Search Result "glucuronidation"


Research Article

New Perspectives on Acyl Glucuronide Risk Assessment in Drug Discovery: Investigation of In vitro Stability, In situ Reactivity, and Bioactivation

Journal: Drug Metabolism Letters
Volume: 12 Issue: 2 Year: 2018 Page: 84-92
Author(s): Mithat Gunduz,Upendra A. Argikar,Amanda L. Cirello,Jennifer L. Dumouchel

Case Studies

Ethyl Glucuronide in Hair (hEtG) after Exposure to Alcohol-based Perfumes

Journal: Current Pharmaceutical Biotechnology
Volume: 19 Issue: 2 Year: 2018 Page: 175-179
Author(s): Cristina Sempio,Luca Morini,Matteo Moretti

Review Article

Saccharolactone: The History, the Myth, and the Practice

Journal: Current Drug Metabolism
Volume: 19 Issue: 4 Year: 2018 Page: 304-309
Author(s): Upendra A. Argikar

Research Article

Quantitative Estimation of Alcohol Marker Ethyl Glucuronide (EtG) in Human Hair by LC-MS/MS: An Application Towards Doping Control & Forensic Science

Journal: Current Chromatography
Volume: 5 Issue: 2 Year: 2018 Page: 112-116
Author(s): Sahu Kapendra,Ahi Shobha,Nasare Mahesh,Singh Satyendra,Beotra Alka,Jain Shila

Research Article

2-Oxo-1,2,3,4-tetrahydropyrimidines Ethyl Esters as Potent β- Glucuronidase Inhibitors: One-pot Synthesis, In vitro and In silico Studies

Journal: Medicinal Chemistry
Volume: 14 Issue: 8 Year: 2018 Page: 818-830
Author(s): Sarosh Iqbal,Nimra N. Shaikh,Khalid M. Khan,Sehrish Naz,Zaheer Ul-Haq,Shahnaz Perveen,Muhammad I. Choudhary

Research Article

In vitro Drug Metabolism Investigation of 7-Ethoxycoumarin in Human, Monkey, Dog and Rat Hepatocytes by High Resolution LC-MS/MS

Journal: Drug Metabolism Letters
Volume: 12 Issue: 1 Year: 2018 Page: 33-53
Author(s): Wan-Yong Feng,Jenny Wen,Kathe Stauber

Research Article

UPLC-MS for Identification of Quercetin Derivatives in Cuphea glutinosa Cham. & Schltdl (Lythraceae) and Evaluation of Antifungal Potential

Journal: Current Pharmaceutical Analysis
Volume: 14 Issue: 6 Year: 2018 Page: 586-594
Author(s): Marí C. Santos,Lidiane S. Farias,Liara Merlugo,Thayse V. de Oliveira,Fábio S. Barbosa,Alexandre M. Fuentefria,Amelia T. Henriques,Cássia V. Garcia,Andreas S. L. Mendez

Research Article

Tissue Distribution of Active Principles from Alpiniae Oxyphyllae Fructus Extract: An Experimental Study in Rats

Journal: Current Pharmaceutical Analysis
Volume: 14 Issue: 0 Year: 2018 Page: 1-8
Author(s): Qi Wen,Hai-Long Li,Shi-Ying Mai,Feng Chen,Yin-Feng Tan

Research Article

A Novel In vitro Experimental System for the Evaluation of Enteric Drug Metabolism: Cofactor-Supplemented Permeabilized Cryopreserved Human Enterocytes (MetMax™ Cryopreserved Human Enterocytes)

Journal: Drug Metabolism Letters
Volume: 12 Issue: 2 Year: 2018 Page: 132-137
Author(s): Albert P. Li,Kirsten Amaral,Ming-Chih D. Ho

Review Article

UDP-glucuronosyltransferases: Structure, Function and Drug Design Studies

Journal: Current Medicinal Chemistry
Volume: 25 Issue: 2 Year: 2018 Page: 3247-3255
Author(s): Erica Candido Costa Mano,Luis Paulo Barbour Scott,Kathia M. Honorio

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