Search Result "quinazolines"


Research Article

Resolving the Mystery of Ring Opening in the Synthesis of Benzo[d][1, 3]oxazin-4-one and Quinazolin-4(3H)-one

Journal: Letters in Organic Chemistry
Volume: 16 Issue: 1 Year: 2019 Page: 898-905
Author(s): Harun Patel,Rahul Pawara,Sanjay Surana

Research Article

New Quinazoline-Sulfonylurea Conjugates: Design, Synthesis and Hypoglycemic Activity

Journal: Medicinal Chemistry
Volume: 15 Issue: 6 Year: 2019 Page: 632-645
Author(s): Sahar M. Abou-Seri,AlShaimaa M. Taha,Mona A. Mohamed,Nour M. Abdelkader

Research Article

2,4-Disubstituted Quinazoline Derivatives Act as Inducers of Tubulin Polymerization: Synthesis and Cytotoxicity

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 19 Issue: 8 Year: 2019 Page: 1048-1057
Author(s): Ebrahim S. Moghadam,Maryam H. Tehrani,René Csuk,Lucie Fischer,Mohammad Ali Faramarzi,Arezoo Rashidi,Iraj Javadi,Mohsen Amini

Research Article

Lemon Juice Mediated Synthesis of 3-Substituted Quinazolin-4(3H)-Ones and their Pharmacological Evaluation

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 19 Issue: 1 Year: 2019 Page: 2001-2009
Author(s): Malavattu G. Prasad,C. Vijaya Lakshmi,Naresh K. Katari,Rajshekhar Karpoormath,Manojit Pal

Research Article

Synthesis, 2D-QSAR Studies and Biological Evaluation of Quinazoline Derivatives as Potent Anti-Trypanosoma cruzi Agents

Journal: Medicinal Chemistry
Volume: 15 Issue: 3 Year: 2019 Page: 265-276
Author(s): Mariela Bollini,Ana María Bruno,María Eugenia Niño,Juan José Casal,Leandro Daniel Sasiambarrena,Damián Ariel González Valdez,Leandro Battini,Vanesa Rocío Puente,María Elisa Lombardo

Research Article

Design, Synthesis and Biological Evaluation of Spiro Cyclohexane-1,2- Quinazoline Derivatives as Potent Dipeptidyl Peptidase IV Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 19 Issue: 3 Year: 2019 Page: 250-269
Author(s): Yasmin M Syam,Somaia S. Abd El-Karim,Tamer Nasr,Samia A. Elseginy,Manal M. Anwar,Mohsen M Kamel,Hanan F. Ali

General Research Article

Design, Synthesis and Antitumor Activity of Quinazoline Derivatives Bearing 2,3-Dihydro-indole or 1,2,3,4-Tetrahydroquinoline

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 5 Year: 2019 Page: 533-546
Author(s): Yiqiang OuYang,Bingbing Zhao,Xiuying Chen,Caolin Wang,Hong Zhang,Shuang Jia,Wufu Zhu,Pengwu Zheng

Research Article

Synthesis, Plasmodium falciparum Inhibitory Activity, Cytotoxicity and Solubility of N2,N4-Disubstituted Quinazoline-2,4-diamines

Journal: Medicinal Chemistry
Volume: 15 Issue: 6 Year: 2019 Page: 691-702
Author(s): Nattakarn Pobsuk,Praphasri Suphakun,Supa Hannongbua,Chanin Nantasenamat,Kiattawee Choowongkomon,M. Paul Gleeson

Research Article open access plus

Synthesis and Biological Evaluation of Some Novel Thiophene-bearing Quinazoline Derivatives as EGFR Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 2 Year: 2019 Page: 102-110
Author(s): Min Zou,Bo Jin,Yanrong Liu,Huiping Chen,Zhuangli Zhang,Changzheng Zhang,Zhihong Zhao,Liyun Zheng

Research Article

Green Chemistry Preparation of thiochromeno[4,3-b]pyran and benzo[h]thiazolo[2,3-b]quinazoline Derivatives using HSBM Technique over ZnAl2O4 Nano-Powders

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 22 Issue: 6 Year: 2019 Page: 421-427
Author(s): Seyyed Jalal Roudbaraki,Sadaf Janghorban,Majid Ghashang

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