Search Result "quinazolines"


Review Article

Bestowal of Quinazoline Scaffold in Anticancer Drug Discovery

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 21 Issue: 1 Year: 2021 Page: 1350-1368
Author(s): Rina Das,Dinesh K. Mehta,Meenakshi Dhanawat

Review Article

Advances on Quinazoline Based Congeners for Anticancer Potential

Journal: Current Organic Chemistry
Volume: 25 Issue: 6 Year: 2021 Page: 695-723
Author(s): Parul Grover,Monika Bhardwaj,Garima Kapoor,Lovekesh Mehta,Roma Ghai,K. Nagarajan

Mini-Review Article

2-Substituted-mercapto-quinazolin-4(3H)-ones as DHFR Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 21 Issue: 1 Year: 2021 Page: 2249-2260
Author(s): Hussein I. El-Subbagh,Mohamed A. Sabry

Review Article

Recent Advances in C–H Activation and Functionalization of Quinazolinones/ Quinazolines

Journal: Current Organic Chemistry
Volume: 25 Issue: 5 Year: 2021 Page: 601-634
Author(s): N. Umadevi,G. Kumar,N.C. Gangi Reddy,B.V. Subba Reddy

Review Article

The Quinazoline-Chalcone and Quinazolinone-Chalcone Hybrids: A Promising Combination for Biological Activity

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 21 Issue: 2 Year: 2021 Page: 186-203
Author(s): Eduardo Bustos Mass,Gilmar Vieira Duarte,Dennis Russowsky

Research Article

Synthesis and Enzymological Characterization of Some 2-(Substitutedphenylamino) quinazolin-4(3H)-one Derivatives as Potent α-Glucosidase Inhibitors In Vitro

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 7 Year: 2021 Page: 723-732
Author(s): Emre Kadir Ayan,Zeynep Soyer,Şirin Uysal

Research Article

Synthesis and Antimicrobial Evaluation of Quinazoline-4[3H]-one Derivatives

Journal: Letters in Organic Chemistry
Volume: 18 Issue: 7 Year: 2021 Page: 547-554
Author(s): Cheenu Chaudhary,Sushil Kumar,Surendra Kumar,S. Riaz Hashim

Research Article

Substituted 3-R-2,8-Dioxo-7,8-dihydro-2H-pyrrolo[1,2-a][1,2,4] triazino[2,3-c]quinazoline-5a(6H)carboxylic Acids and their Salts – a Promising Class of Anti-inflammatory Agents

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2021 Page: 75-88
Author(s): Viktor Stavytskyi,Oleksii Antypenko,Inna Nosulenko,Galyna Berest,Oleksii Voskoboinik,Sergiy Kovalenko

Research Article

Design, Synthesis, Pharmacological evaluation, in silico modeling, prediction of toxicity and metabolism studies of novel 1-(substituted)-2-methyl-3-(4-oxo-2-phenyl quinazolin-3(4H)-yl)isothioureas

Journal: Medicinal Chemistry
Volume: 17 Issue: 4 Year: 2021 Page: 352-368
Author(s): M.T. Sulthana,V. Alagarsamy,K. Chitra

Research Article

Synthesis and Anti-Proliferative Evaluations of New Heterocyclic Derivatives Using 5,6,8,9-tetrahydropyrazolo[5,1-b]quinazolin-7(3H)-one Derivatives Derived from Cyclohexa-1,4-dione

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 21 Issue: 4 Year: 2021 Page: 408-426
Author(s): Mahmoud A.A. Mahmoud,Meshari A. Alsharif,Rafat M. Mohareb

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