Search Result "prodrug"


Review Article

Insight into Prodrugs of Quinolones and Fluoroquinolones

Journal: Infectious Disorders - Drug Targets
Volume: 16 Issue: 3 Year: 2016 Page: 140-161
Author(s): Prabodh Chander Sharma, Mona Piplani, Monika Mittal, Rakesh Pahwa

Review Article

Design of Lipophilic Prodrugs to Improve Drug Delivery and Efficacy

Journal: Current Drug Targets
Volume: 17 Issue: 1 Year: 2016 Page: 1773-1798
Author(s): Abhirup Mandal, Mitesh Patel, Ye Sheng, Ashim K. Mitra

Designing Prodrugs Based on Special Residues of Human Serum Albumin

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 9 Year: 2016 Page: 996-1008
Author(s): Yi Gou,Feng Yang,Hong Liang

Intramolecular Processes and Their Applications in Prodrugs Approaches- Experimental and Computational Studies

Journal: Current Organic Chemistry
Volume: 20 Issue: 3 Year: 2016 Page: 289-315
Author(s): Rafik Karaman,Salma Jumaa,Heba Awwadallah,Samya Salah,Yahya Khawaja,Donia Karaman

Novel Thioester Prodrug of N-acetylcysteine for Odor Masking and Bioavailability Enhancement

Journal: Current Drug Delivery
Volume: 13 Issue: 4 Year: 2016 Page: 611-620
Author(s): Neha V. Bhilare,Suneela S. Dhaneshwar,Akanksha J. Sinha,Amit D. Kandhare,Subhash L. Bodhankar

Synthesis, Biological Evaluation and Pharmacokinetic Studies of Mefenamic Acid - N-Hydroxymethylsuccinimide Ester Prodrug as Safer NSAID

Journal: Medicinal Chemistry
Volume: 12 Issue: 6 Year: 2016 Page: 585-591
Author(s): Asif Husain, Priyanka Ahuja, Aftab Ahmad, Shah A. Khan

Ester Prodrugs of Ketoprofen: Synthesis, In Vitro Stability, In Vivo Biological Evaluation and In Silico Comparative Docking Studies Against COX-1 and COX-2

Journal: Current Drug Discovery Technologies
Volume: 13 Issue: 1 Year: 2016 Page: 41-57
Author(s): Musa Ahmed,Faizul Azam,Abdul Gbaj,Abdulmottaleb E. Zetrini,Amna S. Abodlal,Abir Rghigh,Eman Elmahdi,Amel Hamza,Mabruk Salama,Salah M. Bensaber

Research Article

Bispecific Antibodies for Targeted Delivery of Dendritic Polyglycerol (dPG) Prodrug Conjugates

Journal: Current Cancer Drug Targets
Volume: 16 Issue: 7 Year: 2016 Page: 639-649
Author(s):

Phospholipid-Based Prodrugs for Drug Targeting in Inflammatory Bowel Disease: Computational Optimization and In-Vitro Correlation

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 23 Year: 2016 Page: 2543-2548
Author(s): Arik Dahan,Shimon Ben-Shabat,Noa Cohen,Shahar Keinan,Igor Kurnikov,Aaron Aponick,Ellen M. Zimmermann

Letter Article

Synthesis and Evaluation of A Water-Soluble Epothilone B Prodrug with Remarkably Decreased Toxicity

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 9 Year: 2016 Page: 619-624
Author(s): Hai-Bo Wang,Hongfu Kuang,Wei Zhang,Xiaomeng Zhou,Tianming Zhu

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