Search Result "integrase"


Research Article

Novel Benzoxazin-3-one Derivatives: Design, Synthesis, Molecular Modeling, anti-HIV-1 and Integrase Inhibitory Assay

Journal: Medicinal Chemistry
Volume: 16 Issue: 7 Year: 2020 Page: 938-946
Author(s): Mahdieh Safakish,Zahra Hajimahdi,Rouhollah Vahabpour,Rezvan Zabihollahi,Afshin Zarghi

Research Article

Design, Synthesis and In Vitro Evaluation of 2-Oxo-N-Substituted Phenyl- 2h-Chromene-3-Carboxamide Derivatives as Hiv Integrase Strand Transfer Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 4 Year: 2020 Page: 416-425
Author(s): Pankaj Wadhwa,Priti Jain,Hemant R Jadhav

Research Article

Co-medications and Drug-Drug Interactions in People Living with HIV in Turkey in the Era of Integrase Inhibitors

Journal: Current HIV Research
Volume: 18 Issue: 6 Year: 2020 Page: 415-425
Author(s): Zuhal Yeşilbağ,Emine İlay Şengül,Sevtap Şenoğlu,Özlem Altuntaş Aydın,Hayat Kumbasar Karaosmanoğlu

Research Article

Quantitative Structure-Activity Relationship Study for HIV-1 LEDGF/p75 Inhibitors

Journal: Current Computer-Aided Drug Design
Volume: 16 Issue: 5 Year: 2020 Page: 654-666
Author(s): Yang Li,Yujia Tian,Yao Xi,Zijian Qin,Aixia Yan

Research Article

Design, Synthesis, Molecular Modeling and Anti-HIV Assay of Novel Quinazolinone Incorporated Coumarin Derivatives

Journal: Current HIV Research
Volume: 18 Issue: 1 Year: 2020 Page: 41-51
Author(s): Mahdieh Safakish,Zahra Hajimahdi,Mohammad R. Aghasadeghi,Rouhollah Vahabpour,Afshin Zarghi

Review Article

Styrylquinoline – A Versatile Scaffold in Medicinal Chemistry

Journal: Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2020 Page: 141-154
Author(s): Robert Musiol

General Research Article

Binding Insight of Anti-HIV Phytocompounds with Prime Targets of HIV: A Molecular Dynamics Simulation Analysis

Journal: Current HIV Research
Volume: 18 Issue: 2 Year: 2020 Page: 132-141
Author(s): Jaykant Vora,Mohd Athar,Sonam Sinha,Prakash C. Jha,Neeta Shrivastava

Research Article

In vitro Anti-HIV and Antimicrobial Activities of a Halogenated Monoterpene from a Namibian Plocamium Species of Marine Algae

Journal: Current Bioactive Compounds
Volume: 16 Issue: 3 Year: 2020 Page: 363-367
Author(s): Aina N. Shiyanga,Michael Knott,Petrina Kapewangolo

Review Article

An Overview of Antiretroviral Agents for Treating HIV Infection in Paediatric Population

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 5 Year: 2020 Page: 760-794
Author(s): Rita Melo,Agostinho Lemos,António J. Preto,Beatriz Bueschbell,Pedro Matos-Filipe,Carlos Barreto,José G. Almeida,Rúben D.M. Silva,João D.G. Correia,Irina S. Moreira

Letter Article

Insights into Biophysical Methods to Study Interactions Between HIV-1 Reverse Transcriptase and Non-Nucleoside Reverse Transcriptase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 6 Year: 2020 Page: 745-752
Author(s): Julien Dumond,Jean-Marcel J. Tronchet,Serge Kirkiacharian,Michel Seman,Michèle Reboud-Ravaux

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