Search Result "triazoles"


Research Article

Synthesis and Biological Evaluation of Triazole-Vanillin Molecular Hybrids as Anti-Cancer Agents

Journal: Current Bioactive Compounds
Volume: 13 Issue: 3 Year: 2017 Page: 223-235
Author(s): Gangavaram V. M. Sharma,Kandikonda S. Kumar,Sheri V. Reddy,Arumugam Nagalingam,Kathleen M. Cunningham,Ramesh Ummanni,Helmut Hugel,Dipali Sharma,Sanjay V. Malhotra

Research Article

In vitro α-Glucosidase Inhibition by Non-sugar based Triazoles of Dibenzoazepine, their Structure-Activity Relationship, and Molecular Docking

Journal: Medicinal Chemistry
Volume: 13 Issue: 7 Year: 2017 Page: 698-704
Author(s): Maria A. Khan,Kulsoom Javaid,Abdul Wadood,Alam Jamal,Farhana Batool,Saba Fazal-ur-Rehman,Fatima Z. Basha,Muhammad I. Choudhary

Research Article

1,2,3-Triazole-Isoxazole Based Acetylcholinesterase Inhibitors: Synthesis, Biological Evaluation and Docking Study

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 58-65
Author(s): Zahra Najafi,Mohammad Mahdavi,Mina Saeedi,Reyhaneh Sabourian,Mahnaz Khanavi,Maliheh Safavi,Maliheh Barazandeh Tehrani,Abbas Shafiee,Alireza Foroumadi,Tahmineh Akbarzadeh

Research Article

Synthesis of Novel 1,4-Substituted 1,2,3-Triazoles by Water-Soluble (Salicyladimine) 2Cu Complex Catalyzed Azide-Alkyne Cycloaddition in Water

Journal: Letters in Organic Chemistry
Volume: 14 Issue: 8 Year: 2017 Page: 557-565
Author(s): Yang Liu,Ping Liu,Yan Liu,Yu Wei

Research Article

Synthesis of 1,4-disubstituted 1,2,3-triazole Derivatives Using Click Chemistry and their Src Kinase Activities

Journal: Medicinal Chemistry
Volume: 13 Issue: 1 Year: 2017 Page: 40-48
Author(s):

Research Article

Synthesis, Antibacterial, Antifungal, Antimycobacterial Activity Evaluation of Novel 1,2,4-triazole Derivatives Bearing 4-Aminophenyl Moiety

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 8 Year: 2017 Page: 938-948
Author(s): Betul Kaya Cavusoglu,Leyla Yurttas,Meral Y. Cankilic,Zafer A. Kaplancikli

Research Article

Possible Binding Mode Analysis of Pyrazolo-triazole Hybrids as Potential Anticancer Agents through Validated Molecular Docking and 3D-QSAR Modeling Approaches

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 5 Year: 2017 Page: 515-527
Author(s): Siekh Abdul Amin,Nilanjan Adhikari,Ram K. Agrawal,Tarun Jha,Shovanlal Gayen

Research Article

Quantitative Structure-Activity Relationship and Docking Studies on a Series of Oxadiazole and Triazole Substituted Naphthyridines as HIV-1 Integrase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 10-27
Author(s): Basheerulla Shaik,Vijay Agrawal,Satya P. Gupta,Urvana Menon

Research Article

The Oxime Derivatives of 1-R-1H-Naphtho[2,3-d][1,2,3]triazole-4,9-dione 2-oxides: Synthesis and Properties

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2017 Page: 1814-1823
Author(s): Leonid M. Gornostaev,Vladimir B. Tsvetkov,Alina A. Markova,Tatyana I. Lavrikova,Yulia G. Khalyavina,Anastasia S. Kuznetsova,Dmitry N. Kaluzhny,Alexei V. Shunayev,Maria V. Tsvetkova,Valeria A. Glazunova,Vladimir V. Chernyshev,Alexander A. Shtil

Research Article

Synthesis and Antioxidant Evaluation of Some Novel Benzimidazole Derivatives Containing a Triazole Nucleus

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 2 Year: 2017 Page: 201-208
Author(s): Fatih Y?lmaz, Emre Mente?e, Nimet Balta?

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