis conditions and is readily scaleable.
Keywords: Tetraacyldiborates, Acylation Reagents, Boron-based, anhydrides, chelation
Combinatorial Chemistry & High Throughput Screening
Title: Tetraacyldiborates: Selective and Efficient Acylation Reagents Suitable for Multiple Parallel Synthetic Applications
Volume: 6 Issue: 2
Author(s): Elmer J. Gentry, Hanumaiah Telikepalli, Pusuluri Srinivas and Lester A. Mitscher
Affiliation:
Keywords: Tetraacyldiborates, Acylation Reagents, Boron-based, anhydrides, chelation
Abstract: Boron-based mixed anhydrides are rapidly reactive, easy to prepare, cheap, efficient, and general acylating reagents capable of selectivity when chelation is possible. High yields of various esters, amides and thioesters are quickly obtainable and the products are easy to isolate in high purity. The method is readily used under multiple parallel synthesis conditions and is readily scaleable.
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Cite this article as:
Gentry J. Elmer, Telikepalli Hanumaiah, Srinivas Pusuluri and Mitscher A. Lester, Tetraacyldiborates: Selective and Efficient Acylation Reagents Suitable for Multiple Parallel Synthetic Applications, Combinatorial Chemistry & High Throughput Screening 2003; 6 (2) . https://dx.doi.org/10.2174/1386207033329797
DOI https://dx.doi.org/10.2174/1386207033329797 |
Print ISSN 1386-2073 |
Publisher Name Bentham Science Publisher |
Online ISSN 1875-5402 |
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