Search Result "major metabolites"


Inhibition of Leukotriene Biosynthesis by Secondary Plant Metabolites

Journal: Current Organic Chemistry
Volume: 12 Issue: 8 Year: 2008 Page: 602-618
Author(s): Michael Adams, Rudolf Bauer

Marine Metabolites Overcoming or Circumventing Multidrug Resistance Mediated by ATP-Dependent Transporters: A New Hope for Patient with Tumors Resistant to Conventional Chemotherapy

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 8 Issue: 8 Year: 2008 Page: 886-903
Author(s): Chantal Barthomeuf, Marie-Lise Bourguet-Kondracki, Jean-Michel Kornprobst

In Vitro Screening Techniques for Reactive Metabolites for Minimizing Bioactivation Potential in Drug Discovery

Journal: Current Drug Metabolism
Volume: 9 Issue: 9 Year: 2008 Page: 952-964
Author(s): Chandra Prakash, Raman Sharma, Michelle Gleave, Angus Nedderman

Oxidative Bioactivation and Toxicity of Leflunomide in Immortalized Human Hepatocytes and Kinetics of the Non-Enzymatic to Its Major etabolitie, A77 1726

Journal: Drug Metabolism Letters
Volume: 2 Issue: 3 Year: 2008 Page: 153-157
Author(s): Quee Ming Seah, Lee-Sun New, Eric C.Y. Chan, Urs A. Boeslsterli

Strategies to In Vitro Assessment of Major Human CYP Enzyme Activities by Using Liquid Chromatography Tandem Mass Spectrometry

Journal: Current Drug Metabolism
Volume: 9 Issue: 1 Year: 2008 Page: 12-19
Author(s): A. Lahoz, M. T. Donato, J. V Castell, M. J. Gomez-Lechon

Mentha L. Species (Lamiaceae) as Promising Sources of Bioactive Secondary Metabolites

Journal: Current Pharmaceutical Design
Volume: 14 Issue: 2 Year: 2008 Page: 3141-3150
Author(s): N. Mimica-Dukic, B. Bozin

Troglitazone Thiol Adduct Formation in Human Liver Microsomes: Enzyme Knietics and Reaction Phenotyping

Journal: Drug Metabolism Letters
Volume: 2 Issue: 3 Year: 2008 Page: 184-189
Author(s): Jinping Gan, Qinling Qu, Bing He, Wen C. Shyu, A. David Rodrigues, Kan He

Rapid and Sensitive Characterization of the Metabolite Formation Enzyme Kinetics of Radiolabeled Drugs Using Stop-Flow Liquid Radiochromatography

Journal: Drug Metabolism Letters
Volume: 2 Issue: 1 Year: 2008 Page: 41-46
Author(s): Lifei Wang, Weiping Zhao, Donglu Zhang, Mingshe Zhu

Major Digestive Carbohydrase During Larval Development of Meal Moth, Plodia interpunctella (Lepidoptera: Pyralidae)

Journal: Protein & Peptide Letters
Volume: 15 Issue: 9 Year: 2008 Page: 1022-1026
Author(s): M. P. de Sales, Alonso Alcazar, L. M. Lima, Ticiana M.L. Amorim, J. C.M. Pitanga, R. A. Pereira, L. L.P. Macedo, F. P. Macedo, A. S. Oliveira, Adriana F. Uchoa

Identification of Four Urea Adducts of Andrographolide in Humans

Journal: Drug Metabolism Letters
Volume: 2 Issue: 4 Year: 2008 Page: 261-268
Author(s): Liang Cui, Wan Chan, Feng Qiu, Zongwei Cai, Xinsheng Yao

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